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Report error Found 40 of Enz. Inhib. data with enzyme = 'Casein kinase II subunit alpha' and Substrate = 'CK-2 Peptide Substrate'
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34046BDBM34046(iodinated benzimidazole, 9a)
Affinity DataKi:  19nM ΔG°:  -10.9kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34038BDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  23nM ΔG°:  -10.8kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34044BDBM34044(iodinated benzimidazole, 7a)
Affinity DataKi:  24nM ΔG°:  -10.8kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34051BDBM34051(iodinated benzimidazole, 14)
Affinity DataKi:  27nM ΔG°:  -10.7kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34052BDBM34052(iodinated benzimidazole, 15)
Affinity DataKi:  50nM ΔG°:  -10.4kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34054BDBM34054(iodinated benzimidazole, 17)
Affinity DataKi:  50nM ΔG°:  -10.4kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34053BDBM34053(iodinated benzimidazole, 16)
Affinity DataKi:  54nM ΔG°:  -10.3kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34048BDBM34048(iodinated benzimidazole, 11a)
Affinity DataKi:  70nM ΔG°:  -10.1kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34043BDBM34043(iodinated benzimidazole, 6a)
Affinity DataKi:  75nM ΔG°:  -10.1kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34050BDBM34050(iodinated benzimidazole, 13a)
Affinity DataKi:  90nM ΔG°:  -9.99kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34040BDBM34040(iodinated benzimidazole, 3a)
Affinity DataKi:  100nM ΔG°:  -9.93kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34049BDBM34049(iodinated benzimidazole, 12a)
Affinity DataKi:  120nM ΔG°:  -9.81kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34047BDBM34047(iodinated benzimidazole, 10a)
Affinity DataKi:  120nM ΔG°:  -9.81kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34056BDBM34056(iodinated benzimidazole, 23)
Affinity DataKi:  130nM ΔG°:  -9.77kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34055BDBM34055(iodinated benzimidazole, 21)
Affinity DataKi:  140nM ΔG°:  -9.72kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34039BDBM34039(iodinated benzimidazole, 2a)
Affinity DataKi:  160nM ΔG°:  -9.64kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34058BDBM34058(iodinated benzimidazole, 27)
Affinity DataKi:  160nM ΔG°:  -9.64kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11319BDBM11319(IQA | 2-{8-oxo-1,9-diazatetracyclo[8.7.0.0^{2,7}.0...)
Affinity DataKi:  170nM ΔG°:  -9.14kcal/mole IC50: 390nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34057BDBM34057(iodinated benzimidazole, 25)
Affinity DataKi:  180nM ΔG°:  -9.56kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34045BDBM34045(iodinated benzimidazole, 8a)
Affinity DataKi:  330nM ΔG°:  -9.19kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Maize)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11315BDBM11315(1,4-diamino-5,8-dihydroxy-9,10-dihydroanthracene-9...)
Affinity DataKi:  350nM ΔG°:  -8.71kcal/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11323BDBM11323(CHEMBL177820 | 4,5,6,7-tetrabromo-1H-1,2,3-benzotr...)
Affinity DataKi:  400nM ΔG°:  -8.63kcal/mole IC50: 500nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34041BDBM34041(iodinated benzimidazole, 4a)
Affinity DataKi:  460nM ΔG°:  -8.99kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34042BDBM34042(iodinated benzimidazole, 5a)
Affinity DataKi:  590nM ΔG°:  -8.83kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Padova

LigandChemical structure of BindingDB Monomer ID 7458BDBM7458(Naringenin, 18 | 5,7-dihydroxy-2-(4-hydroxyphenyl)...)
Affinity DataKi:  740nM ΔG°:  -8.27kcal/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Maize)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11313BDBM11313(4,5-dihydroxy-1-nitro-9,10-dihydroanthracene-9,10-...)
Affinity DataKi:  780nM ΔG°:  -8.24kcal/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Maize)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11314BDBM11314(1,8-dihydroxy-4-nitro-9H-xanthen-9-one | 1,8-dihyd...)
Affinity DataKi:  800nM ΔG°:  -8.23kcal/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11318BDBM11318(1,3,8-trihydroxy-6-methylanthra-9,10-quinone | CHE...)
Affinity DataKi:  1.85E+3nM ΔG°:  -7.74kcal/mole IC50: 890nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Padova

LigandChemical structure of BindingDB Monomer ID 7460BDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataKi:  1.18E+3nM ΔG°:  -8.00kcal/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34059BDBM34059(brominated benzimidazole, 20)
Affinity DataKi:  1.34E+3nM ΔG°:  -8.33kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34060BDBM34060(brominated benzimidazole, 22)
Affinity DataKi:  1.45E+3nM ΔG°:  -8.28kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34062BDBM34062(brominated benzimidazole, 26)
Affinity DataKi:  1.51E+3nM ΔG°:  -8.25kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Maize)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11318BDBM11318(1,3,8-trihydroxy-6-methylanthra-9,10-quinone | CHE...)
Affinity DataKi:  1.85E+3nM ΔG°:  -7.74kcal/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Rat)
University of Padova

LigandChemical structure of BindingDB Monomer ID 34061BDBM34061(brominated benzimidazole, 24)
Affinity DataKi:  1.91E+3nM ΔG°:  -8.11kcal/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11322BDBM11322(N-(3-chlorophenyl)-4-(2-{[2-(1H-imidazol-4-yl)ethy...)
Affinity DataIC50: 3.20E+3nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11320BDBM11320(3-{[4-(2-{[3-(1,1,2,2-tetrafluoroethoxy)phenyl]ami...)
Affinity DataIC50: 3.60E+3nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11324BDBM11324(CHEMBL375530 | (2R,3R,4S,5R)-2-(5,6-dichloro-1H-1,...)
Affinity DataKi:  4.50E+3nM ΔG°:  -7.22kcal/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11321BDBM11321(4-{2-[(2-aminoethyl)amino]pyridin-4-yl}-N-(3-chlor...)
Affinity DataIC50: 9.60E+3nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Maize)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11316BDBM11316(1,8-dihydroxy-anthraquinone | 1,8-dihydroxy-9,10-d...)
Affinity DataKi: >4.00E+4nM ΔG°: >-5.94kcal/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Maize)
University of Padova

LigandChemical structure of BindingDB Monomer ID 11317BDBM11317(1,8-dihydroxy-9H-xanthen-9-one | Xanthenone-relate...)
Affinity DataKi: >4.00E+4nM ΔG°: >-5.94kcal/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2006
Entry Details Article
PubMed