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LigandPNGBDBM16315(CP-744809 | CHEMBL240725 | 6-[(5-chloro-3-methyl-1...)
Affinity DataIC50: 0.840nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM16315(CP-744809 | CHEMBL240725 | 6-[(5-chloro-3-methyl-1...)
Affinity DataIC50: 1nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM16633(6-[(5-fluoro-3-methyl-1-benzofuran-2-)sulfonyl]-2,...)
Affinity DataIC50: 3nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16452((4-oxo-3-{[5-(trifluoromethyl)-1,3-benzothiazol-2-...)
Affinity DataIC50: 4nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM16634(6-{[3-methyl-5-(trifluoromethyl)-1-benzofuran-2-]s...)
Affinity DataIC50: 5nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16636(6-[(5-chloro-3-ethyl-1-benzofuran-2-)sulfonyl]-2,3...)
Affinity DataIC50: 6nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16635(6-[(3,5-dimethyl-1-benzofuran-2-)sulfonyl]-2,3-dih...)
Affinity DataIC50: 13nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16638(6-[(3-phenyl-1-benzofuran-2-)sulfonyl]-2,3-dihydro...)
Affinity DataIC50: 23nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16457(CHEMBL240722 | 6-[(5-chloro-1-benzofuran-2-)sulfon...)
Affinity DataIC50: 25nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16457(CHEMBL240722 | 6-[(5-chloro-1-benzofuran-2-)sulfon...)
Affinity DataIC50: 25nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2007
Entry Details Article
PubMed
LigandPNGBDBM16620(6-{[(2-chloro-6-fluorophenyl)methane]sulfonyl}-2,3...)
Affinity DataIC50: 26nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16640(6-[(5-chloro-3-phenyl-1-benzofuran-2-)sulfonyl]-2,...)
Affinity DataIC50: 34nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16616(6-{[(2,3-dichlorophenyl)methane]sulfonyl}-2,3-dihy...)
Affinity DataIC50: 35nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16622(6-({[2-fluoro-3-(trifluoromethyl)phenyl]methane}su...)
Affinity DataIC50: 44nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16639(6-{[3-(4-fluorophenyl)-1-benzofuran-2-]sulfonyl}-2...)
Affinity DataIC50: 49nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16604(6-[(2,6-dichlorobenzene)sulfonyl]-2,3-dihydropyrid...)
Affinity DataIC50: 50nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16617(6-{[(2,6-dichlorophenyl)methane]sulfonyl}-2,3-dihy...)
Affinity DataIC50: 52nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16621(6-{[(3-chloro-2-fluorophenyl)methane]sulfonyl}-2,3...)
Affinity DataIC50: 54nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16642(6-[(5-chloro-3-methyl-1-benzothiophene-2-)sulfonyl...)
Affinity DataIC50: 55nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16602(6-[(2,3-dichlorobenzene)sulfonyl]-2,3-dihydropyrid...)
Affinity DataIC50: 55nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16615(6-({[3-(trifluoromethyl)phenyl]methane}sulfonyl)-2...)
Affinity DataIC50: 72nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16603(6-[(2,5-dichlorobenzene)sulfonyl]-2,3-dihydropyrid...)
Affinity DataIC50: 73nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50065954(5-Chloro-1H-indole-2-carboxylic acid ((S)-1-dimeth...)
Affinity DataIC50: 82nMAssay Description:In vitro inhibitory activity against recombinant human liver glycogen phosphorylase a (rHLGPa) catalyzed release of phosphate from glucose-1-phosphat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM16631(6-[(5,7-dichloro-1-benzofuran-2-)sulfonyl]-2,3-dih...)
Affinity DataIC50: 87nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16637(6-{[5-chloro-3-(propan-2-yl)-1-benzofuran-2-]sulfo...)
Affinity DataIC50: 92nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50065955(5-Bromo-1H-indole-2-carboxylic acid ((1S,2R)-1-ben...)
Affinity DataIC50: 97nMAssay Description:In vitro inhibitory activity against recombinant human liver glycogen phosphorylase a (rHLGPa) catalyzed release of phosphate from glucose-1-phosphat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50065951(5-Chloro-1H-indole-2-carboxylic acid ((S)-1-methyl...)
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory activity against recombinant human liver glycogen phosphorylase a (rHLGPa) catalyzed release of phosphate from glucose-1-phosphat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50065944(5-Bromo-1H-indole-2-carboxylic acid ((S)-1-dimethy...)
