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TargetPeroxisome proliferator-activated receptor alpha(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50607785(CHEMBL5219536)
Affinity DataEC50:  5.82E+4nMAssay Description:Partial agonist activity at PPARalpha (unknown origin) assessed as increase in PRIP/RAP250 coactivator peptide requirement by Lanthascreen TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50099491(cid_3392731 | CHEMBL21241 | 2-(4-{2-[3-Cyclohexyl-...)
Affinity DataEC50:  20nMAssay Description:Partial agonist activity at PPARalpha (unknown origin) assessed as increase in PRIP/RAP250 coactivator peptide requirement by Lanthascreen TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50607785(CHEMBL5219536)
Affinity DataEC50:  5.08E+4nMAssay Description:Partial agonist activity at PPARgamma (unknown origin) assessed as increase in fluorescein labeled PRIP/RAP250 coactivator peptide requirement by Lan...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50085048((S)-2-(2-benzoylphenylamino)-3-(4-(2-(methyl(pyrid...)
Affinity DataEC50:  50nMAssay Description:Partial agonist activity at PPARgamma (unknown origin) assessed as increase in fluorescein labeled PRIP/RAP250 coactivator peptide requirement by Lan...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50103521(CHEBI:8228 | Actos | Duetact | Pioglitazone | US20...)
Affinity DataEC50:  6.70E+3nMAssay Description:Partial agonist activity at PPARgamma (unknown origin) assessed as increase in fluorescein labeled PRIP/RAP250 coactivator peptide requirement by Lan...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50607785(CHEMBL5219536)
Affinity DataEC50:  5.39E+4nMAssay Description:Partial agonist activity at PPARdelta (unknown origin) assessed as increase in fluorescein labeled PRIP/RAP250 coactivator peptide requirement by Lan...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataEC50:  700nMAssay Description:Partial agonist activity at PPARdelta (unknown origin) assessed as increase in fluorescein labeled PRIP/RAP250 coactivator peptide requirement by Lan...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at RXRalpha-LBD (unknown origin) assessed as transactivation by measuring increase in fluorescein-labelled coactivator PGC-1alpha pe...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor RXR-alpha(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50607785(CHEMBL5219536)
Affinity DataEC50:  5.29E+4nMAssay Description:Agonist activity at RXRalpha-LBD (unknown origin) assessed as transactivation by measuring increase in fluorescein-labelled coactivator PGC-1alpha pe...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetMitogen-activated protein kinase 7(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50434069(CHEMBL2381339 | US9676792, Compound 24)
Affinity DataEC50: >3.00E+4nMAssay Description:Inhibition of GST-tagged full length human ERK5 transfected in HEK293 cells assessed as inhibition of AP1 transcriptional activity after 24 hrs by du...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50434070(CHEMBL2381340)
Affinity DataEC50:  4.20E+3nMAssay Description:Inhibition of GST-tagged full length human ERK5 transfected in HEK293 cells assessed as inhibition of AP1 transcriptional activity after 24 hrs by du...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50383274(CHEMBL1229592 | US9670213, WZ4002 | US10167264, WZ...)
Affinity DataKd:  150nMAssay Description:Binding affinity to JAK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109424(CHEMBL3601107)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109426(CHEMBL3600393)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109427(CHEMBL3601109)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109428(CHEMBL3601110)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109431(CHEMBL3601113)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109432(CHEMBL3601114)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109433(CHEMBL3601116)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109490(CHEMBL3601117)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109527(CHEMBL3601120)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109528(CHEMBL3601115)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109502(CHEMBL3601706)
Affinity DataIC50: 0.580nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109430(CHEMBL3601112)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109492(CHEMBL3601119)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109493(CHEMBL3601121)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109529(CHEMBL3601242)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109425(CHEMBL3601108)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109491(CHEMBL3601118)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109509(CHEMBL3601713)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109519(CHEMBL3601723)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109501(CHEMBL3601705)
Affinity DataIC50: 0.870nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109408(CHEMBL3601227)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109413(CHEMBL3601233)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109522(CHEMBL3601726)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109429(CHEMBL3601111)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109407(CHEMBL3601226)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109508(CHEMBL3601712)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109504(CHEMBL3601708)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109531(CHEMBL3601231)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109412(CHEMBL3601232)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109423(CHEMBL3601106)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109506(CHEMBL3601710)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109421(CHEMBL3601243)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TBK1(Human)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401913(CHEMBL2207214)
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TBK1(Human)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401915(CHEMBL2207212)
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TBK1(Human)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401928(CHEMBL2207195)
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase TBK1(Human)
Mrc Technology

Curated by ChEMBL
LigandPNGBDBM50401907(CHEMBL2207181)
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109409(CHEMBL3601228)
Affinity DataIC50: 2nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50109503(CHEMBL3601707)
Affinity DataIC50: 2nMAssay Description:Inhibition of JAK3 (unknown origin) by Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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