Compile Data Set for Download or QSAR
Report error Found 11 of Enz. Inhib. data with enzyme = 'Androgen receptor' and Substrate = 'SRC2-3 peptide'
TargetAndrogen receptor(Human)
St. Jude Research Hospital

LigandChemical structure of BindingDB Monomer ID 35910BDBM35910(flufenamic acid analogue, 36)
Affinity DataEC50:  3.00E+4nMpH: 7.2 T: 2°CAssay Description:AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
St. Jude Research Hospital

LigandChemical structure of BindingDB Monomer ID 35911BDBM35911(flufenamic acid analogue, 37)
Affinity DataEC50:  3.90E+4nMpH: 7.2 T: 2°CAssay Description:AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
St. Jude Research Hospital

LigandChemical structure of BindingDB Monomer ID 35912BDBM35912(flufenamic acid analogue, 38)
Affinity DataEC50:  4.25E+4nMpH: 7.2 T: 2°CAssay Description:AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
St. Jude Research Hospital

LigandChemical structure of BindingDB Monomer ID 35913BDBM35913(flufenamic acid analogue, 39)
Affinity DataEC50:  4.85E+4nMpH: 7.2 T: 2°CAssay Description:AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
St. Jude Research Hospital

LigandChemical structure of BindingDB Monomer ID 35914BDBM35914(flufenamic acid analogue, 40)
Affinity DataEC50:  5.40E+4nMAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
St. Jude Research Hospital

LigandChemical structure of BindingDB Monomer ID 35908BDBM35908(flufenamic acid analogue, 41 | flufenamic acid ana...)
Affinity DataEC50:  5.60E+4nMAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
St. Jude Research Hospital

LigandChemical structure of BindingDB Monomer ID 35916BDBM35916(flufenamic acid analogue, 42)
Affinity DataEC50:  6.40E+4nMAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
St. Jude Research Hospital

LigandChemical structure of BindingDB Monomer ID 17636BDBM17636(2-{[3-(trifluoromethyl)phenyl]amino}benzoic acid |...)
Affinity DataEC50:  6.70E+4nMAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Human)
St. Jude Research Hospital

LigandChemical structure of BindingDB Monomer ID 35917BDBM35917(flufenamic acid analogue, 43)
Affinity DataEC50:  7.55E+4nMAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
St. Jude Research Hospital

LigandChemical structure of BindingDB Monomer ID 35918BDBM35918(flufenamic acid analogue, 44)
Affinity DataEC50:  8.30E+4nMAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
St. Jude Research Hospital

LigandChemical structure of BindingDB Monomer ID 35919BDBM35919(flufenamic acid analogue, 45)
Affinity DataEC50:  9.30E+4nMAssay Description:A radiolabeled ligand competition scintillation proximity assay (SPA) for the androgen receptor (AR) using Ni-coated 384-well FlashPlates. It measure...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2009
Entry Details Article
PubMed