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Found 6 Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 1' and Ligand = 'BDBM50416487'
TargetSolute carrier family 22 member 1(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50416487(CHEMBL1236196 | TETRABUTYLAMMONIUM)
Affinity DataKi:  7.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier family 22 member 1(RAT)
University Of California

Curated by ChEMBL
LigandPNGBDBM50416487(CHEMBL1236196 | TETRABUTYLAMMONIUM)
Affinity DataKi:  1.70E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier family 22 member 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50416487(CHEMBL1236196 | TETRABUTYLAMMONIUM)
Affinity DataKi:  2.96E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier family 22 member 1(RAT)
University Of California

Curated by ChEMBL
LigandPNGBDBM50416487(CHEMBL1236196 | TETRABUTYLAMMONIUM)
Affinity DataIC50:  3.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
University Of California

Curated by ChEMBL
LigandPNGBDBM50416487(CHEMBL1236196 | TETRABUTYLAMMONIUM)
Affinity DataIC50:  7.90E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 50 uM) in OCT1-expressing MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50416487(CHEMBL1236196 | TETRABUTYLAMMONIUM)
Affinity DataIC50:  5.20E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in OCT1-expressing HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed