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Found 7 Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 1' and Ligand = 'BDBM50420192'
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£T

Curated by ChEMBL
LigandPNGBDBM50420192(CHEMBL2074851)
Affinity DataKi:  130nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£T

Curated by ChEMBL
LigandPNGBDBM50420192(CHEMBL2074851)
Affinity DataKi:  670nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£T

Curated by ChEMBL
LigandPNGBDBM50420192(CHEMBL2074851)
Affinity DataIC50:  400nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the presence of bicarbonate) (TEA: 20 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£T

Curated by ChEMBL
LigandPNGBDBM50420192(CHEMBL2074851)
Affinity DataIC50:  450nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (in the absence of bicarbonate) (TEA: 20 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£T

Curated by ChEMBL
LigandPNGBDBM50420192(CHEMBL2074851)
Affinity DataIC50:  510nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£T

Curated by ChEMBL
LigandPNGBDBM50420192(CHEMBL2074851)
Affinity DataIC50:  8.90E+4nMAssay Description:TP_TRANSPORTER: inhibition of Amantadine uptake (in the presence of bicarbonate) (Amantadine: 10 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
Bayerische Julius-Maximilians-Universit£T

Curated by ChEMBL
LigandPNGBDBM50420192(CHEMBL2074851)
Affinity DataIC50: >2.00E+5nMAssay Description:TP_TRANSPORTER: inhibition of Amantadine uptake (in the presence of bicarbonate) (Amantadine: 10 uM) in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed