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Report error Found 93 of Enz. Inhib. data with enzyme = 'Amine oxidase [flavin-containing] B' and Substrate = 'BDBM10990'
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11014((-)-(S)1 | (5S)-5-(4-chlorophenyl)-3-(4-methylphen...)
Affinity DataKi:  1nM ΔG°:  -12.8kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11004(5-(4-chlorophenyl)-3-(4-methylphenyl)-4,5-dihydro-...)
Affinity DataKi:  1.5nM ΔG°:  -12.6kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11015((5R)-5-(4-chlorophenyl)-3-(4-methylphenyl)-4,5-dih...)
Affinity DataKi:  2.70nM ΔG°:  -12.2kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86779(Phthalonitrile analogue, 4h)
Affinity DataIC50: 4.80nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11010(5-(4-chlorophenyl)-3-(thiophen-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  6nM ΔG°:  -11.7kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86776(Phthalonitrile analogue, 4e)
Affinity DataIC50: 6.60nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86773(Phthalonitrile analogue, 4b)
Affinity DataIC50: 7.90nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11005(3,5-bis(4-methylphenyl)-4,5-dihydro-1H-pyrazole-1-...)
Affinity DataKi:  10nM ΔG°:  -11.4kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11011(5-(4-methylphenyl)-3-(thiophen-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  10nM ΔG°:  -11.4kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86774(Phthalonitrile analogue, 4c)
Affinity DataIC50: 18nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15592(N-Methyl,N-(benzyl),N-(pyrrol-2-ylmethyl)amine | C...)
Affinity DataKi:  20nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15611(N-Methyl,N-(propargyl),N-(pyrrol-2-ylmethyl)amine ...)
Affinity DataKi:  20nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11012(5-(furan-2-yl)-3-(thiophen-2-yl)-4,5-dihydro-1H-py...)
Affinity DataKi:  20nM ΔG°:  -11.0kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15604(N-[(1R)-1-cyclohexylethyl]-N-methyl-1H-pyrrole-2-c...)
Affinity DataKi:  30nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86786(Benzonitrile analogue, 5f)
Affinity DataIC50: 41nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11008(3-(4-fluorophenyl)-5-(4-methylphenyl)-4,5-dihydro-...)
Affinity DataKi:  50nM ΔG°:  -10.4kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11013(3,5-bis(thiophen-2-yl)-4,5-dihydro-1H-pyrazole-1-c...)
Affinity DataKi:  50nM ΔG°:  -10.4kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
University of Bari

LigandPNGBDBM19183(3-(3-nitrophenyl)-4aH,9H,9aH-indeno[1,2-e][1,2,4]t...)
Affinity DataIC50: 80nMAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15586(N-methyl-N-(2-phenylethyl)-1H-pyrrole-2-carboxamid...)
Affinity DataKi:  120nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86775(Phthalonitrile analogue, 4d)
Affinity DataIC50: 136nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11006(5-(furan-2-yl)-3-(4-methylphenyl)-4,5-dihydro-1H-p...)
Affinity DataKi:  170nM ΔG°:  -9.63kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86784(Benzonitrile analogue, 5d)
Affinity DataIC50: 174nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86780(Phthalonitrile analogue, 4i)
Affinity DataIC50: 226nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86777(Phthalonitrile analogue, 4f)
Affinity DataIC50: 244nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86782(Benzonitrile analogue, 5b)
Affinity DataIC50: 249nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86785(Benzonitrile analogue, 5e)
Affinity DataIC50: 266nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11009(3-(4-fluorophenyl)-5-(furan-2-yl)-4,5-dihydro-1H-p...)
Affinity DataKi:  370nM ΔG°:  -9.15kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86783(Benzonitrile analogue, 5c)
Affinity DataIC50: 379nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86778(Phthalonitrile analogue, 4g)
Affinity DataIC50: 568nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15610(N-(Propargyl),N-(pyrrol-2-ylmethyl)amine | prop-2-...)
Affinity DataKi:  620nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15595((2-phenylethyl)(1H-pyrrol-2-ylmethyl)amine | N-(2-...)
Affinity DataKi:  700nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86781(Benzonitrile analogue, 5a)
Affinity DataIC50: 785nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
University of Bari

LigandPNGBDBM19184(3-(3-nitrophenyl)-4aH,5H,9bH-indeno[2,1-e][1,2,4]t...)
Affinity DataIC50: 912nMAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataKi:  970nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11007(5-(4-chlorophenyl)-3-(4-fluorophenyl)-4,5-dihydro-...)
Affinity DataKi:  1.00E+3nM ΔG°:  -8.54kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86790(Benzyl phenyl ether analogue, 6b)
Affinity DataIC50: 1.32E+3nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86787(Benzonitrile analogue, 5g)
Affinity DataIC50: 1.35E+3nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86788(Benzonitrile analogue, 5h)
Affinity DataIC50: 1.39E+3nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11017((5R)-5-(4-chlorophenyl)-3-(4-fluorophenyl)-4,5-dih...)
Affinity DataKi:  1.40E+3nM ΔG°:  -8.33kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15601(methyl(1-phenylethyl)(1H-pyrrol-2-ylmethyl)amine |...)
Affinity DataKi:  1.50E+3nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
University of Bari

LigandPNGBDBM19168(3-(4-fluorophenoxymethyl)-5H-indeno[1,2-c]pyridazi...)
Affinity DataIC50: 1.90E+3nMAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15597(N-Methyl,N-(3-phenylpropyl),N-(pyrrol-2-ylmethyl)a...)
Affinity DataKi:  2.00E+3nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11016((5S)-5-(4-chlorophenyl)-3-(4-fluorophenyl)-4,5-dih...)
Affinity DataKi:  2.40E+3nM ΔG°:  -8.00kcal/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15590(N-methyl-N-(4-phenylbutyl)-1H-pyrrole-2-carboxamid...)
Affinity DataKi:  2.50E+3nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15598(methyl(4-phenylbutyl)(1H-pyrrol-2-ylmethyl)amine |...)
Affinity DataKi:  2.50E+3nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
University of Bari

LigandPNGBDBM19167(3-(phenoxymethyl)-5H-indeno[1,2-c]pyridazin-5-one ...)
Affinity DataIC50: 2.51E+3nMAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
North-West University

LigandPNGBDBM86791(Benzyl phenyl ether analogue, 6c)
Affinity DataIC50: 3.05E+3nMpH: 7.4 T: 2°CAssay Description:MAO inhibition potencies of phthalonitrile, benzonitrile and benzyl phenyl ether analogs, recombinant human MAO-A and -B were employed as enzyme sour...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15603(N-[(1S)-1-cyclohexylethyl]-1H-pyrrole-2-carboxamid...)
Affinity DataKi:  3.50E+3nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15602(N-[(1R)-1-cyclohexylethyl]-1H-pyrrole-2-carboxamid...)
Affinity DataKi:  3.60E+3nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM15605(N-[(1S)-1-cyclohexylethyl]-N-methyl-1H-pyrrole-2-c...)
Affinity DataKi:  4.10E+3nMAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kinuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2007
Entry Details Article
PubMed
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