Compile Data Set for Download or QSAR
Report error Found 24 of Enz. Inhib. data with enzyme = 'Cathepsin S' and Substrate = 'BDBM22047'
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31970BDBM31970(Dipeptidyl nitrile inhibitor, 1)
Affinity DataIC50: 126nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31977BDBM31977(Dipeptidyl nitrile inhibitor, 10)
Affinity DataIC50: 200nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31988BDBM31988(Dipeptidyl nitrile inhibitor, 21)
Affinity DataIC50: 200nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31980BDBM31980(Dipeptidyl nitrile inhibitor, 13)
Affinity DataIC50: 316nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31975BDBM31975(Dipeptidyl nitrile inhibitor, 8)
Affinity DataIC50: 398nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31974BDBM31974(Dipeptidyl nitrile inhibitor, 7)
Affinity DataIC50: 631nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31993BDBM31993(Dipeptidyl nitrile inhibitor, 26)
Affinity DataIC50: 794nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31986BDBM31986(Dipeptidyl nitrile inhibitor, 19)
Affinity DataIC50: 794nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31987BDBM31987(Dipeptidyl nitrile inhibitor, 20)
Affinity DataIC50: 794nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31989BDBM31989(Dipeptidyl nitrile inhibitor, 22)
Affinity DataIC50: 794nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31990BDBM31990(Dipeptidyl nitrile inhibitor, 23)
Affinity DataIC50: 794nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31991BDBM31991(Dipeptidyl nitrile inhibitor, 24)
Affinity DataIC50: 794nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31984BDBM31984(Dipeptidyl nitrile inhibitor, 17)
Affinity DataIC50: 1.00E+3nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31992BDBM31992(Dipeptidyl nitrile inhibitor, 25)
Affinity DataIC50: 1.00E+3nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31978BDBM31978(Dipeptidyl nitrile inhibitor, 11)
Affinity DataIC50: 1.26E+3nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31985BDBM31985(Dipeptidyl nitrile inhibitor, 18)
Affinity DataIC50: 1.26E+3nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31976BDBM31976(Dipeptidyl nitrile inhibitor, 9)
Affinity DataIC50: 1.59E+3nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31979BDBM31979(Dipeptidyl nitrile inhibitor, 12)
Affinity DataIC50: 2.00E+3nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31972BDBM31972(Dipeptidyl nitrile inhibitor, 5)
Affinity DataIC50: 2.00E+3nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31971BDBM31971(Dipeptidyl nitrile inhibitor, 4)
Affinity DataIC50: 2.51E+3nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31973BDBM31973(Dipeptidyl nitrile inhibitor, 6)
Affinity DataIC50: 2.51E+3nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31981BDBM31981(Dipeptidyl nitrile inhibitor, 14)
Affinity DataIC50: 3.16E+3nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31983BDBM31983(Dipeptidyl nitrile inhibitor, 16)
Affinity DataIC50: 3.16E+3nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed
TargetCathepsin S(Human)
AstraZeneca

LigandChemical structure of BindingDB Monomer ID 31982BDBM31982(Dipeptidyl nitrile inhibitor, 15)
Affinity DataIC50: 1.00E+4nMAssay Description:IC50 values for inhibition of Cathepsins were determined from dose dependent inhibition of cleavage of fluorogenic, AMC-tagged, peptide substrates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2009
Entry Details Article
PubMed