Compile Data Set for Download or QSAR
Found 645 with Last Name = 'jong' and Initial = 'l'
TargetNociceptin receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM21842((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-[(2S)-6-amino-2-[(2...)
Affinity DataKi:  0.0600nMAssay Description:Binding affinity for human nociceptin (NOP) receptor using [3H]N/OFQ as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137564(1'-(4-isopropylcyclohexyl)-2-methyl-5-phenyl-(3aR,...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity for human nociceptin (NOP) receptor using [3H]N/OFQ as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137565(1-((2R,6S,9aR)-6-Phenyl-octahydro-quinolizin-2-yl)...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity for human opioid receptor kappa 1 using [3H]- U-69,593 as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137567(1-((2R,6S,9aR)-6-Cyclohexyl-octahydro-quinolizin-2...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity for human opioid receptor kappa 1 using [3H]- U-69,593 as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137566(1-Ethyl-3-((2R,6S,9aR)-6-phenyl-octahydro-quinoliz...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity for human opioid receptor mu 1 using [3H]- DAMGO as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137565(1-((2R,6S,9aR)-6-Phenyl-octahydro-quinolizin-2-yl)...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity for human opioid receptor mu 1 using [3H]- DAMGO as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137565(1-((2R,6S,9aR)-6-Phenyl-octahydro-quinolizin-2-yl)...)
Affinity DataKi:  5.70nMAssay Description:Binding affinity for human nociceptin (NOP) receptor using [3H]N/OFQ as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137563(1-Ethyl-3-((2S,6S,9aR)-6-phenyl-octahydro-quinoliz...)
Affinity DataKi:  18nMAssay Description:Binding affinity for human opioid receptor mu 1 using [3H]- DAMGO as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137566(1-Ethyl-3-((2R,6S,9aR)-6-phenyl-octahydro-quinoliz...)
Affinity DataKi:  20nMAssay Description:Binding affinity for human nociceptin (NOP) receptor using [3H]N/OFQ as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137566(1-Ethyl-3-((2R,6S,9aR)-6-phenyl-octahydro-quinoliz...)
Affinity DataKi:  23nMAssay Description:Binding affinity for human opioid receptor kappa 1 using [3H]- U-69,593 as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137567(1-((2R,6S,9aR)-6-Cyclohexyl-octahydro-quinolizin-2...)
Affinity DataKi:  29nMAssay Description:Binding affinity for human nociceptin (NOP) receptor using [3H]N/OFQ as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137567(1-((2R,6S,9aR)-6-Cyclohexyl-octahydro-quinolizin-2...)
Affinity DataKi:  47nMAssay Description:Binding affinity for human opioid receptor mu 1 using [3H]- DAMGO as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137561(1-((2S,6S,9aR)-6-Phenyl-octahydro-quinolizin-2-yl)...)
Affinity DataKi:  48nMAssay Description:Binding affinity for human opioid receptor mu 1 using [3H]- DAMGO as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137568(1-((2S,6S,9aR)-6-Cyclohexyl-octahydro-quinolizin-2...)
Affinity DataKi:  119nMAssay Description:Binding affinity for human opioid receptor mu 1 using [3H]- DAMGO as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137568(1-((2S,6S,9aR)-6-Cyclohexyl-octahydro-quinolizin-2...)
Affinity DataKi:  189nMAssay Description:Binding affinity for human nociceptin (NOP) receptor using [3H]N/OFQ as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137568(1-((2S,6S,9aR)-6-Cyclohexyl-octahydro-quinolizin-2...)
Affinity DataKi:  227nMAssay Description:Binding affinity for human opioid receptor kappa 1 using [3H]- U-69,593 as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137561(1-((2S,6S,9aR)-6-Phenyl-octahydro-quinolizin-2-yl)...)
Affinity DataKi:  271nMAssay Description:Binding affinity for human opioid receptor kappa 1 using [3H]- U-69,593 as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137563(1-Ethyl-3-((2S,6S,9aR)-6-phenyl-octahydro-quinoliz...)
Affinity DataKi:  535nMAssay Description:Binding affinity for human nociceptin (NOP) receptor using [3H]N/OFQ as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137561(1-((2S,6S,9aR)-6-Phenyl-octahydro-quinolizin-2-yl)...)
Affinity DataKi:  786nMAssay Description:Binding affinity for human nociceptin (NOP) receptor using [3H]N/OFQ as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137563(1-Ethyl-3-((2S,6S,9aR)-6-phenyl-octahydro-quinoliz...)
Affinity DataKi:  987nMAssay Description:Binding affinity for human opioid receptor kappa 1 using [3H]- U-69,593 as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137566(1-Ethyl-3-((2R,6S,9aR)-6-phenyl-octahydro-quinoliz...)
Affinity DataKi:  1.49E+3nMAssay Description:Binding affinity for human opioid receptor delta 1 using [3H]- CL-DPDPE as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137565(1-((2R,6S,9aR)-6-Phenyl-octahydro-quinolizin-2-yl)...)
Affinity DataKi:  1.72E+3nMAssay Description:Binding affinity for human opioid receptor delta 1 using [3H]- CL-DPDPE as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137563(1-Ethyl-3-((2S,6S,9aR)-6-phenyl-octahydro-quinoliz...)
Affinity DataKi:  1.84E+3nMAssay Description:Binding affinity for human opioid receptor delta 1 using [3H]- CL-DPDPE as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137567(1-((2R,6S,9aR)-6-Cyclohexyl-octahydro-quinolizin-2...)
Affinity DataKi:  2.08E+3nMAssay Description:Binding affinity for human opioid receptor delta 1 using [3H]- CL-DPDPE as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate racemase(Helicobacter pylori)
AstraZeneca Global Structural Chemistry

