Compile Data Set for Download or QSAR
Report error Found 1 of Enz. Inhib. data with enzyme = '3-phosphoinositide-dependent protein kinase 1' and Substrate = 'PDK1 Peptide Substrate'
Target3-phosphoinositide-dependent protein kinase 1(Human)
Berlex Biosciences

LigandChemical structure of BindingDB Monomer ID 17004BDBM17004([(3Z)-2-oxo-3-[1-(1H-pyrrol-2-yl)ethylidene]-2,3-d...)
Affinity DataIC50: 6nMAssay Description:PDK1 inhibitory activity is measured directly using PDK1, a peptide substrate, 33PATP, and compound followed by capture on P81 phospho-cellulose pape...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2007
Entry Details Article
PubMed