Compile Data Set for Download or QSAR
Report error Found 10 of Enz. Inhib. data with enzyme = 'cGMP-dependent protein kinase 1' and Substrate = 'Histone H1'
LigandChemical structure of BindingDB Monomer ID 10840BDBM10840(4-(5-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50: 400nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
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Date in BDB:
8/26/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 10842BDBM10842(3-(2-aminopyrimidin-4-yl)-7-bromo-1H-indol-4-ol | ...)
Affinity DataIC50: 600nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 10843BDBM10843(4-(5,6-dibromo-1H-indol-3-yl)pyrimidin-2-amine | M...)
Affinity DataIC50: 600nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 10841BDBM10841(4-(6-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50: 800nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 10839BDBM10839(3-(2-aminopyrimidin-4-yl)-6-bromo-1H-indol-4-ol | ...)
Affinity DataIC50: 1.00E+3nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 10838BDBM10838(3-(2-aminopyrimidin-4-yl)-1H-indol-4-ol | Meridian...)
Affinity DataIC50: 2.00E+5nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 10844BDBM10844(4-(1H-indol-3-yl)pyrimidin-2-amine | Meridianin G)
Affinity DataIC50: 4.00E+5nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 10845BDBM10845(4-(5-bromo-1H-indol-2-yl)pyrimidin-2-amine | isome...)
Affinity DataIC50: 1.00E+6nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 10846BDBM10846(4-(1H-indol-2-yl)pyrimidin-2-amine | isomeridianin...)
Affinity DataIC50: 1.00E+6nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2006
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 7533BDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 1.00E+6nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30°C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2006
Entry Details Article
PubMed