Affinity DataIC50: 20nMAssay Description:Antagonist activity of TTNPB (10 nM) function at retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataKd: 7nMAssay Description:Ability to displace 3[H]-(all-E)-retinoic acid (5 nM) from beta retinoic acid receptor (beta RAR) using transactivation assayMore data for this Ligand-Target Pair
Affinity DataKd: 7nMAssay Description:Ability to inhibit TTNPB-induced transactivation at retinoic acid receptor gammaMore data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Binding constant for baculovirus-expressed Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair