Compile Data Set for Download or QSAR
Report error Found 109 of Enz. Inhib. data with enzyme = 'Cannabinoid receptor 1' and Substrate = 'BDBM21244'
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21279(N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iod...)
Affinity DataKi:  2.30nMAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21263(N-cyclohexyl-1-(3,4-dichlorophenyl)-4-methyl-5-(1H...)
Affinity DataKi:  5.60nM ΔG°:  -11.4kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM29079(cyclopropanolamide, 12a | racemic | cyclopropanola...)
Affinity DataKi:  11nM ΔG°:  -11.0kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM22988(Arachidonoyl ethanolamide | Arachidonoylethanolami...)
Affinity DataKi:  11nM ΔG°:  -11.0kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  12nMAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21284(1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopr...)
Affinity DataKi:  12nM ΔG°:  -11.0kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21290(6-bromo-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethy...)
Affinity DataKi:  13nM ΔG°:  -10.9kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  13.3nM ΔG°:  -10.9kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM29078(cyclopropanolamide, 13a | racemic | cyclopropanola...)
Affinity DataKi:  14nM ΔG°:  -10.9kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21289(6-chloro-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetrameth...)
Affinity DataKi:  14nM ΔG°:  -10.9kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21266(N-cyclohexyl-1-(3,4-dichlorophenyl)-5-(2,5-dimethy...)
Affinity DataKi:  14nM ΔG°:  -10.9kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM29087(cyclopropanolamide, 14a)
Affinity DataKi:  20nM ΔG°:  -10.7kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21333(methyl 1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethyl...)
Affinity DataKi:  25nMAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM29078(cyclopropanolamide, 13a | racemic | cyclopropanola...)
Affinity DataKi:  27nM ΔG°:  -10.5kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21277(N-cyclohexyl-5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-met...)
Affinity DataKi:  28nMAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM29088(cyclopropanolamide, 11a)
Affinity DataKi:  28nM ΔG°:  -10.5kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21264(1-(3,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1...)
Affinity DataKi:  28nM ΔG°:  -10.5kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21291(6-methyl-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetrameth...)
Affinity DataKi:  28nM ΔG°:  -10.5kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21309(5-(oxan-4-ylmethyl)-7-[(2,2,3,3-tetramethylcyclopr...)
Affinity DataKi:  28nM ΔG°:  -10.5kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21259(1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)meth...)
Affinity DataKi:  28nM ΔG°:  -10.5kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21261(1-(3,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)...)
Affinity DataKi:  30nM ΔG°:  -10.4kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21331(1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopr...)
Affinity DataKi:  31nMAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM29079(cyclopropanolamide, 12a | racemic | cyclopropanola...)
Affinity DataKi:  32nM ΔG°:  -10.4kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21304(6-(benzyloxy)-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetr...)
Affinity DataKi:  33nM ΔG°:  -10.4kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21262(1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)meth...)
Affinity DataKi:  35nM ΔG°:  -10.3kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21272(N-[(3,4-dichlorophenyl)methyl]-1-(2,4-difluorophen...)
Affinity DataKi:  35nM ΔG°:  -10.3kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21273(N-cyclohexyl-1-(2,4-difluorophenyl)-5-(2,5-dimethy...)
Affinity DataKi:  35nM ΔG°:  -10.3kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21256(1-(2,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)meth...)
Affinity DataKi:  37nM ΔG°:  -10.3kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21258(1-(2,4-dichlorophenyl)-5-(2,5-dimethyl-1H-pyrrol-1...)
Affinity DataKi:  38nM ΔG°:  -10.3kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21300(6-methoxy-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramet...)
Affinity DataKi:  40nM ΔG°:  -10.3kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21260(N-cyclohexyl-1-(2,4-dichlorophenyl)-5-(2,5-dimethy...)
Affinity DataKi:  42nM ΔG°:  -10.2kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21301(7-methoxy-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramet...)
Affinity DataKi:  45nM ΔG°:  -10.2kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21257(N-cyclohexyl-1-(2,4-dichlorophenyl)-4-methyl-5-(1H...)
Affinity DataKi:  56nM ΔG°:  -10.1kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21285(4,5,6,7-tetrafluoro-1-(oxan-4-ylmethyl)-3-[(2,2,3,...)
Affinity DataKi:  66nM ΔG°:  -9.95kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21292(1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopr...)
Affinity DataKi:  70nM ΔG°:  -9.92kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21276(5-(2,5-dimethyl-1H-pyrrol-1-yl)-4-methyl-N-(piperi...)
Affinity DataKi:  110nMAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21250(1-(4-chlorophenyl)-4-methyl-N-(piperidin-1-yl)-5-(...)
Affinity DataKi:  110nM ΔG°:  -9.65kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21251(1-(4-chlorophenyl)-N-(cyclohexylmethyl)-4-methyl-5...)
Affinity DataKi:  110nM ΔG°:  -9.65kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
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Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21295(1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopr...)
Affinity DataKi:  204nM ΔG°:  -9.27kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
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Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21334(1-(oxan-4-ylmethyl)-6-phenyl-3-[(2,2,3,3-tetrameth...)
Affinity DataKi:  228nMAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21303(5-(benzyloxy)-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetr...)
Affinity DataKi:  238nM ΔG°:  -9.18kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
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Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21297(1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopr...)
Affinity DataKi:  246nM ΔG°:  -9.16kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
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Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21247(4-cyano-N-[(3,4-dichlorophenyl)methyl]-1-phenyl-5-...)
Affinity DataKi:  280nM ΔG°:  -9.08kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
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Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21249(1-(4-chlorophenyl)-N-cyclohexyl-5-(1H-pyrrol-1-yl)...)
Affinity DataKi:  280nM ΔG°:  -9.08kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21265(1-(3,4-dichlorophenyl)-N-[(3,4-dichlorophenyl)meth...)
Affinity DataKi:  280nM ΔG°:  -9.08kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21275(N-[(3,4-dichlorophenyl)methyl]-4-methyl-5-(1H-pyrr...)
Affinity DataKi:  280nMAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21299(5-methoxy-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramet...)
Affinity DataKi:  282nM ΔG°:  -9.08kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21294(1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopr...)
Affinity DataKi:  388nM ΔG°:  -8.89kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21308(1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetramethylcyclopr...)
Affinity DataKi:  395nM ΔG°:  -8.88kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
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Date in BDB:
4/7/2008
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Sapienza University of Rome

LigandPNGBDBM21287(5-chloro-1-(oxan-4-ylmethyl)-3-[(2,2,3,3-tetrameth...)
Affinity DataKi:  512nM ΔG°:  -8.72kcal/molepH: 7.4 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibition c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2008
Entry Details Article
PubMed
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