Compile Data Set for Download or QSAR
Report error Found 29 of Enz. Inhib. data with enzyme = 'Adenosine receptor A2a' and Substrate = 'BDBM21241'
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21220BDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataKi:  16nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21229BDBM21229(N-[6-propoxy-2-(propylsulfanyl)pyrimidin-4-yl]prop...)
Affinity DataKi:  71nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21173BDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  337nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
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Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21225BDBM21225(N-[2-(methylsulfanyl)-6-propoxypyrimidin-4-yl]prop...)
Affinity DataKi:  398nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21221BDBM21221(2-Cl-IB-MECA | CHEMBL431733 | C-IBzA-MU | 2-chloro...)
Affinity DataKi:  401nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
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Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21215BDBM21215(2-(1H-benzimidazol-2-yl)quinoxaline | 2-(1H-1,3-be...)
Affinity DataKi:  561nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21217BDBM21217(2-(4-methyl-1H-1,3-benzodiazol-2-yl)quinoxaline | ...)
Affinity DataKi:  833nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21224BDBM21224(N-[2-(methylsulfanyl)-6-propoxypyrimidin-4-yl]acet...)
Affinity DataKi:  1.12E+3nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21216BDBM21216(2-[4-(ethylsulfanyl)-1H-1,3-benzodiazol-2-yl]quino...)
Affinity DataKi:  3.44E+3nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21232BDBM21232(N-{6-[(2-chlorophenyl)methoxy]-2-(propylsulfanyl)p...)
Affinity DataKi:  4.15E+3nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21213BDBM21213(2-[5-(pyridin-2-yl)-4H-1,2,4-triazol-3-yl]pyridine...)
Affinity DataKi: >1.00E+4nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21214BDBM21214(3-(3-chloro-1H-pyrazol-5-yl)-1,2-dihydroquinoxalin...)
Affinity DataKi: >1.00E+4nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21218BDBM21218(CHEMBL200480 | 4,9,14-trimethyl-3,5,8,10,13,15-hex...)
Affinity DataKi: >1.00E+4nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21219BDBM21219(7-methyl-6,7-dihydro[1,3]thiazolo[3,2-a][1,2,3]tri...)
Affinity DataKi: >1.00E+4nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21222BDBM21222(N-[6-methoxy-2-(methylsulfanyl)pyrimidin-4-yl]acet...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21223BDBM21223(N-[6-methoxy-2-(methylsulfanyl)pyrimidin-4-yl]prop...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21226BDBM21226(N-[6-methoxy-2-(propylsulfanyl)pyrimidin-4-yl]acet...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21227BDBM21227(N-[6-methoxy-2-(propylsulfanyl)pyrimidin-4-yl]prop...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21228BDBM21228(N-[6-propoxy-2-(propylsulfanyl)pyrimidin-4-yl]acet...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21230BDBM21230(N-[2-(benzylsulfanyl)-6-propoxypyrimidin-4-yl]acet...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21231BDBM21231(N-[6-(benzyloxy)-2-(propylsulfanyl)pyrimidin-4-yl]...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21233BDBM21233(N-{6-[(3-chlorophenyl)methoxy]-2-(propylsulfanyl)p...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21234BDBM21234(N-{6-[(4-chlorophenyl)methoxy]-2-(propylsulfanyl)p...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21235BDBM21235(N-{6-[(2,4-dichlorophenyl)methoxy]-2-(propylsulfan...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21236BDBM21236(N-{6-[(4-methoxyphenyl)methoxy]-2-(propylsulfanyl)...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21237BDBM21237(N-[6-(2-phenylethoxy)-2-(propylsulfanyl)pyrimidin-...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21238BDBM21238(N-[6-(cyclohexylmethoxy)-2-(propylsulfanyl)pyrimid...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21239BDBM21239(N-{6-[(4-chlorophenyl)methoxy]-2-(ethylsulfanyl)py...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Napoli

LigandChemical structure of BindingDB Monomer ID 21240BDBM21240(N-[2-(tert-butylsulfanyl)-6-[(4-chlorophenyl)metho...)
Affinity DataAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2008
Entry Details Article
PubMed