Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50005246'
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataIC50: 960nMAssay Description:Inhibition of [3H]dopamine uptake at dopamine transporter expressed in rat striatal homogenate after 5 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataKi:  24.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2012
Entry Details Article
PubMed
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataKi:  34nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataKi:  116nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2012
Entry Details
PubMed
TargetSodium-dependent dopamine transporter(Human)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataKi:  190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2012
Entry Details
PubMed
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataKi:  400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2012
Entry Details Article
PubMed
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataKi:  2.90E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2011
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
National Institute On Drug Abuse

Curated by PDSP Ki Database
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2012
Entry Details
PubMed