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibition of Helicobacter pylori glutamate racemaseMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137568(1-((2S,6S,9aR)-6-Cyclohexyl-octahydro-quinolizin-2...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human opioid receptor delta 1 using [3H]- CL-DPDPE as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
SRI International

Curated by ChEMBL
LigandPNGBDBM50137561(1-((2S,6S,9aR)-6-Phenyl-octahydro-quinolizin-2-yl)...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for human opioid receptor delta 1 using [3H]- CL-DPDPE as radioligand transfected into CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548859(WO2022098806, Compound 2-120)
Affinity DataIC50:  0.0100nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548828(WO2022098806, Compound 2-89)
Affinity DataIC50:  0.0100nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548847(WO2022098806, Compound 2-108)
Affinity DataIC50:  0.0100nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548860(WO2022098806, Compound 2-121)
Affinity DataIC50:  0.0200nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548834(WO2022098806, Compound 2-180 | WO2022098806, Compo...)
Affinity DataIC50:  0.0200nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548817(WO2022098806, Compound 2-78)
Affinity DataIC50:  0.0200nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548823(WO2022098806, Compound 2-84)
Affinity DataIC50:  0.0200nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548829(WO2022098806, Compound 2-179 | WO2022098806, Compo...)
Affinity DataIC50:  0.0200nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548850(WO2022098806, Compound 2-111)
Affinity DataIC50:  0.0200nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548727(WO2022098806, Compound 1-123)
Affinity DataIC50:  0.0200nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548846(WO2022098806, Compound 2-107 | WO2022098806, Compo...)
Affinity DataIC50:  0.0300nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548867(WO2022098806, Compound 2-128)
Affinity DataIC50:  0.0300nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548897(WO2022098806, Compound 2-158)
Affinity DataIC50:  0.0300nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548863(WO2022098806, Compound 2-124 | WO2022098806, Compo...)
Affinity DataIC50:  0.0300nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548914(WO2022098806, Compound 2-175)
Affinity DataIC50:  0.0300nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548815(WO2022098806, Compound 2-76)
Affinity DataIC50:  0.0300nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548818(WO2022098806, Compound 2-79)
Affinity DataIC50:  0.0300nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548821(WO2022098806, Compound 2-82)
Affinity DataIC50:  0.0300nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548824(WO2022098806, Compound 2-85)
Affinity DataIC50:  0.0300nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548922(WO2022098806, Compound 2-183)
Affinity DataIC50:  0.0400nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548858(WO2022098806, Compound 2-119)
Affinity DataIC50:  0.0400nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548763(WO2022098806, Compound 2-114 | WO2022098806, Compo...)
Affinity DataIC50:  0.0400nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 1(Homo sapiens (Human))
MERCK SHARP & DOHME LLC

WIPO
LigandPNGBDBM548878(WO2022098806, Compound 2-139)
Affinity DataIC50:  0.0400nMAssay Description: To each well of black Corning #3820384-well plate, an ECHO was used to dispense 7.5 nL of DMSO or Test compound in DMSO. A 1.5x kinase solution, 5 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Displayed 1 to 50 (of 645 total ) | Next | Last >>
Jump to: