Compile Data Set for Download or QSAR
Report error Found 7 of Enz. Inhib. data with enzyme = 'Adenosine receptor A3' and Substrate = 'BDBM10852'
TargetAdenosine receptor A3(Human)
Vernalis (R&D)

LigandPNGBDBM35829(pyrimidine-4-carboxamide, 111)
Affinity DataKi:  366nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Vernalis (R&D)

LigandPNGBDBM35837(pyrimidine-4-carboxamide, 119)
Affinity DataKi:  741nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Vernalis (R&D)

LigandPNGBDBM35786(pyrimidine-4-carboxamide, 27)
Affinity DataKi:  896nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Vernalis (R&D)

LigandPNGBDBM35833(pyrimidine-4-carboxamide, 115)
Affinity DataKi:  1.15E+3nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Vernalis (R&D)

LigandPNGBDBM35839(pyrimidine-4-carboxamide, 121)
Affinity DataKi:  1.63E+3nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Vernalis (R&D)

LigandPNGBDBM35836(pyrimidine-4-carboxamide, 118)
Affinity DataKi:  2.10E+3nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Vernalis (R&D)

LigandPNGBDBM35834(pyrimidine-4-carboxamide, 116)
Affinity DataKi:  9.09E+3nMAssay Description:Binding assays were performed in a total volume of 250 uL, containing radioligand, membranes and test compounds. Following 60 (A2B, A3) or 90 (A1, A2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed