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TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508101(CHEMBL4521388)
Affinity DataEC50:  1.66E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508102(CHEMBL4537335)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508103(CHEMBL4589453)
Affinity DataEC50:  2.25E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508104(CHEMBL4591405)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508105(CHEMBL4542891)
Affinity DataEC50:  730nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508106(CHEMBL4517263)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508107(CHEMBL4574542)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508108(CHEMBL4567211)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508109(CHEMBL4592935)
Affinity DataEC50:  1.03E+4nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508110(CHEMBL4444760)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508111(CHEMBL4520827)
Affinity DataEC50:  460nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508113(CHEMBL4453360)
Affinity DataEC50:  2.72E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508114(CHEMBL4466241)
Affinity DataEC50:  1.32E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508115(CHEMBL4469751)
Affinity DataEC50:  1.81E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508116(CHEMBL4535401)
Affinity DataEC50:  2.78E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508117(CHEMBL4463602)
Affinity DataEC50:  2.53E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508118(CHEMBL4436393)
Affinity DataEC50:  7.36E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508119(CHEMBL4472191)
Affinity DataEC50:  1.23E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508120(CHEMBL4531918)
Affinity DataEC50:  2.62E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508121(CHEMBL4527893)
Affinity DataEC50:  2.36E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508122(CHEMBL4456647)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508123(CHEMBL4452865)
Affinity DataEC50:  3.31E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508112(CHEMBL4546437)
Affinity DataEC50:  1.73E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508124(CHEMBL4443588)
Affinity DataEC50:  1.53E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535728(CHEMBL4556396)
Affinity DataEC50:  2.55E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535729(CHEMBL4541559)
Affinity DataEC50:  3.39E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535730(CHEMBL4550608)
Affinity DataEC50:  1.05E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535731(CHEMBL4435259)
Affinity DataEC50:  4.25E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535732(CHEMBL4448988)
Affinity DataEC50:  2.41E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535733(CHEMBL4447835)
Affinity DataEC50:  1.48E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535734(CHEMBL4444888)
Affinity DataEC50:  1.32E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535735(CHEMBL4440354)
Affinity DataEC50:  1.38E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535736(CHEMBL4468084)
Affinity DataEC50:  4.21E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535737(CHEMBL4546069)
Affinity DataEC50:  280nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535738(CHEMBL4463957)
Affinity DataEC50:  1.14E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535739(CHEMBL4468637)
Affinity DataEC50:  1.39E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535740(CHEMBL4465311)
Affinity DataEC50:  590nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50535741(CHEMBL4464717)
Affinity DataEC50:  1.75E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) assessed as receptor transactivation after 24 hrs by TK-PPRE-Luc expressing cells based luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50581458(CHEMBL5092802)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human recombinant glutaminyl cyclase using H-Gln-AMC hydrobromide as substrate measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50581397(CHEMBL5085353)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human recombinant glutaminyl cyclase using H-Gln-AMC hydrobromide as substrate measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50581442(CHEMBL5086776)
Affinity DataIC50: 0.460nMAssay Description:Inhibition of human recombinant glutaminyl cyclase using H-Gln-AMC hydrobromide as substrate measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50581399(CHEMBL5085226)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human recombinant glutaminyl cyclase using H-Gln-AMC hydrobromide as substrate measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50581400(CHEMBL5075575)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human recombinant glutaminyl cyclase using H-Gln-AMC hydrobromide as substrate measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50581426(CHEMBL5089771)
Affinity DataIC50: 0.710nMAssay Description:Inhibition of human recombinant glutaminyl cyclase using H-Gln-AMC hydrobromide as substrate measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50581398(CHEMBL5083519)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human recombinant glutaminyl cyclase using H-Gln-AMC hydrobromide as substrate measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50581412(CHEMBL5088732)
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant glutaminyl cyclase using H-Gln-AMC hydrobromide as substrate measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50581450(CHEMBL5085670)
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant glutaminyl cyclase using H-Gln-AMC hydrobromide as substrate measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50581445(CHEMBL5089285)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human recombinant glutaminyl cyclase using H-Gln-AMC hydrobromide as substrate measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508111(CHEMBL4520827)
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50581441(CHEMBL5081653)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human recombinant glutaminyl cyclase using H-Gln-AMC hydrobromide as substrate measured after 15 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
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