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TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268927(CHEMBL4105014)
Affinity DataEC50:  53nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268928(CHEMBL4097314)
Affinity DataEC50:  67nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268929(CHEMBL4087235)
Affinity DataEC50:  64nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268930(CHEMBL4064998)
Affinity DataEC50:  199nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268931(CHEMBL4099911)
Affinity DataEC50:  57nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268932(CHEMBL4081913)
Affinity DataEC50:  105nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268933(CHEMBL4093173)
Affinity DataEC50:  319nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268939(CHEMBL4061409)
Affinity DataEC50:  155nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268940(CHEMBL4087173)
Affinity DataEC50:  321nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268941(CHEMBL4066367)
Affinity DataEC50:  171nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268942(CHEMBL4061666)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268943(CHEMBL4089778)
Affinity DataEC50:  77nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268944(CHEMBL4070332)
Affinity DataEC50:  92nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268945(CHEMBL4105139)
Affinity DataEC50:  156nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268955(CHEMBL4078440)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Korea Research Institute of Chemical Technology

Curated by ChEMBL
LigandPNGBDBM50268956(CHEMBL4067537)
Affinity DataEC50:  98nMAssay Description:Agonist activity at human GPR119 expressed in CHOK1 cells harboring CRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/8/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50285942(CHEMBL4169194)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286055(CHEMBL4171474)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286056(CHEMBL4172104)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286057(CHEMBL4172579)
Affinity DataEC50:  60nMAssay Description:Agonist activity at recombinant rat CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286058(CHEMBL4161506)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at recombinant human CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286055(CHEMBL4171474)
Affinity DataEC50:  59nMAssay Description:Agonist activity at recombinant human CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286059(CHEMBL4164926)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286056(CHEMBL4172104)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at recombinant human CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286058(CHEMBL4161506)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286056(CHEMBL4172104)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at recombinant rat CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286060(CHEMBL4161266)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286058(CHEMBL4161506)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286061(CHEMBL4166597)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286055(CHEMBL4171474)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286062(CHEMBL4168131)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286057(CHEMBL4172579)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286063(CHEMBL4164688)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286064(CHEMBL4174510)
Affinity DataEC50:  840nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286056(CHEMBL4172104)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286065(CHEMBL4175548)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286059(CHEMBL4164926)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286065(CHEMBL4175548)
Affinity DataEC50:  5.90nMAssay Description:Agonist activity at recombinant human CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286061(CHEMBL4166597)
Affinity DataEC50:  3.80nMAssay Description:Agonist activity at recombinant human CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286064(CHEMBL4174510)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at recombinant human CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286063(CHEMBL4164688)
Affinity DataEC50:  17nMAssay Description:Agonist activity at recombinant human CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286057(CHEMBL4172579)
Affinity DataEC50:  105nMAssay Description:Agonist activity at recombinant human CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286062(CHEMBL4168131)
Affinity DataEC50:  46nMAssay Description:Agonist activity at recombinant human CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286066(CHEMBL4162987)
Affinity DataEC50:  26nMAssay Description:Agonist activity at recombinant human CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50040961(CHEMBL3354952)
Affinity DataEC50:  64nMAssay Description:Agonist activity at recombinant human CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286066(CHEMBL4162987)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286067(CHEMBL4160855)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286062(CHEMBL4168131)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286057(CHEMBL4172579)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286063(CHEMBL4164688)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
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