Compile Data Set for Download or QSAR
Report error Found 4 of Enz. Inhib. data with enzyme = 'Alpha-2A adrenergic receptor [16-465]' and Substrate = 'BDBM14062'
TargetAlpha-2A adrenergic receptor [16-465](Rat)
University of Queensland

LigandPNGBDBM13014(7,8-Dichloro-1,2,3,4-tetrahydro-isoquinoline; hydr...)
Affinity DataKi:  21nM ΔG°:  -10.5kcal/molepH: 7.7 T: 2°CAssay Description:The binding affinity of compound was evaluated using [3H] Clonidine as ligand in competition binding experiments. Nonspecific binding was determined ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2007
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
University of Queensland

LigandPNGBDBM14060(CHEMBL26828 | 7-Iodo-1,2,3,4-tetrahydroisoquinolin...)
Affinity DataKi:  220nM ΔG°:  -9.08kcal/molepH: 7.7 T: 2°CAssay Description:The binding affinity of compound was evaluated using [3H] Clonidine as ligand in competition binding experiments. Nonspecific binding was determined ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2007
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
University of Queensland

LigandPNGBDBM14061(8,9-Dichloro-2,3,4,5-tetrahydro-1H-2-benzazepine |...)
Affinity DataKi:  4.50E+3nM ΔG°:  -7.29kcal/molepH: 7.7 T: 2°CAssay Description:The binding affinity of compound was evaluated using [3H] Clonidine as ligand in competition binding experiments. Nonspecific binding was determined ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2007
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor [16-465](Rat)
University of Queensland

LigandPNGBDBM13017(1,2,3,4-tetrahydroisoquinoline-7-sulfonamide | CHE...)
Affinity DataKi:  1.00E+5nM ΔG°:  -5.45kcal/molepH: 7.7 T: 2°CAssay Description:The binding affinity of compound was evaluated using [3H] Clonidine as ligand in competition binding experiments. Nonspecific binding was determined ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2007
Entry Details Article
PubMed