Compile Data Set for Download or QSAR
Report error Found 10 of Enz. Inhib. data with enzyme = 'Cannabinoid receptor 2' and Substrate = 'BDBM21278'
TargetCannabinoid receptor 2(Human)
Acadia Pharmaceuticals

LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  398nM ΔG°:  -8.64kcal/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Acadia Pharmaceuticals

LigandPNGBDBM29100(dibenzothiazepine, 12h)
Affinity DataKi:  1.00E+3nM ΔG°:  -8.10kcal/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Acadia Pharmaceuticals

LigandPNGBDBM29097(dibenzothiazepine, 12c)
Affinity DataKi:  1.26E+3nM ΔG°:  -7.96kcal/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Acadia Pharmaceuticals

LigandPNGBDBM29094(3-(4-chlorophenyl)-N''''-(4-chlorophenylsulfonyl)-...)
Affinity DataKi:  2.00E+3nM ΔG°:  -7.69kcal/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Acadia Pharmaceuticals

LigandPNGBDBM29099(dibenzothiazepine, 12g)
Affinity DataKi:  5.01E+3nM ΔG°:  -7.15kcal/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Acadia Pharmaceuticals

LigandPNGBDBM29096(dibenzothiazepine, 12b)
Affinity DatapH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Acadia Pharmaceuticals

LigandPNGBDBM29098(dibenzothiazepine, 12e)
Affinity DatapH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Acadia Pharmaceuticals

LigandPNGBDBM29101(dibenzothiazepine, 12j)
Affinity DatapH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Acadia Pharmaceuticals

LigandPNGBDBM29102(dibenzothiazepine, 12k)
Affinity DatapH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Acadia Pharmaceuticals

LigandPNGBDBM29095(dibenzothiazepine, 12a)
Affinity DatapH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2009
Entry Details Article
PubMed