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory activity against recombinant human liver glycogen phosphorylase a (rHLGPa) catalyzed release of phosphate from glucose-1-phosphat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50065965(5-Chloro-1H-indole-2-carboxylic acid [2-((R)-dimet...)
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory activity against recombinant human liver glycogen phosphorylase a (rHLGPa) catalyzed release of phosphate from glucose-1-phosphat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM16612(6-{[(2-chlorophenyl)methane]sulfonyl}-2,3-dihydrop...)
Affinity DataIC50: 118nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16451(6-[(4-bromo-2-fluorobenzene)sulfonyl]-2,3-dihydrop...)
Affinity DataIC50: 140nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16629(6-[(3-methyl-1-benzofuran-2-)sulfonyl]-2,3-dihydro...)
Affinity DataIC50: 140nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16312(CHEMBL266497 | (4S)-6-fluoro-2,3-dihydrospiro[1-be...)
Affinity DataIC50: 140nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2007
Entry Details Article
PubMed
LigandPNGBDBM16451(6-[(4-bromo-2-fluorobenzene)sulfonyl]-2,3-dihydrop...)
Affinity DataIC50: 140nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2007
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50065943((S)-2-[(5-Chloro-1H-indole-2-carbonyl)-amino]-3-ph...)
Affinity DataIC50: 140nMAssay Description:In vitro inhibitory activity against recombinant human liver glycogen phosphorylase a (rHLGPa) catalyzed release of phosphate from glucose-1-phosphat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM16456(CHEMBL241777 | Heterocyclic Sulfonylpyridazinone, ...)
Affinity DataIC50: 150nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2007
Entry Details Article
PubMed
LigandPNGBDBM16456(CHEMBL241777 | Heterocyclic Sulfonylpyridazinone, ...)
Affinity DataIC50: 150nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16609(6-(alpha-Naphthylmethylbenzenesulfonyl)-2H-pyridaz...)
Affinity DataIC50: 150nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16455(Heterocyclic Sulfonylpyridazinone, 19w | 6-(1-benz...)
Affinity DataIC50: 150nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2007
Entry Details Article
PubMed
LigandPNGBDBM16641(6-[(5-methyl-1-benzothiophene-2-)sulfonyl]-2,3-dih...)
Affinity DataIC50: 160nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16444(Phenyl-Substituted Sulfonylpyridazinone, 8c | 6-[(...)
Affinity DataIC50: 170nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2007
Entry Details Article
PubMed
LigandPNGBDBM16444(Phenyl-Substituted Sulfonylpyridazinone, 8c | 6-[(...)
Affinity DataIC50: 170nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50065962(5-Fluoro-1H-indole-2-carboxylic acid ((1S,2R)-1-be...)
Affinity DataIC50: 170nMAssay Description:In vitro inhibitory activity against recombinant human liver glycogen phosphorylase a (rHLGPa) catalyzed release of phosphate from glucose-1-phosphat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM16607(6-{[3-(trifluoromethyl)benzene]sulfonyl}-2,3-dihyd...)
Affinity DataIC50: 175nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16455(Heterocyclic Sulfonylpyridazinone, 19w | 6-(1-benz...)
Affinity DataIC50: 180nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16449(Phenyl-Substituted Sulfonylpyridazinone, 8l | 6-[(...)
Affinity DataIC50: 190nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16449(Phenyl-Substituted Sulfonylpyridazinone, 8l | 6-[(...)
Affinity DataIC50: 190nMpH: 7.0 T: 2°CAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2007
Entry Details Article
PubMed
LigandPNGBDBM16632(6-[(6-chloro-3-methyl-1-benzofuran-2-)sulfonyl]-2,...)
Affinity DataIC50: 190nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
LigandPNGBDBM16628(6-[(5,7-dichloro-1H-indole-2-)sulfonyl]-2,3-dihydr...)
Affinity DataIC50: 200nMAssay Description:The activity of the enzyme was determined spectrophotometrically by monitoring the change in absorbance at 340 nm, which is due to the disappearance ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2007
Entry Details Article
PubMed
TargetGlycogen phosphorylase, liver form(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM35346(5-CHLORO-1H-INDOLE-2-CARBOXYLIC ACID [1-(4-FLUOROB...)
Affinity DataIC50: 205nMAssay Description:In vitro inhibitory activity against recombinant human liver glycogen phosphorylase a (rHLGPa) catalyzed release of phosphate from glucose-1-phosphat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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