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LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123147(US8742113, 239)
Affinity DataIC50:  1nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123148(US8742113, 242)
Affinity DataIC50:  1nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123131(US8742113, 15)
Affinity DataIC50:  2nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123146(US8742113, 233)
Affinity DataIC50:  2nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

LigandPNGBDBM50237689(CHEMBL4066943)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237692(CHEMBL4091162)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123142(US8742113, 142)
Affinity DataIC50:  3nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123144(US8742113, 173)
Affinity DataIC50:  3nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123143(US8742113, 157)
Affinity DataIC50:  3nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123137(US8742113, 89)
Affinity DataIC50:  3nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123140(US8742113, 126)
Affinity DataIC50:  3nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

LigandPNGBDBM50237682(CHEMBL4083363)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of 1 nM AVP-induced cAMP accumulation in cells expressing human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237673(CHEMBL4098085)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237695(CHEMBL4072935)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237701(CHEMBL4098908)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237702(CHEMBL4070220)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123138(US8742113, 91)
Affinity DataIC50:  4nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123149(US8742113, 244)
Affinity DataIC50:  4nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123134(US8742113, 68)
Affinity DataIC50:  4nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123145(US8742113, 226)
Affinity DataIC50:  4nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123139(US8742113, 102)
Affinity DataIC50:  4nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

LigandPNGBDBM50237698(CHEMBL4090216)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237690(CHEMBL4084928)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237688(CHEMBL4091575)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  5nMAssay Description:Inhibition of CLK1 (unknown origin) pretreated for 30 mins followed by substrate addition measured after 5 hrs in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123136(US8742113, 81)
Affinity DataIC50:  5nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

TargetDual specificity protein kinase CLK2(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of CLK2 (unknown origin) pretreated for 30 mins followed by substrate addition measured after 5 hrs in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237691(CHEMBL4080872)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123133(US8742113, 63)
Affinity DataIC50:  6nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

LigandPNGBDBM50237686(CHEMBL4062056)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237694(CHEMBL4061554)
Affinity DataIC50:  8nMAssay Description:Inhibition of 1 nM AVP-induced cAMP accumulation in cells expressing human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123151(US8742113, 246)
Affinity DataIC50:  8nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123150(US8742113, 245)
Affinity DataIC50:  8nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123141(US8742113, 129)
Affinity DataIC50:  9nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

LigandPNGBDBM50237697(CHEMBL4085578)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of 1 nM AVP-induced cAMP accumulation in cells expressing human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237675(CHEMBL4087825)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123132(US8742113, 22)
Affinity DataIC50:  10nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM123135(US8742113, 78)
Affinity DataIC50:  11nMpH: 7.5Assay Description:Measurement of kinase activity was carried out using an MSA assay kit (QuickScout Screening Assist Kit, Carna Biosciences, Inc.). Assay buffer (20 mM...More data for this Ligand-Target Pair
In DepthDetails US Patent

LigandPNGBDBM50237687(CHEMBL4083793)
Affinity DataIC50:  12nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237699(CHEMBL4060978)
Affinity DataIC50:  12nMAssay Description:Inhibition of 1 nM AVP-induced cAMP accumulation in cells expressing human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237674(CHEMBL4099816)
Affinity DataIC50:  18nMAssay Description:Inhibition of 1 nM AVP-induced cAMP accumulation in cells expressing human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237677(CHEMBL4062207)
Affinity DataIC50:  23nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237700(CHEMBL4070681)
Affinity DataIC50:  29nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237693(CHEMBL4083382)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237678(CHEMBL4082371)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  30nMAssay Description:Inhibition of PIM1 (unknown origin) in presence of 1 mM ATP without preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  34nMAssay Description:Inhibition of PIM1 (unknown origin) in presence of 1 mM ATP with preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237676(CHEMBL4066501)
Affinity DataIC50:  36nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Human)
Sbi Biotech

US Patent
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  36nMAssay Description:Inhibition of CDC7 in human SW-620 cells assessed as reduction in phosphorylation of MCM2 at Ser40 residue incubated for 48 hrs by Western blot analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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