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TargetFree fatty acid receptor 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265904(CHEMBL4079621)
Affinity DataEC50:  4.30E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415310(CHEMBL595238)
Affinity DataEC50:  25.1nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415118(CHEMBL576919)
Affinity DataEC50: >3.16E+4nMAssay Description:Agonist activity at human CB2 receptor expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415112(CHEMBL569535)
Affinity DataEC50: >3.16E+4nMAssay Description:Agonist activity at human CB1 receptor expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415309(CHEMBL608700)
Affinity DataEC50: >3.16E+4nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265860(CHEMBL4082804)
Affinity DataEC50: >1.70E+4nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50302371(1-[7-(3-Chloro-phenylamino)-3-methyl-1H-pyrrolo[2,...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human recombinant cannabinoid CB2 receptor expressed in MMY23 Saccharomyces cerevisiae assessed as degradation of FDGlu to fluore...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415315(CHEMBL593835)
Affinity DataEC50:  1.58E+3nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265883(CHEMBL4068825)
Affinity DataEC50:  1.90E+4nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50067499((6aR,10aR)-3-(1,1-dimethyl-heptyl)-9-hydroxymethyl...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human recombinant cannabinoid CB1 receptor expressed in MMY23 Saccharomyces cerevisiae assessed as degradation of FDGlu to fluore...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50302385(1-[7-(2-Chloro-phenylamino)-3-methyl-1H-pyrrolo[2,...)
Affinity DataEC50:  1.58E+4nMAssay Description:Agonist activity at human recombinant cannabinoid CB1 receptor expressed in MMY23 Saccharomyces cerevisiae assessed as degradation of FDGlu to fluore...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415124(CHEMBL577348)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human CB2 receptor expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50302373(7-(3-Chloro-phenylamino)-3-methyl-1H-pyrrolo[2,3-c...)
Affinity DataEC50:  265nMAssay Description:Agonist activity at human recombinant cannabinoid CB2 receptor expressed in MMY23 Saccharomyces cerevisiae assessed as degradation of FDGlu to fluore...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415319(CHEMBL595450)
Affinity DataEC50: >3.16E+4nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415316(CHEMBL596590)
Affinity DataEC50: >3.16E+4nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Mouse)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265897(CHEMBL4096579)
Affinity DataEC50:  17nMAssay Description:Agonist activity at mouse GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415322(CHEMBL608698)
Affinity DataEC50:  631nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50302375(7-(3-Chloro-phenylamino)-3-methyl-1H-pyrrolo[2,3-c...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human recombinant cannabinoid CB1 receptor expressed in MMY23 Saccharomyces cerevisiae assessed as degradation of FDGlu to fluore...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265877(CHEMBL4101071)
Affinity DataEC50:  710nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415104(CHEMBL570201)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human CB2 receptor expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415326(CHEMBL593581)
Affinity DataEC50: >3.16E+4nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50211839(2-(3-chloro-phenylamino)-4-trifluoromethyl-pyrimid...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in Saccharomyces cerevisiae cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415320(CHEMBL596155)
Affinity DataEC50: >3.16E+4nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415313(CHEMBL594531)
Affinity DataEC50: >3.16E+4nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265899(CHEMBL4087992)
Affinity DataEC50:  250nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50413240(CHEMBL471412)
Affinity DataEC50:  123nMAssay Description:Antagonist activity at human recombinant C5a receptor expressed in HEK cells assessed as inhibition of C5a-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415315(CHEMBL593835)
Affinity DataEC50: >3.16E+4nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265879(CHEMBL4065429)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50211871(2-(2,5-dichlorophenylamino)-4-trifluoromethylpyrim...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in Saccharomyces cerevisiae cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50211879(2-(3-chloro-phenylamino)-4-trifluoromethyl-pyrimid...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in Saccharomyces cerevisiae cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50211875(2-(3-chloro-phenylamino)-4-trifluoromethyl-pyrimid...)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in Saccharomyces cerevisiae cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50302380(1-[7-(3-Bromo-phenylamino)-3-methyl-1H-pyrrolo[2,3...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human recombinant cannabinoid CB2 receptor expressed in MMY23 Saccharomyces cerevisiae assessed as degradation of FDGlu to fluore...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415325(CHEMBL608702)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415334(CHEMBL610489)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265897(CHEMBL4096579)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265909(CHEMBL4082057)
Affinity DataEC50: >1.70E+4nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50211865(furan-2-ylmethyl 2-morpholino-4-(trifluoromethyl)p...)
Affinity DataEC50:  630nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in Saccharomyces cerevisiae cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415314(CHEMBL593834)
Affinity DataEC50: >3.16E+4nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50211870(2-(3-bromophenylamino)-4-trifluoromethylpyrimidine...)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in Saccharomyces cerevisiae cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265895(CHEMBL4097537)
Affinity DataEC50:  470nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Mouse)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265911(CHEMBL4078553)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at mouse GPR40 expressed in HEK293 cells assessed as increase in intracellular calcium level after 5 mins by FLUO-4-AM dye-based FLI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265912(CHEMBL4078374)
Affinity DataEC50:  4.10E+3nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50211856(2-phenylamino-4-trifluoromethylpyrimidine-5-carbox...)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in Saccharomyces cerevisiae cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415307(CHEMBL594281)
Affinity DataEC50: >3.16E+4nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265891(CHEMBL4060171)
Affinity DataEC50:  850nMAssay Description:Agonist activity at human GPR120 expressed in CHO-FlpIn cells after 15 mins by DMR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415110(CHEMBL577986)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human CB2 receptor expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415131(CHEMBL569949)
Affinity DataEC50:  63.1nMAssay Description:Agonist activity at human CB2 receptor expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415313(CHEMBL594531)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50211876(2-(3-chlorophenylamino)-4-trifluoromethylpyrimidin...)
Affinity DataEC50:  245nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in Saccharomyces cerevisiae cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50415115(CHEMBL583341)
Affinity DataEC50:  6.31E+3nMAssay Description:Agonist activity at human CB2 receptor expressed in yeast cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
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