Report error Found 204 with Last Name = 'jacobson' and Initial = 'mp'
Affinity DataEC50: 46nMAssay Description:Modulation of ProLink-fused human CXCR7 expressed in CHOK1 cell membranes assessed as induction of EA-tagged beta-arrestin recruitment after 30 mins ...More data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Modulation of ProLink-fused human CXCR7 expressed in CHOK1 cell membranes assessed as induction of EA-tagged beta-arrestin recruitment after 30 mins ...More data for this Ligand-Target Pair
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco
Curated by ChEMBL
University of California At San Francisco
Curated by ChEMBL
Affinity DataKd: 660nMAssay Description:Binding affinity to human HSC70 after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco
Curated by ChEMBL
University of California At San Francisco
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human HSC70 after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco
Curated by ChEMBL
University of California At San Francisco
Curated by ChEMBL
Affinity DataKd: 2.38E+3nMAssay Description:Binding affinity to human HSC70 Y149A mutant after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco
Curated by ChEMBL
University of California At San Francisco
Curated by ChEMBL
Affinity DataKd: 8.25E+3nMAssay Description:Binding affinity to human HSC70 T222A mutant after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco
Curated by ChEMBL
University of California At San Francisco
Curated by ChEMBL
Affinity DataKd: 1.38E+4nMAssay Description:Binding affinity to human HSC70 L228A mutant after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco
Curated by ChEMBL
University of California At San Francisco
Curated by ChEMBL
Affinity DataKd: 2.43E+4nMAssay Description:Binding affinity to human HSC70 H227A mutant after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
TargetHeat shock cognate 71 kDa protein(Human)
University of California At San Francisco
Curated by ChEMBL
University of California At San Francisco
Curated by ChEMBL
Affinity DataKd: 5.54E+3nMAssay Description:Binding affinity to human HSC70 Y149W mutant after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15B(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataEC50: 600nMAssay Description:Inhibition of human 15-LOX-2 expressed in HEK293T cells assessed as a reduction in 15-HETE production using arachidonic acid as substrate incubated f...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15B(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataEC50: 750nMAssay Description:Inhibition of human 15-LOX-2 expressed in HEK293T cells assessed as a reduction in 15-HETE production using arachidonic acid as substrate incubated f...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15B(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataEC50: 3.10E+4nMAssay Description:Inhibition of human 15-LOX-2 expressed in HEK293T cells assessed as a reduction in 15-HETE production using arachidonic acid as substrate incubated f...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15B(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataEC50: 1.30E+3nMAssay Description:Inhibition of human 15-LOX-2 expressed in HEK293T cells assessed as a reduction in 15-HETE production using arachidonic acid as substrate incubated f...More data for this Ligand-Target Pair
TargetSterol 14-alpha demethylase(Trypanosoma cruzi (strain CL Brener))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataKd: 4.80nMAssay Description:Binding affinity to Trypanosoma cruzi sterol 14-alpha-demethylase by UV-SpectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of CYP3A4 using in human liver microsomes using testosterone as substrate after 5 to 15 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of CYP3A4 using in human liver microsomes using midazolam as substrate after 5 to 15 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of CYP2D6 in human liver microsomes using bufuralol as substrate after 5 to 15 minsMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 Q547L mutant expressed in sf9 cells using arachidonic acid as substrate by UV-Visible spectrophot...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of wild type human N-terminal His6-tagged 15-LOX-1 expressed in sf9 cells using arachidonic acid or linoleic acid as substrate by UV-Visib...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 R402L mutant expressed in sf9 cells using arachidonic acid or linoleic acid as substrate by UV-Vi...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of wild type human N-terminal His-tagged 12-LOX using arachidonic acid as substrate by UV-Vis spectroscopy analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 R404L mutant expressed in sf9 cells using arachidonic acid or linoleic acid as substrate by UV-Vi...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 I417A mutant expressed in sf9 cells using arachidonic acid or linoleic acid as substrate by UV-Vi...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 F414I mutant expressed in sf9 cells using arachidonic acid or linoleic acid as substrate by UV-Vi...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 R402L mutant expressed in sf9 cells using arachidonic acid or linoleic acid as substrate by UV-Vi...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 E356Q mutant expressed in sf9 cells using arachidonic acid as substrate by UV-Visible spectrophot...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 I417A mutant expressed in sf9 cells using arachidonic acid or linoleic acid as substrate by UV-Vi...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 F414W mutant expressed in sf9 cells using arachidonic acid as substrate by UV-Visible spectrophot...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of N-terminal His6-tagged human 12/15-LOX using arachidonic acid as substrate by UV-visible spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 205nMAssay Description:Inhibition of CYP2C9 in human liver microsomes using tolbutamide as substrate after 5 to 15 minsMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 R404L mutant expressed in sf9 cells using arachidonic acid or linoleic acid as substrate by UV-Vi...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 Q547L mutant expressed in sf9 cells using arachidonic acid as substrate by UV-Visible spectrophot...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of wild type human N-terminal His6-tagged 15-LOX-1 expressed in sf9 cells using arachidonic acid or linoleic acid as substrate by UV-Visib...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15B(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of human 15-LOX-2 assessed as enzymatic rate using arachidonic acid as substrate by UV/Vis spectrophotometric analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of wild type human N-terminal His-tagged 12-LOX using arachidonic acid as substrate by UV-Vis spectroscopy analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 L407A mutant expressed in sf9 cells using arachidonic acid as substrate by UV-Visible spectrophot...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15B(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of human 15-LOX-2 assessed as enzymatic rate using arachidonic acid as substrate by UV/Vis spectrophotometric analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 770nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 F414W mutant expressed in sf9 cells using arachidonic acid as substrate by UV-Visible spectrophot...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 810nMAssay Description:Inhibition of human 12/15-LOX expressed in HEK293 cells after 30 mins by microplate reader analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 870nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 E356Q mutant expressed in sf9 cells using arachidonic acid as substrate by UV-Visible spectrophot...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15B(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 870nMAssay Description:Inhibition of human 15-LOX-2 assessed as enzymatic rate using arachidonic acid as substrate by UV/Vis spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of CYP2C8 in human liver microsomes using paclitaxel as substrate after 5 to 15 minsMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15B(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human 15-LOX-2 assessed as enzymatic rate using arachidonic acid as substrate by UV/Vis spectrophotometric analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15B(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human 15-LOX-2 assessed as enzymatic rate using arachidonic acid as substrate by UV/Vis spectrophotometric analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of N-terminal His6-tagged human 12/15-LOX using arachidonic acid as substrate by UV-visible spectrophotometric analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of N-terminal His6-tagged human 12/15-LOX using arachidonic acid as substrate by UV-visible spectrophotometric analysisMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human N-terminal His6-tagged 15-LOX-1 F414I mutant expressed in sf9 cells using arachidonic acid or linoleic acid as substrate by UV-Vi...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of N-terminal His6-tagged human 12/15-LOX using arachidonic acid as substrate by UV-visible spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 6.29E+3nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate after 5 to 15 minsMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid lipoxygenase ALOX15(Human)
University of California Santa Cruz
Curated by ChEMBL
University of California Santa Cruz
Curated by ChEMBL
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of N-terminal His6-tagged human 12/15-LOX using arachidonic acid as substrate by UV-visible spectrophotometric analysisMore data for this Ligand-Target Pair
