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TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 13nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM50005215(CHEMBL3109274)
Affinity DataIC50: 15nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM5875(N-[5-(ethanesulfonyl)-2-methoxyphenyl]-5-[3-(pyrid...)
Affinity DataIC50: 17nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataIC50: 31nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM50005212(CHEMBL3109275)
Affinity DataIC50: 51nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Universit�� Di Firenze

LigandPNGBDBM237337(N-(3-morpholinopropyl)benzene-1,4-disulfonamide (I...)
Affinity DataIC50: 57.7nMpH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Universit�� Di Firenze

LigandPNGBDBM237338(N-(4-diethylaminoethoxybenzyl)benzene-1,4-bis-sulf...)
Affinity DataIC50: 59.8nMpH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Universit�� Di Firenze

LigandPNGBDBM237337(N-(3-morpholinopropyl)benzene-1,4-disulfonamide (I...)
Affinity DataIC50: 65.8nMpH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Universit�� Di Firenze

LigandPNGBDBM237338(N-(4-diethylaminoethoxybenzyl)benzene-1,4-bis-sulf...)
Affinity DataIC50: 81.1nMpH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM50005213(CHEMBL3109276)
Affinity DataIC50: 170nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Comenius University

Curated by ChEMBL
LigandPNGBDBM50005214(CHEMBL3109277)
Affinity DataIC50: 202nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR2 expressed in Sf9 cells by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2014
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Universit�� Di Firenze

LigandPNGBDBM237336(4-Sulfamoyl-N-(3-morpholinopropyl)benzamide (I-1))
Affinity DataIC50: 216nMpH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
Universit�� Di Firenze

LigandPNGBDBM237336(4-Sulfamoyl-N-(3-morpholinopropyl)benzamide (I-1))
Affinity DataIC50: 231nMpH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 4(Human)
Universit�� Di Firenze

LigandPNGBDBM237337(N-(3-morpholinopropyl)benzene-1,4-disulfonamide (I...)
Affinity DataIC50: 499nMpH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 4(Human)
Universit�� Di Firenze

LigandPNGBDBM237338(N-(4-diethylaminoethoxybenzyl)benzene-1,4-bis-sulf...)
Affinity DataIC50: 508nMpH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
Universit�� Di Firenze

LigandPNGBDBM237337(N-(3-morpholinopropyl)benzene-1,4-disulfonamide (I...)
Affinity DataIC50: 517nMpH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 4(Human)
Universit�� Di Firenze

LigandPNGBDBM237336(4-Sulfamoyl-N-(3-morpholinopropyl)benzamide (I-1))
Affinity DataIC50: 611nMpH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
Universit�� Di Firenze

LigandPNGBDBM237336(4-Sulfamoyl-N-(3-morpholinopropyl)benzamide (I-1))
Affinity DataIC50: 645nMpH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
Universit�� Di Firenze

LigandPNGBDBM237338(N-(4-diethylaminoethoxybenzyl)benzene-1,4-bis-sulf...)
Affinity DataIC50: 737nMpH: 7.5 T: 2°CAssay Description:An Applied Photophysics stopped-flow instrument has been used for assaying the CA catalysed CO2 hydration activity [Khalifah et al., J. Biol. Chem., ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details Article
PubMed