Compile Data Set for Download or QSAR
Report error Found 287 with Last Name = 'deluca' and Initial = 'hf'
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50198705(CHEMBL226435 | (2Z)-(20R)-1alpha,25-dihydroxy-2-[(...)
Affinity DataEC50:  2.20nMAssay Description:Inhibition of human VDR induced-transcriptional transactivation of luciferase reporter gene in COS7 cells after 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50198705(CHEMBL226435 | (2Z)-(20R)-1alpha,25-dihydroxy-2-[(...)
Affinity DataEC50:  0.5nMAssay Description:Inhibition of human VDR induced-transcriptional transactivation of luciferase reporter gene in COS7 cells after 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50198707((2Z)-(20S)-1alpha,25-dihydroxy-2-[2''''-(fluoroeth...)
Affinity DataEC50:  1.10nMAssay Description:Inhibition of human VDR induced-transcriptional transactivation of luciferase reporter gene in COS7 cells after 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50198707((2Z)-(20S)-1alpha,25-dihydroxy-2-[2''''-(fluoroeth...)
Affinity DataEC50:  0.0700nMAssay Description:Inhibition of human VDR induced-transcriptional transactivation of luciferase reporter gene in COS7 cells after 24 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244240((20S)-(2E)-1-alpha-25-Dihydroxy-2-[2-(hydroxy)-eth...)
Affinity DataEC50:  0.0260nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50412385(CHEMBL2021488)
Affinity DataEC50:  0.0900nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50005618(CHEMBL2021484)
Affinity DataEC50:  0.00210nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244241((20R)-(2E)-1-alpha-25-Dihydroxy-2-[2-(hydroxy)-eth...)
Affinity DataEC50:  0.200nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244165(CHEMBL514116 | (20R)-1-alpha,25-Dihydroxy-2-alpha-...)
Affinity DataEC50:  0.0240nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244269(CHEMBL513573 | (20R)-1-alpha-2-alpha-25-Trihydroxy...)
Affinity DataEC50:  0.120nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50412386(CHEMBL2021486)
Affinity DataEC50:  0.0580nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244241((20R)-(2E)-1-alpha-25-Dihydroxy-2-[2-(hydroxy)-eth...)
Affinity DataEC50:  0.0290nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244165(CHEMBL514116 | (20R)-1-alpha,25-Dihydroxy-2-alpha-...)
Affinity DataEC50:  0.115nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244268((20S)-1-alpha-2-alpha-25-Trihydroxy-2beta-methyl-1...)
Affinity DataEC50:  1.90nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244269(CHEMBL513573 | (20R)-1-alpha-2-alpha-25-Trihydroxy...)
Affinity DataEC50:  4.5nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244164((20S)-1-alpha-25-Dihydroxy-2-alpha-(2-hydroxyethox...)
Affinity DataEC50:  0.0270nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244268((20S)-1-alpha-2-alpha-25-Trihydroxy-2beta-methyl-1...)
Affinity DataEC50:  0.0170nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244240((20S)-(2E)-1-alpha-25-Dihydroxy-2-[2-(hydroxy)-eth...)
Affinity DataEC50:  0.0850nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50412385(CHEMBL2021488)
Affinity DataEC50:  0.0900nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Mouse)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50412386(CHEMBL2021486)
Affinity DataEC50:  0.0300nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50292704((25R)-26-adamantyl-1R,25-hydroxy-2-methylene-22,23...)
Affinity DataEC50:  24nMAssay Description:Agonist activity at VDR assessed as receptor transactivation by transient transcription assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50292705((25R)-25-Adamantyl-1alpha,25-dihydroxy-2-methylene...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at VDR assessed as receptor transactivation by transient transcription assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50292706((24R)-24-Adamantyl-1r,24-dihydroxy-2-methylene-22,...)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at VDR assessed as receptor transactivation by transient transcription assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.200nMAssay Description:Activity at rat recombinant full length VDR expressed in rat ROS 17/2.8 cells transfected with 24-hydroxylase gene promoter assessed as transcription...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50292630((5R)-5-{(2R)-2-[(1R,3R,7E)-1,3-Dihydroxy-2-methyle...)
Affinity DataEC50:  100nMAssay Description:Activity at rat recombinant full length VDR expressed in rat ROS 17/2.8 cells transfected with 24-hydroxylase gene promoter assessed as transcription...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50292629((23S)-25-dehydro-2-methylene-19-nor-1alpha-hydroxy...)
Affinity DataEC50:  2nMAssay Description:Activity at rat recombinant full length VDR expressed in rat ROS 17/2.8 cells transfected with 24-hydroxylase gene promoter assessed as transcription...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.200nMAssay Description:Activity at VDR in rat ROS 17/2.8 cells assessed as transcriptional activation of 24-hydroxylase gene promoter after 16 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50293269((1R,3R)-5-[(E)-(5'S,7'S)-11'-hydroxy-5',7',11'-tri...)
Affinity DataEC50:  90nMAssay Description:Activity at VDR in rat ROS 17/2.8 cells assessed as transcriptional activation of 24-hydroxylase gene promoter after 16 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50293270((1R,3R)-5-[(E)-(5'R,7'S)-11'-Hydroxy-5',7',11'-tri...)
