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TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257567(CHEMBL4081244)
Affinity DataEC50:  158nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257518(CHEMBL4063313)
Affinity DataKd:  1.5nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257559(CHEMBL4103808)
Affinity DataKd:  9.20nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257520(CHEMBL4074421)
Affinity DataEC50:  33nMAssay Description:Displacement of [3H]-JNJ46281222 from human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257523(CHEMBL4067298)
Affinity DataEC50:  30nMAssay Description:Displacement of [3H]-JNJ46281222 from human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257525(CHEMBL4091370)
Affinity DataEC50:  5.90nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257596(CHEMBL4060306)
Affinity DataEC50:  30nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257605(CHEMBL4088239)
Affinity DataEC50:  93nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257599(CHEMBL4100691)
Affinity DataKd:  8.10nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257558(CHEMBL4093620)
Affinity DataEC50:  251nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257527(CHEMBL4088960)
Affinity DataEC50:  224nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257554(CHEMBL4075258)
Affinity DataKd:  15nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257524(CHEMBL4080973)
Affinity DataKd:  2.5nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257519(CHEMBL4075417)
Affinity DataKd:  10nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257592(CHEMBL4062535)
Affinity DataEC50:  224nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257595(CHEMBL4087196)
Affinity DataKd:  1.10nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257548(CHEMBL4104081)
Affinity DataEC50:  9.30nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50335255(3'-((2-cyclopentyl-6,7-dimethyl-1-oxo-2,3-dihydro-...)
Affinity DataEC50:  93nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257576(CHEMBL4072262)
Affinity DataEC50:  19nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257546(CHEMBL4064589)
Affinity DataEC50:  19nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257552(CHEMBL4092105)
Affinity DataKd:  100nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257520(CHEMBL4074421)
Affinity DataKd:  13nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257594(CHEMBL4089416)
Affinity DataKd:  13nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257551(CHEMBL4077609)
Affinity DataKd:  3nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257597(CHEMBL4075537)
Affinity DataKd:  16nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257545(CHEMBL4067290)
Affinity DataKd:  12nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257598(CHEMBL4092275)
Affinity DataKd:  20nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257547(CHEMBL4076286)
Affinity DataKd:  54nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257509(CHEMBL4076639)
Affinity DataKd:  10nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257526(CHEMBL4072134)
Affinity DataEC50:  151nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257556(CHEMBL4101354)
Affinity DataEC50:  2.90nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50051571(CHEMBL3337510)
Affinity DataEC50:  79nMAssay Description:Displacement of [3H]-JNJ46281222 from human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257606(CHEMBL4073628)
Affinity DataEC50:  7.80nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257546(CHEMBL4064589)
Affinity DataEC50:  19nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cells assessed as cellular impedance measured for 20 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257555(CHEMBL4074664)
Affinity DataEC50:  12nMAssay Description:Displacement of [3H]-JNJ46281222 from human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257523(CHEMBL4067298)
Affinity DataKd:  2.10nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257524(CHEMBL4080973)
Affinity DataEC50:  8.70nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257559(CHEMBL4103808)
Affinity DataEC50:  56nMAssay Description:Displacement of [3H]-JNJ46281222 from human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257560(CHEMBL4085882)
Affinity DataEC50:  100nMAssay Description:Displacement of [3H]-JNJ46281222 from human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257601(CHEMBL4089955)
Affinity DataEC50:  65nMAssay Description:Displacement of [3H]-JNJ46281222 from human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257518(CHEMBL4063313)
Affinity DataEC50:  1.10nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257600(CHEMBL4066051)
Affinity DataEC50:  17nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257596(CHEMBL4060306)
Affinity DataKd:  6.10nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257593(CHEMBL4067421)
Affinity DataEC50:  17nMAssay Description:Displacement of [3H]-JNJ46281222 from human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes after 60 mins by liquid scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257550(CHEMBL4075762)
Affinity DataKd:  11nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257558(CHEMBL4093620)
Affinity DataKd:  38nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50194618(CHEMBL3937907 | US20240050427, Compound 1)
Affinity DataEC50:  562nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257519(CHEMBL4075417)
Affinity DataEC50:  78nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257598(CHEMBL4092275)
Affinity DataEC50:  148nMAssay Description:Positive allosteric modulation of human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes assessed as increase in glutamate-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50257525(CHEMBL4091370)
Affinity DataKd:  2.90nMAssay Description:Binding affinity to human metabotropic glutamate receptor 2 expressed in CHOK1 cell membranes by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
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