Compile Data Set for Download or QSAR
Report error Found 62 of Enz. Inhib. data with enzyme = '5-hydroxytryptamine receptor 1A' and Substrate = 'BDBM21393'
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29563(1-(m-trifluorophenyl)piperazine, 10)
Affinity DataKi:  0.300nM ΔG°:  -13.5kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29567(1-(m-trifluorophenyl)piperazine, 14)
Affinity DataKi:  1.30nM ΔG°:  -12.6kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29565(1-(m-trifluorophenyl)piperazine, 12)
Affinity DataKi:  1.5nM ΔG°:  -12.5kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  2.10nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29566(1-(m-trifluorophenyl)piperazine, 13)
Affinity DataKi:  2.20nM ΔG°:  -12.3kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29561(1-(m-trifluorophenyl)piperazine, 8)
Affinity DataKi:  2.60nM ΔG°:  -12.2kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29560(1-(m-trifluorophenyl)piperazine, 7)
Affinity DataKi:  3nM ΔG°:  -12.1kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29546(benzimidazolone scaffold, 15d)
Affinity DataKi:  3.40nM ΔG°:  -12.0kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21370(CHEMBL389718 | 6-[4-(2-acetylphenyl)piperazin-1-yl...)
Affinity DataKi:  3.85nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29557(1-(m-trifluorophenyl)piperazine, 4)
Affinity DataKi:  4nM ΔG°:  -11.9kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29558(1-(m-trifluorophenyl)piperazine, 5)
Affinity DataKi:  4nM ΔG°:  -11.9kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29562(1-(m-trifluorophenyl)piperazine, 9)
Affinity DataKi:  5.90nM ΔG°:  -11.7kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29548(benzimidazolone scaffold, 15f)
Affinity DataKi:  6nM ΔG°:  -11.7kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21368(CHEMBL224820 | 6-[4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  8.60nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29559(1-(m-trifluorophenyl)piperazine, 6)
Affinity DataKi:  9nM ΔG°:  -11.4kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29552(benzimidazolone scaffold, 15j)
Affinity DataKi:  12nM ΔG°:  -11.2kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21375(6-[4-(2-cyanophenyl)piperazin-1-yl]-N-(1,2,3,4-tet...)
Affinity DataKi:  16.6nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29556(1-(m-trifluorophenyl)piperazine, 3)
Affinity DataKi:  21nM ΔG°:  -10.9kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29540(benzimidazolone scaffold, 8h)
Affinity DataKi:  22nM ΔG°:  -10.9kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21371(CHEMBL225512 | 6-[4-(2-hydroxyphenyl)piperazin-1-y...)
Affinity DataKi:  24nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29544(benzimidazolone scaffold, 15b)
Affinity DataKi:  25nM ΔG°:  -10.8kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29541(benzimidazolone scaffold, 17d)
Affinity DataKi:  26nM ΔG°:  -10.8kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29545(benzimidazolone scaffold, 15c)
Affinity DataKi:  26nM ΔG°:  -10.8kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21389(6-[4-(2-fluorophenyl)piperazin-1-yl]-N-(1,2,3,4-te...)
Affinity DataKi:  29.2nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29550(benzimidazolone scaffold, 15h)
Affinity DataKi:  33nM ΔG°:  -10.6kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29564(1-(m-trifluorophenyl)piperazine, 11)
Affinity DataKi:  34nM ΔG°:  -10.6kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29542(benzimidazolone scaffold, 17f)
Affinity DataKi:  36nM ΔG°:  -10.6kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21390(6-[4-(pyridin-2-yl)piperazin-1-yl]-N-(1,2,3,4-tetr...)
Affinity DataKi:  36.4nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29551(benzimidazolone scaffold, 15i)
Affinity DataKi:  48nM ΔG°:  -10.4kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21367(CHEMBL225284 | 6-{4-[2-(methylsulfanyl)phenyl]pipe...)
Affinity DataKi:  52.7nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21380(6-[4-(2-butylphenyl)piperazin-1-yl]-N-(1,2,3,4-tet...)
Affinity DataKi:  60nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21383(6-[4-(2-phenylphenyl)piperazin-1-yl]-N-(1,2,3,4-te...)
Affinity DataKi:  60.9nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29553(benzimidazolone scaffold, 15k)
Affinity DataKi:  66nM ΔG°:  -10.2kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21378(6-[4-(2-ethylphenyl)piperazin-1-yl]-N-(1,2,3,4-tet...)
Affinity DataKi:  79.2nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29547(benzimidazolone scaffold, 15e)
Affinity DataKi:  84nM ΔG°:  -10.0kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21374(CHEMBL222477 | 6-[4-(2-chlorophenyl)piperazin-1-yl...)
Affinity DataKi:  96nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21384(6-{4-[2-(dimethylamino)phenyl]piperazin-1-yl}-N-(1...)
Affinity DataKi:  112nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21372(CHEMBL222188 | 6-(4-phenylpiperazin-1-yl)-N-(1,2,3...)
Affinity DataKi:  128nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21385(6-{4-[2-(methylamino)phenyl]piperazin-1-yl}-N-(1,2...)
Affinity DataKi:  133nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21381(6-{4-[2-(propan-2-yl)phenyl]piperazin-1-yl}-N-(1,2...)
Affinity DataKi:  167nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21379(6-[4-(2-propylphenyl)piperazin-1-yl]-N-(1,2,3,4-te...)
Affinity DataKi:  168nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29537(benzimidazolone scaffold, 8e)
Affinity DataKi:  168nM ΔG°:  -9.61kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29539(benzimidazolone scaffold, 8g)
Affinity DataKi:  182nM ΔG°:  -9.56kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21373(6-[4-(2-nitrophenyl)piperazin-1-yl]-N-(1,2,3,4-tet...)
Affinity DataKi:  183nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21391(1-oxido-2-{4-[5-(1,2,3,4-tetrahydronaphthalen-1-yl...)
Affinity DataKi:  194nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29549(benzimidazolone scaffold, 15g)
Affinity DataKi:  269nM ΔG°:  -9.32kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universita Degli Studi Di Bari

LigandPNGBDBM21369(CHEMBL222755 | 6-[4-(2-methylphenyl)piperazin-1-yl...)
Affinity DataKi:  279nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29536(benzimidazolone scaffold, 8d)
Affinity DataKi:  340nM ΔG°:  -9.17kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29538(benzimidazolone scaffold, 8f)
Affinity DataKi:  375nM ΔG°:  -9.11kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Polish Academy of Sciences

LigandPNGBDBM29543(benzimidazolone scaffold, 15a)
Affinity DataKi:  392nM ΔG°:  -9.09kcal/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein and test compounds. After incubation, the reaction stopped b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/7/2009
Entry Details Article
PubMed
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