Affinity DataEC50:  3nMAssay Description:Activity at VDR in rat ROS 17/2.8 cells assessed as transcriptional activation of 24-hydroxylase gene promoter after 16 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50293271((7Z)-(20S)-1alpha,25-Dihydroxy-2-methylene-8(12),1...)
Affinity DataEC50:  100nMAssay Description:Activity at VDR in rat ROS 17/2.8 cells assessed as transcriptional activation of 24-hydroxylase gene promoter after 16 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50293272((20S)-1alpha,25-Dihydroxy-2-methylene-8(12),14(17)...)
Affinity DataEC50:  100nMAssay Description:Activity at VDR in rat ROS 17/2.8 cells assessed as transcriptional activation of 24-hydroxylase gene promoter after 16 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50293268((1R,3R)-5-((R)-11-hydroxy-7,11-dimethyldodec-2-eny...)
Affinity DataEC50:  50nMAssay Description:Activity at VDR in rat ROS 17/2.8 cells assessed as transcriptional activation of 24-hydroxylase gene promoter after 16 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.300nMAssay Description:Activity at VDR in rat osteosarcoma cells assessed as induction of 24-hydroxylase reporter gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50304584(1alpha,25-Dihydroxy-2-methylene-19,21-dinorvitamin...)
Affinity DataEC50:  0.200nMAssay Description:Activity at VDR in rat osteosarcoma cells assessed as induction of 24-hydroxylase reporter gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50304585((20S)-1alpha,25-Dihydroxy-2-methylene-18,19-dinorv...)
Affinity DataEC50:  0.0200nMAssay Description:Activity at VDR in rat osteosarcoma cells assessed as induction of 24-hydroxylase reporter gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50304583(1alpha,25-Dihydroxy-2-methylene-18,19,21-trinorvit...)
Affinity DataEC50:  0.0600nMAssay Description:Activity at VDR in rat osteosarcoma cells assessed as induction of 24-hydroxylase reporter gene transcription by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at rat VDR in ROS 17/2.8 cells transfected with Cyp24a1 reporter plasmid assessed as increase in Cyp24a1 transcription after 16 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50293268((1R,3R)-5-((R)-11-hydroxy-7,11-dimethyldodec-2-eny...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at rat VDR in ROS 17/2.8 cells transfected with Cyp24a1 reporter plasmid assessed as increase in Cyp24a1 transcription after 16 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50359362(CHEMBL1929240)
Affinity DataEC50:  2nMAssay Description:Agonist activity at rat VDR in ROS 17/2.8 cells transfected with Cyp24a1 reporter plasmid assessed as increase in Cyp24a1 transcription after 16 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50359363(CHEMBL1929241)
Affinity DataEC50:  30nMAssay Description:Agonist activity at rat VDR in ROS 17/2.8 cells transfected with Cyp24a1 reporter plasmid assessed as increase in Cyp24a1 transcription after 16 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Bovine)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50205233((20S,22R)-22-methyl-1-alpha-25-dihydroxy-vitamin D...)
Affinity DataEC50:  0.0180nMAssay Description:Displacement of [3H]1,25-(OH)2D3 from vitamin D receptor in bovine thymusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Bovine)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50205234((20S,22R)-22-methyl-1-alpha-25-dihydroxy-vitamin D...)
Affinity DataEC50:  0.0310nMAssay Description:Displacement of [3H]1,25-(OH)2D3 from vitamin D receptor in bovine thymusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Bovine)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.0710nMAssay Description:Displacement of [3H]1,25-(OH)2D3 from vitamin D receptor in bovine thymusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.5nMAssay Description:Induction of transactivation of human VDR responsive gene in COS7 cells by rat osteopontin luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50205234((20S,22R)-22-methyl-1-alpha-25-dihydroxy-vitamin D...)
Affinity DataEC50:  0.00300nMAssay Description:Induction of transactivation of human VDR responsive gene in COS7 cells by rat osteopontin luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50205233((20S,22R)-22-methyl-1-alpha-25-dihydroxy-vitamin D...)
Affinity DataEC50:  0.00200nMAssay Description:Induction of transactivation of human VDR responsive gene in COS7 cells by rat osteopontin luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50205235((20S,22R)-22-methyl-1-alpha-25-dihydroxy-vitamin D...)
Affinity DataEC50:  0.200nMAssay Description:Induction of transactivation of human VDR responsive gene in COS7 cells by rat osteopontin luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Bovine)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50205235((20S,22R)-22-methyl-1-alpha-25-dihydroxy-vitamin D...)
Affinity DataEC50:  0.890nMAssay Description:Displacement of [3H]1,25-(OH)2D3 from vitamin D receptor in bovine thymusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.200nMAssay Description:Activity at VDR in rat osteosarcoma cells assessed as 24-hydroxylase transcription by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2012
Entry Details Article
PubMed
TargetVitamin D3 receptor(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50292315((5R,8aR,Z)-7-((E)-2-((3aS,7aR)-1-((R)-6-hydroxy-6-...)
Affinity DataEC50:  100nMAssay Description:Activity at VDR in rat osteosarcoma cells assessed as 24-hydroxylase transcription by reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2012
Entry Details Article
PubMed
Displayed 1 to 50 (of 287 total ) | Next | Last >>
Jump to: