Report error Found 530 with Last Name = 'hoffman' and Initial = 'a'
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 1.68E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 49nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: >100nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.75E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 990nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 390nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 130nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel by isothermal calorimetric titrationMore data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 2.17E+3nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel by isothermal calorimetric titrationMore data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 1.30E+4nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage c...More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
University of Vienna
Curated by ChEMBL
University of Vienna
Curated by ChEMBL
Affinity DataEC50: 3.18E+4nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
Affinity DataEC50: 3.96E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Human)
University of Basel
Curated by ChEMBL
University of Basel
Curated by ChEMBL
Affinity DataEC50: 6.72E+4nMAssay Description:Modulation of GABAA alpha1beta3gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of EC3 to 10 GABA-induc...More data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 9.00E+3nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage c...More data for this Ligand-Target Pair
Affinity DataEC50: 2.25E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 320nMAssay Description:Binding affinity to C-terminal amidated influenza A virus A/Udorn/72 (H3N2) M2 transmembrane domain (22 to 46 residues) in DPC micelles at pH 8 asses...More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 28nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 2.10E+5nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 M2 proton channel S31N mutant expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage...More data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 3.20E+3nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage c...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
University of Vienna
Curated by ChEMBL
University of Vienna
Curated by ChEMBL
Affinity DataEC50: 5.53E+4nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 2.17E+3nMAssay Description:Binding affinity to C-terminal amidated influenza A virus A/Udorn/72 (H3N2) M2 transmembrane domain (22 to 46 residues) in DPC micelles at pH 8 asses...More data for this Ligand-Target Pair
Affinity DataEC50: >100nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0970nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 640nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 8.80E+4nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage c...More data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 340nMAssay Description:Binding affinity to C-terminal amidated influenza A virus A/Udorn/72 (H3N2) M2 transmembrane domain (22 to 46 residues) in DPC micelles at pH 8 asses...More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
University of Vienna
Curated by ChEMBL
University of Vienna
Curated by ChEMBL
Affinity DataEC50: 1.02E+5nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Human)
University of Basel
Curated by ChEMBL
University of Basel
Curated by ChEMBL
Affinity DataEC50: 2.95E+4nMAssay Description:Modulation of GABAA alpha1beta3gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as modulation of GABA-induced chloride ...More data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 1.20E+4nMAssay Description:Binding affinity to Influenza A virus M2 transmembrane domain by analytical ultracentrifugation methodMore data for this Ligand-Target Pair
Affinity DataEC50: 1.19E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 310nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0630nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 320nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel by isothermal calorimetric titrationMore data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 340nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel by isothermal calorimetric titrationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens
Curated by ChEMBL
National and Kapodistrian University of Athens
Curated by ChEMBL
Affinity DataKd: 1.80E+6nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 M2 proton channel S31N mutant expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Human)
University of Basel
Curated by ChEMBL
University of Basel
Curated by ChEMBL
Affinity DataEC50: 8.08E+4nMAssay Description:Modulation of GABAA alpha2beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of EC3 to 10 GABA-induc...More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 64nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding affinity to TYK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.46E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 770nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >100nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem
Curated by ChEMBL
The Hebrew University of Jerusalem
Curated by ChEMBL
Affinity DataEC50: 1.18E+4nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair









3D Structure (crystal)


















