Report error Found 1215 with Last Name = 'garcia' and Initial = 's'
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 96nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 189nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 970nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as induction of intracellular calcium release after 15 mins by FLIPR ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 483nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as induction of intracellular calcium release after 15 mins by FLIPR ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as induction of intracellular calcium release after 15 mins by FLIPR ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as induction of intracellular calcium release after 15 mins by FLIPR ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as induction of intracellular calcium release after 15 mins by FLIPR ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 70nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 73nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 85nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 484nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 2.16E+3nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 51nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 298nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 67nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 194nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 363nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human GHSR1a expressed in HEK293 cells assessed as induction of intracellular calcium release after 15 mins by FLIPR ...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 86nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 439nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 306nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 121nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 937nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 117nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 1.28E+3nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Human)
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Sib Swiss Institute of Bioinformatics
Curated by ChEMBL
Affinity DataEC50: 634nMAssay Description:Inverse agonist at recombinant human GHSR1a expressed in HEK293 cells assessed as decrease in IP1 accumulation after 1 hr by IP1-d2-based HTRF assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Baker's yeast)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: 178nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Baker's yeast)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: 467nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Baker's yeast)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: 223nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Baker's yeast)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: 524nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Baker's yeast)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Baker's yeast)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Baker's yeast)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: 183nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Baker's yeast)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: 121nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Baker's yeast)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Baker's yeast)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 6(Human)
Centro De Investigaci£N Lilly S.A. Avda. De La Industria
Curated by ChEMBL
Centro De Investigaci£N Lilly S.A. Avda. De La Industria
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human recombinant mGlu6 stably expressed in golden hamster AV12 cell membrane co-expressing Galpha15 assessed as assessed as incr...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Human)
Centro De Investigaci£N Lilly S.A. Avda. De La Industria
Curated by ChEMBL
Centro De Investigaci£N Lilly S.A. Avda. De La Industria
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human recombinant mGlu1 stably expressed in golden hamster AV12 cell membrane co-expressing Gq assessed as assessed as increase i...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Human)
Centro De Investigaci£N Lilly S.A. Avda. De La Industria
Curated by ChEMBL
Centro De Investigaci£N Lilly S.A. Avda. De La Industria
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human recombinant mGlu4 stably expressed in golden hamster AV12 cell membrane co-expressing Galpha15 assessed as assessed as incr...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Human)
Centro De Investigaci£N Lilly S.A. Avda. De La Industria
Curated by ChEMBL
Centro De Investigaci£N Lilly S.A. Avda. De La Industria
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human recombinant mGlu5 stably expressed in golden hamster AV12 cell membrane co-expressing Gq assessed as assessed as increase i...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 8(Human)
Centro De Investigaci£N Lilly S.A. Avda. De La Industria
Curated by ChEMBL
Centro De Investigaci£N Lilly S.A. Avda. De La Industria
Curated by ChEMBL
Affinity DataEC50: 1.77E+3nMAssay Description:Antagonist activity at human recombinant mGlu8 stably expressed in golden hamster AV12 cell membrane co-expressing Galpha15 assessed as reduction in ...More data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Competitive inhibition of HIS-FLAG-tagged recombinant Leishmania infantum TryR expressed in Escherichia coli assessed as dissociation constant by SPR...More data for this Ligand-Target Pair
Affinity DataEC50: 0.950nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as ERK phosphorylation incubated for 2 hrs by Alphascreen surefire...More data for this Ligand-Target Pair
Affinity DataEC50: 9.85E+3nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as ERK phosphorylation incubated for 2 hrs by Alphascreen surefire...More data for this Ligand-Target Pair
Affinity DataEC50: 5.86E+3nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO-K1 cells assessed as ERK phosphorylation incubated for 2 hrs by Alphascreen surefire...More data for this Ligand-Target Pair
