Compile Data Set for Download or QSAR
Report error Found 16 of Enz. Inhib. data with enzyme = 'Angiopoietin-1 receptor' and Substrate = 'poly-Glu-Ala-Tyr'
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8800BDBM8800(N-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)cyclohe...)
Affinity DataIC50: 137nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8808BDBM8808(3-{4-[(1H-indol-2-ylmethyl)amino]phenyl}-1-[4-(4-m...)
Affinity DataIC50: 203nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8793BDBM8793(CHEMBL45177 | 7-[4-(4-methylpiperazin-1-yl)cyclohe...)
Affinity DataIC50: 250nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8806BDBM8806((1R,2R)-N-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl...)
Affinity DataIC50: 275nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8798BDBM8798(CHEMBL47787 | benzyl N-(4-{4-amino-1-[4-(4-methylp...)
Affinity DataIC50: 521nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8795BDBM8795(1-[4-(4-methylpiperazin-1-yl)cyclohexyl]-3-[4-(phe...)
Affinity DataIC50: 606nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8794BDBM8794(1-[4-(4-methylpiperazin-1-yl)cyclohexyl]-3-(4-phen...)
Affinity DataIC50: 750nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8801BDBM8801([(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)cyclohex...)
Affinity DataIC50: 888nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8805BDBM8805(N-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)cyclohe...)
Affinity DataIC50: 910nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8799BDBM8799(3-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)cyclohe...)
Affinity DataIC50: 933nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8807BDBM8807(N-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)cyclohe...)
Affinity DataIC50: 1.02E+3nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8802BDBM8802(3-[4-(benzylamino)-3-methoxyphenyl]-1-[4-(4-methyl...)
Affinity DataIC50: 1.13E+3nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8804BDBM8804(N-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)cyclohe...)
Affinity DataIC50: 1.44E+3nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8803BDBM8803(N-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)cyclohe...)
Affinity DataIC50: 2.45E+3nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8797BDBM8797(N-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)cyclohe...)
Affinity DataIC50: 4.68E+3nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Abbott Bioresearch Center

LigandChemical structure of BindingDB Monomer ID 8796BDBM8796(3-(4-benzoylphenyl)-1-[4-(4-methylpiperazin-1-yl)c...)
Affinity DataIC50: 5.73E+3nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2006
Entry Details Article
PubMed