TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical
Curated by PDSP Ki Database
Yamanouchi Pharmaceutical
Curated by PDSP Ki Database
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical
Curated by PDSP Ki Database
Yamanouchi Pharmaceutical
Curated by PDSP Ki Database
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Affinity DataKi: 1.36nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 mins by saturation binding assayMore data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Affinity DataKi: 1.48nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical
Curated by PDSP Ki Database
Yamanouchi Pharmaceutical
Curated by PDSP Ki Database
Affinity DataIC50: 3.30nMAssay Description:Tested for the inhibition to V2 subtype receptor using [3H]- (VS2) as radioligand at 3 nM and arginine-vasopressin at 2 microM in LLCPKI cellsMore data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Affinity DataIC50: 242nMAssay Description:Binding affinity to vasopression V2 receptor (unknown origin) on isolated cell membrane by vasopression-self competition binding assayMore data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute Of New Drug Research
Curated by PDSP Ki Database
Affinity DataEC50: 40nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Yamanouchi Pharmaceutical
Curated by PDSP Ki Database
Yamanouchi Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKd: 1.5nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat kidney Vasopressin V2 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.5nMAssay Description:Inhibition of radioligand [3H]AVP binding to V2 receptor in bovine kidney inner medulla membraneMore data for this Ligand-Target Pair