Compile Data Set for Download or QSAR
Report error Found 25 of Enz. Inhib. data with enzyme = 'Aryl hydrocarbon receptor' and Substrate = 'BDBM23927'
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23936BDBM23936(1,3-dichloro-5-[(E)-2-[4-(trifluoromethyl)phenyl]e...)
Affinity DataKi:  0.200nM ΔG°:  -12.3kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
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Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23929BDBM23929(1,3-dichloro-5-[(E)-2-(4-chlorophenyl)ethenyl]benz...)
Affinity DataKi:  1.20nM ΔG°:  -11.3kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
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Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23937BDBM23937(1,3-dichloro-5-[(E)-2-(4-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  1.40nM ΔG°:  -11.2kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
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Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23932BDBM23932(1,3-bis(trifluoromethyl)-5-[(E)-2-[4-(trifluoromet...)
Affinity DataKi:  2.10nM ΔG°:  -11.0kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23933BDBM23933(1-[(E)-2-(4-fluorophenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  3.10nM ΔG°:  -10.8kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23931BDBM23931(1,3-difluoro-5-[(E)-2-(4-fluorophenyl)ethenyl]benz...)
Affinity DataKi:  3.80nM ΔG°:  -10.7kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23934BDBM23934(1-[(E)-2-(4-ethoxyphenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  5nM ΔG°:  -10.5kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23939BDBM23939(1,3-dichloro-5-[(E)-2-(3-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  5.70nM ΔG°:  -10.4kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23938BDBM23938(1,3-dichloro-5-[(E)-2-[3-(trifluoromethyl)phenyl]e...)
Affinity DataKi:  6.80nM ΔG°:  -10.4kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23928BDBM23928(CHEMBL296411 | 1,3-dimethoxy-5-[(E)-2-(4-methoxyph...)
Affinity DataKi:  7.70nM ΔG°:  -10.3kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23930BDBM23930(1,3-difluoro-5-[(E)-2-(4-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  9.20nM ΔG°:  -10.2kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23949BDBM23949(1,3-dichloro-5-[(Z)-2-(4-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  12nM ΔG°:  -10.0kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23941BDBM23941(1,3-dichloro-5-[(Z)-2-(4-chlorophenyl)ethenyl]benz...)
Affinity DataKi:  13nM ΔG°:  -9.99kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23948BDBM23948(1,3-dichloro-5-[(Z)-2-[4-(trifluoromethyl)phenyl]e...)
Affinity DataKi:  14nM ΔG°:  -9.95kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23950BDBM23950(1,3-dichloro-5-[(Z)-2-[3-(trifluoromethyl)phenyl]e...)
Affinity DataKi:  19nM ΔG°:  -9.78kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23935BDBM23935(1-[(E)-2-(4-butoxyphenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  20nM ΔG°:  -9.76kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23942BDBM23942(1,3-difluoro-5-[(Z)-2-(4-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  22nM ΔG°:  -9.70kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23951BDBM23951(1,3-dichloro-5-[(Z)-2-(3-methoxyphenyl)ethenyl]ben...)
Affinity DataKi:  24nM ΔG°:  -9.66kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23947BDBM23947(1-[(Z)-2-(4-butoxyphenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  43nM ΔG°:  -9.34kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23944BDBM23944(1,3-bis(trifluoromethyl)-5-[(Z)-2-[4-(trifluoromet...)
Affinity DataKi:  60nM ΔG°:  -9.15kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23943BDBM23943(1,3-difluoro-5-[(Z)-2-(4-fluorophenyl)ethenyl]benz...)
Affinity DataKi:  63nM ΔG°:  -9.12kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23946BDBM23946(1-[(Z)-2-(4-ethoxyphenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  65nM ΔG°:  -9.11kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23940BDBM23940(1,3-dimethoxy-5-[(Z)-2-(4-methoxyphenyl)ethenyl]be...)
Affinity DataKi:  75nM ΔG°:  -9.03kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23945BDBM23945(1-[(Z)-2-(4-fluorophenyl)ethenyl]-3,5-dimethoxyben...)
Affinity DataKi:  96nM ΔG°:  -8.89kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed
TargetAryl hydrocarbon receptor(Rabbit)
Institut Claudius Regaud

LigandChemical structure of BindingDB Monomer ID 23926BDBM23926(5-[(E)-2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol...)
Affinity DataKi:  169nM ΔG°:  -8.58kcal/molepH: 7.6 T: 2°CAssay Description:Cytosols from rabbit liver were incubated with [3H]-TCDD and 12 concentrations of unlabeled test ligands. IC50 values were determined using the itera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2008
Entry Details Article
PubMed