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Found 1 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor alpha' and Ligand = 'BDBM50244760'
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50244760((E)-4-{3-[3-Adamantan-1-yl-4-(2-methoxy-ethoxymeth...)
Affinity DataIC50:  4.47E+3nMAssay Description:Antagonist activity at Gal4-fused RARalpha (unknown origin) transfected in HEK293 cells assessed as inhibition of ATRA-induced transcriptional activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed