Compile Data Set for Download or QSAR
Report error Found 677 with Last Name = 'gwaltney' and Initial = 'sl'
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242755(CHEMBL4101006)
Affinity DataEC50:  120nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242756(CHEMBL4083023)
Affinity DataEC50:  80nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242757(CHEMBL4090814)
Affinity DataEC50:  100nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242758(CHEMBL4085525)
Affinity DataEC50:  100nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242759(CHEMBL4063950)
Affinity DataEC50:  100nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242767(CHEMBL4072542)
Affinity DataEC50:  3.10E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242768(CHEMBL4060580)
Affinity DataEC50:  7.90E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242769(CHEMBL4082468)
Affinity DataEC50:  5.00E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242770(CHEMBL4071981)
Affinity DataEC50:  1.60E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242772(CHEMBL4091218)
Affinity DataEC50:  200nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242781(CHEMBL4083428)
Affinity DataEC50:  40nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242782(CHEMBL4101417)
Affinity DataEC50:  31nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242783(CHEMBL4072997)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242784(CHEMBL4090191)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242785(CHEMBL4069128)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242786(CHEMBL4082347)
Affinity DataEC50:  1.00E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242792(CHEMBL4071846)
Affinity DataEC50:  4.00E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242793(CHEMBL4098841)
Affinity DataEC50:  630nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242794(CHEMBL4091097)
Affinity DataEC50:  1.20E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242795(CHEMBL4098957)
Affinity DataEC50:  1.20E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242796(CHEMBL4063355)
Affinity DataEC50:  790nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242797(CHEMBL4093697)
Affinity DataEC50:  500nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242798(CHEMBL4060445)
Affinity DataEC50:  2.00E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242814(CHEMBL4063218)
Affinity DataEC50:  630nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242815(CHEMBL4062882)
Affinity DataEC50:  100nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242816(CHEMBL4093271)
Affinity DataEC50:  120nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM16181(1-[2-(4-cyanophenyl)-2-hydroxy-2-(1-methyl-1H-imid...)
Affinity DataEC50:  4nMAssay Description:Inhibition of Ras farnesylation in Human Ha-Ras oncogene-transformed BALB/c 3T3 cells (EJ3 cells)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50126323(1-{3-[3-(4-Cyano-benzyl)-3H-imidazol-4-yl]-propion...)
Affinity DataEC50:  28nMAssay Description:Inhibition of Ras farnesylation in Human Ha-Ras oncogene-transformed BALB/c 3T3 cells (EJ3 cells)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50126324(1-{2-[3-(4-Cyano-3-naphthalen-1-yl-benzyl)-3H-imid...)
Affinity DataEC50: >100nMAssay Description:Inhibition of Ras farnesylation in Human Ha-Ras oncogene-transformed BALB/c 3T3 cells (EJ3 cells)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50126320(1-{[(4-Cyano-phenyl)-(3-methyl-3H-imidazol-4-yl)-m...)
Affinity DataEC50:  0.5nMAssay Description:Inhibition of Ras farnesylation in Human Ha-Ras oncogene-transformed BALB/c 3T3 cells (EJ3 cells)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM17335(1-[(2R)-2-{[(4-cyanophenyl)methyl](methyl)amino}-3...)
Affinity DataEC50: >100nMAssay Description:Inhibition of Ras farnesylation in Human Ha-Ras oncogene-transformed BALB/c 3T3 cells (EJ3 cells)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50126327(1-{2-[3-(3-Chloro-4-cyano-benzyl)-3H-imidazol-4-yl...)
Affinity DataEC50: >100nMAssay Description:Inhibition of Ras farnesylation in Human Ha-Ras oncogene-transformed BALB/c 3T3 cells (EJ3 cells)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50126318(1-{2-[3-(4-Chloro-benzyl)-3H-imidazol-4-yl]-acetyl...)
Affinity DataEC50: >100nMAssay Description:Inhibition of Ras farnesylation in Human Ha-Ras oncogene-transformed BALB/c 3T3 cells (EJ3 cells)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50126325(4-Cyano-5-naphthalen-1-yl-3,6-dihydro-2H-pyridine-...)
Affinity DataEC50:  97nMAssay Description:Inhibition of Ras farnesylation in Human Ha-Ras oncogene-transformed BALB/c 3T3 cells (EJ3 cells)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50126322(4-Cyano-5-naphthalen-1-yl-3,6-dihydro-2H-pyridine-...)
Affinity DataEC50: >1nMAssay Description:Inhibition of Ras farnesylation in Human Ha-Ras oncogene-transformed BALB/c 3T3 cells (EJ3 cells)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50126317(1-{2-[3-(4-Cyano-benzyl)-3H-imidazol-4-yl]-acetyl}...)
Affinity DataEC50:  3.90nMAssay Description:Inhibition of Ras farnesylation in Human Ha-Ras oncogene-transformed BALB/c 3T3 cells (EJ3 cells)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50126326(1-[(4-Cyano-phenyl)-(3-methyl-3H-imidazol-4-yl)-me...)
Affinity DataEC50:  31nMAssay Description:Inhibition of Ras farnesylation in Human Ha-Ras oncogene-transformed BALB/c 3T3 cells (EJ3 cells)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50135356(6-[(2'-Chloro-6-cyano-biphenyl-3-yl)-(3-methyl-3H-...)
Affinity DataEC50: >100nMAssay Description:In vitro effective concentration against farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50135358(6-[(3-Bromo-4-cyano-phenyl)-(3-methyl-3H-imidazol-...)
Affinity DataEC50:  39nMAssay Description:In vitro effective concentration against farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM17325(CHEMBL29982 | (2S)-2-[(4-{[butyl(2-cyclohexylethyl...)
Affinity DataEC50:  16nMAssay Description:In vitro effective concentration against farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50135366(6-[(3-Chloro-4-cyano-phenyl)-(3-methyl-3H-imidazol...)
Affinity DataEC50:  16nMAssay Description:In vitro effective concentration against farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50135365(6-[(4-Cyano-phenyl)-(3-methyl-3H-imidazol-4-yl)-me...)
Affinity DataEC50: >100nMAssay Description:In vitro effective concentration against farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50135362(6-[(4-Cyano-phenyl)-(3-methyl-3H-imidazol-4-yl)-me...)
Affinity DataEC50:  86nMAssay Description:In vitro effective concentration against farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50135370(6-[(3'-Chloro-6-cyano-biphenyl-3-yl)-(3-methyl-3H-...)
Affinity DataEC50:  21nMAssay Description:In vitro effective concentration against farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50135369(5-(3-Chloro-4-fluoro-phenyl)-6-[(4-cyano-phenyl)-(...)
Affinity DataEC50:  15nMAssay Description:In vitro effective concentration against farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50135363(6-[(4-Cyano-phenyl)-(3-methyl-3H-imidazol-4-yl)-me...)
Affinity DataEC50:  10nMAssay Description:In vitro effective concentration against farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50135367(5-Benzo[1,3]dioxol-5-yl-6-[(4-cyano-phenyl)-(3-met...)
Affinity DataEC50:  2.10nMAssay Description:In vitro effective concentration against farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50135361(6-[(4-Cyano-phenyl)-(3-methyl-3H-imidazol-4-yl)-me...)
Affinity DataEC50:  3.90nMAssay Description:In vitro effective concentration against farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50135353(5-(3-Chloro-phenyl)-6-[(4-cyano-phenyl)-(3-methyl-...)
Affinity DataEC50:  0.5nMAssay Description:In vitro effective concentration against farnesyltransferase (FT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50135379(6-[(4-Cyano-phenyl)-(3-methyl-3H-imidazol-4-yl)-me...)
Affinity DataEC50:  1.20nMAssay Description:In vitro effective concentration against farnesyltransferase (FT); Not activeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 677 total ) | Next | Last >>
Jump to: