Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma' and Ligand = 'BDBM50324896'
TargetRetinoic acid receptor RXR-alpha/RXR-beta/RXR-gamma(Homo sapiens (Human))
Arizona State University

Curated by ChEMBL
LigandPNGBDBM50324896(6-[N-Ethyl(5,5,8,8-tetramethyl-5,6,7,8-tetrahydro-...)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human RXR binding domain and activation domain expressed in human HCT116 cells assessed as rexinoid activity incubated for 24 hrs...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed