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LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition Protein kinase C (PKC)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142090(2'-(N,N-Dimethyl-carbamimidoyl)-biphenyl-4-carboxy...)
Affinity DataIC50: 0.200nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142163(5-chloro-N-(5-chloropyridin-2-yl)-2-(4-((2-iminoox...)
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142161(5-Chloro-N-(5-chloro-pyridin-2-yl)-2-(4-{[methyl-(...)
Affinity DataIC50: 0.300nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142111(1-{4'-[4-Chloro-2-(5-chloro-pyridin-2-ylcarbamoyl)...)
Affinity DataIC50: 0.400nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249166(2-(azetidin-1-yl)-N-(4-chloro-2-(5-chloropyridin-2...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117334(4-[6,7-Bis-(2-methoxy-ethoxy)-quinazolin-4-yl]-pip...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of wild type Platelet-derived growth factor receptor beta phosphorylation in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117342(4-[6,7-Bis-(2-methoxy-ethoxy)-quinazolin-4-yl]-pip...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of wild type Platelet-derived growth factor receptor beta phosphorylation in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249117(5-chloro-N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimeth...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249118(5-chloro-N-(5-chloropyridin-2-yl)-3-(dimethylamino...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249119(5-chloro-N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimeth...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249121(N-(4-chloro-2-(5-chloropyridin-2-ylcarbamoyl)pheny...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249165(N-(4-chloro-2-(5-chloropyridin-2-ylcarbamoyl)pheny...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193861(5-chloro-N-(5-chloro-pyridin-2-yl)-2-[4-(N,N-dimet...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249327(5-chloro-N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimeth...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249326(5-chloro-N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimeth...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142125(2'-(Acetimidoylamino-methyl)-biphenyl-4-carboxylic...)
Affinity DataIC50: 0.700nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142169(5-Chloro-N-(5-chloro-pyridin-2-yl)-2-[4-(N,N'-dime...)
Affinity DataIC50: 0.700nMAssay Description:In vitro inhibitory activity against coagulation factor X.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249331(5-chloro-N-(4-chlorophenyl)-2-(4-(N,N-dimethylcarb...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193840(1-(2-(4-chloro-2-(5-chloropyridin-2-ylcarbamoyl)ph...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249388(N-(4-chloro-2-(5-chloropyridin-2-ylcarbamoyl)pheny...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249423(N-(2-(5-chloropyridin-2-ylcarbamoyl)-4-methoxyphen...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249116(N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimethylcarbami...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142154({4-[4-Chloro-2-(5-chloro-pyridin-2-ylcarbamoyl)-ph...)
Affinity DataIC50: 0.800nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142178(5-Chloro-N-(5-chloro-pyridin-2-yl)-2-[4-(N,N',N''-...)
Affinity DataIC50: 0.800nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249329(5-chloro-2-(4-(N,N-dimethylcarbamimidoyl)benzamido...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142112(2'-Dimethylamino-biphenyl-4-carboxylic acid [4-chl...)
Affinity DataIC50: 0.900nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142142(5-Chloro-N-(5-chloro-pyridin-2-yl)-2-[4-(N',N'-dim...)
Affinity DataIC50: 0.900nMAssay Description:In vitro inhibitory activity against coagulation factor X.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142177(2-{4-[(Acetimidoyl-methyl-amino)-methyl]-benzoylam...)
Affinity DataIC50: 0.900nMAssay Description:In vitro inhibitory activity against coagulation factor X.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249160(5-chloro-N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimeth...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249360(5-chloro-2-(4-(N,N-dimethylcarbamimidoyl)benzamido...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249123(5-chloro-N-(5-chloropyridin-2-yl)-2-(4-(N-ethyl-N-...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193842(1-(2-(2-(5-chloropyridin-2-ylcarbamoyl)-4-methoxyp...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50140388(2-(6-Chloro-naphthalen-2-yl)-5-methyl-2H-pyrazole-...)
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50140394(2-(6-Chloro-naphthalen-2-yl)-5-methyl-2H-pyrazole-...)
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50140410(2-(6-Chloro-naphthalen-2-yl)-5-trifluoromethyl-2H-...)
Affinity DataIC50: 1nMAssay Description:Binding affinity for human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142129(2'-(4-Hydroxy-piperidin-1-yl)-biphenyl-4-carboxyli...)
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142139(5-Chloro-N-(5-chloro-pyridin-2-yl)-2-{4-[(N-methyl...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249389(2-(azepan-1-yl)-N-(4-chloro-2-(5-chloropyridin-2-y...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249391(N-(4-chloro-2-(5-chloropyridin-2-ylcarbamoyl)pheny...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249156(N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimethylcarbami...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Extracellular signal-regulated kinase 2 (Erk2)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDual specificity mitogen-activated protein kinase kinase 6(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Mitogen activated protein kinase kinase 6More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Mitogen activated protein kinase kinase 4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50117354(4-[6,7-Bis-(2-methoxy-ethoxy)-quinazolin-4-yl]-pip...)
Affinity DataIC50: 1nMAssay Description:Inhibition of wild type Platelet-derived growth factor receptor beta phosphorylation in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142135(2-[4-({[2-(Acetimidoyl-methyl-amino)-ethyl]-methyl...)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249328(5-chloro-2-(4-(N,N-dimethylcarbamimidoyl)benzamido...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249362(5-chloro-N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimeth...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50142126(2'-Guanidinomethyl-biphenyl-4-carboxylic acid [4-c...)
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCoagulation factor X(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50249159(5-chloro-N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimeth...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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