Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'cGMP-dependent protein kinase' and Ligand = 'BDBM50467123'
TargetcGMP-dependent protein kinase(malaria parasite P. falciparum)
Lifearc

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50467123BDBM50467123(CHEMBL4288103)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of Plasmodium falciparum protein kinase GMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(malaria parasite P. falciparum)
Lifearc

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50467123BDBM50467123(CHEMBL4288103)
Affinity DataIC50: 2nMAssay Description:Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(malaria parasite P. falciparum)
Lifearc

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50467123BDBM50467123(CHEMBL4288103)
Affinity DataIC50: 2nMAssay Description:Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed