Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-alpha' and Ligand = 'BDBM50129725'
TargetRetinoic acid receptor RXR-alpha(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50129725(7-(2-Butoxy-3,5-diisopropyl-phenyl)-3-methyl-octa-...)
Affinity DataEC50:  4nMAssay Description:Effective concentration for antagonistic activity against RXR-alpha expressed in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50129725(7-(2-Butoxy-3,5-diisopropyl-phenyl)-3-methyl-octa-...)
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against Retinoic acid receptor RXR-alpha antagonist was determined in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50129725(7-(2-Butoxy-3,5-diisopropyl-phenyl)-3-methyl-octa-...)
Affinity DataKi:  4nMAssay Description:Binding affinity against Retinoic acid receptor RXR-alpha was determined in vitro by using [3H]9-cis-RA as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50129725(7-(2-Butoxy-3,5-diisopropyl-phenyl)-3-methyl-octa-...)
Affinity DataKi:  4nMAssay Description:Ability to displace [3H]9-cis-RA from Retinoid X receptor alpha in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed