Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'cGMP-dependent protein kinase 1' and Ligand = 'BDBM101618'
TargetcGMP-dependent protein kinase 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 101618BDBM101618(US8530652, 114)
Affinity DataKi:  15nMAssay Description:Inhibition of human PRKG1 assessed as inhibition constant in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetcGMP-dependent protein kinase 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 101618BDBM101618(US8530652, 114)
Affinity DataIC50: 34nMAssay Description:Inhibition of human PRKG1 in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetcGMP-dependent protein kinase 1(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 101618BDBM101618(US8530652, 114)
Affinity DataIC50: 3.37E+3nMAssay Description:Inhibition of human PRKG1 in presence of ATP by cellular assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed