Compile Data Set for Download or QSAR
Report error Found 7 of Enz. Inhib. data with enzyme = 'Beta-2 adrenergic receptor' and Substrate = 'BDBM25393'
TargetBeta-2 adrenergic receptor(Human)
Monash University

LigandChemical structure of BindingDB Monomer ID 25392BDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataKi:  136nM ΔG°:  -9.27kcal/molepH: 7.4 T: 2°CAssay Description:The displacement of [125I]-(-)iodopindolol binding from the beta2AR was determined using DDT1 MF-2 cell membranes. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2008
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Monash University

LigandChemical structure of BindingDB Monomer ID 25398BDBM25398(N-[5-(2-{[6-({9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hy...)
Affinity DataKi:  311nM ΔG°:  -8.78kcal/molepH: 7.4 T: 2°CAssay Description:The displacement of [125I]-(-)iodopindolol binding from the beta2AR was determined using DDT1 MF-2 cell membranes. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2008
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Monash University

LigandChemical structure of BindingDB Monomer ID 25396BDBM25396(N-[5-(2-{[4-({9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hy...)
Affinity DataKi:  863nM ΔG°:  -8.18kcal/molepH: 7.4 T: 2°CAssay Description:The displacement of [125I]-(-)iodopindolol binding from the beta2AR was determined using DDT1 MF-2 cell membranes. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2008
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Monash University

LigandChemical structure of BindingDB Monomer ID 25399BDBM25399(N-[5-(1-{9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxy...)
Affinity DataKi:  2.30E+3nM ΔG°:  -7.61kcal/molepH: 7.4 T: 2°CAssay Description:The displacement of [125I]-(-)iodopindolol binding from the beta2AR was determined using DDT1 MF-2 cell membranes. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2008
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Monash University

LigandChemical structure of BindingDB Monomer ID 25397BDBM25397((2R,3R,4S,5R)-2-{6-[(4-{[2-(3-amino-4-hydroxypheny...)
Affinity DataKi:  4.31E+3nM ΔG°:  -7.24kcal/molepH: 7.4 T: 2°CAssay Description:The displacement of [125I]-(-)iodopindolol binding from the beta2AR was determined using DDT1 MF-2 cell membranes. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2008
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Monash University

LigandChemical structure of BindingDB Monomer ID 25394BDBM25394(N-[5-(2-{[2-({9-[(2R,3R,4S,5R)-3,4-dihydroxy-5-(hy...)
Affinity DataKi: >1.00E+4nM ΔG°: >-6.75kcal/molepH: 7.4 T: 2°CAssay Description:The displacement of [125I]-(-)iodopindolol binding from the beta2AR was determined using DDT1 MF-2 cell membranes. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2008
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Monash University

LigandChemical structure of BindingDB Monomer ID 25395BDBM25395((2R,3R,4S,5R)-2-{6-[(2-{[2-(3-amino-4-hydroxypheny...)
Affinity DataKi: >1.00E+4nM ΔG°: >-6.75kcal/molepH: 7.4 T: 2°CAssay Description:The displacement of [125I]-(-)iodopindolol binding from the beta2AR was determined using DDT1 MF-2 cell membranes. Nonspecific binding was determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2008
Entry Details Article
PubMed