Compile Data Set for Download or QSAR
Report error Found 3 of Enz. Inhib. data with enzyme = '17-beta-hydroxysteroid dehydrogenase type 1' and Substrate = '17beta-estradiol (E2)'
LigandPNGBDBM17290(EM1745 | E2-adenosine hybrid compound, 8 | [5-(6-a...)
Affinity DataKi:  3nM ΔG°:  -12.1kcal/molepH: 7.5 T: 2°CAssay Description:For steady-state kinetic study of hybrid inhibitors, a Fluorolog 3 instrument was used to monitor the fluorescent signal of NADPH formed during estra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2007
Entry Details Article
PubMed
LigandPNGBDBM17293([5-(6-amino-9H-purin-9-yl)-3,4-dihydroxyoxolan-2-y...)
Affinity DataKi:  2.50E+5nM ΔG°:  -5.11kcal/molepH: 7.5 T: 2°CAssay Description:For steady-state kinetic study of hybrid inhibitors, a Fluorolog 3 instrument was used to monitor the fluorescent signal of NADPH formed during estra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2007
Entry Details Article
PubMed
LigandPNGBDBM17294(Compound 11 | (13S,14S,15S)-15-methyl-13-nonyltetr...)
Affinity DatapH: 7.5 T: 2°CAssay Description:For steady-state kinetic study of hybrid inhibitors, a Fluorolog 3 instrument was used to monitor the fluorescent signal of NADPH formed during estra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2007
Entry Details Article
PubMed