Compile Data Set for Download or QSAR
Report error Found 4 of Enz. Inhib. data with enzyme = 'Casein kinase I isoform delta' and Substrate = 'CK1 Peptide Substrate'
TargetCasein kinase I isoform delta(Rat)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM6870(4-({5-amino-1-[(3-methylthiophen-2-yl)carbonyl]-1H...)
Affinity DataIC50: 570nMAssay Description:The enzyme was assayed with a biotinylated peptide substrate and test compounds in the presence of 10 uM ATP/[gamma-33P]ATP in a streptavidin coated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2005
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM6878(5-amino-N-(2,6-difluorophenyl)-3-[(4-sulfamoylphen...)
Affinity DataIC50: 2.80E+3nMAssay Description:The enzyme was assayed with a biotinylated peptide substrate and test compounds in the presence of 10 uM ATP/[gamma-33P]ATP in a streptavidin coated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2005
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM6866(1-Acyl-1H-[1,2,4]triazole-3,5-diamine Analogue 3b ...)
Affinity DataIC50: 1.12E+4nMAssay Description:The enzyme was assayed with a biotinylated peptide substrate and test compounds in the presence of 10 uM ATP/[gamma-33P]ATP in a streptavidin coated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2005
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Rat)
Johnson & Johnson Pharmaceutical

LigandPNGBDBM6867(4-({5-amino-1-[(2,6-difluoro-3-methylphenyl)carbon...)
Affinity DataIC50: 1.00E+5nMAssay Description:The enzyme was assayed with a biotinylated peptide substrate and test compounds in the presence of 10 uM ATP/[gamma-33P]ATP in a streptavidin coated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2005
Entry Details Article
PubMed