Compile Data Set for Download or QSAR
Report error Found 6081 with Last Name = 'kim' and Initial = 'sh'
LigandPNGBDBM28776((3E)-3-(methoxyimino)-2-({4-[2-(5-methyl-2-phenyl-...)
Affinity DataEC50:  2.10nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28777((3E)-3-(ethoxyimino)-2-({4-[2-(5-methyl-2-phenyl-1...)
Affinity DataEC50:  1nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28778((3E)-2-({4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)e...)
Affinity DataEC50:  0.550nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28779((3E)-2-({4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)e...)
Affinity DataEC50:  0.300nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28780((3E)-3-(butoxyimino)-2-({4-[2-(5-methyl-2-phenyl-1...)
Affinity DataEC50:  0.190nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28781((3E)-3-[(cyclopropylmethoxy)imino]-2-({4-[2-(5-met...)
Affinity DataEC50:  0.360nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28782((3E)-3-(methoxyimino)-2-({4-[2-(5-methyl-2-phenyl-...)
Affinity DataEC50:  0.310nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28783(E/Z=4/1 | (3E)-3-(ethoxyimino)-2-({4-[2-(5-methyl-...)
Affinity DataEC50:  0.100nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28784((3E)-3-{[(4-fluorophenyl)methoxy]imino}-2-({4-[2-(...)
Affinity DataEC50:  0.540nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28785((3Z)-3-{[(4-fluorophenyl)methoxy]imino}-2-({4-[2-(...)
Affinity DataEC50:  5nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28786((3E)-3-(ethoxyimino)-2-({4-[(5-methyl-2-phenyl-1,3...)
Affinity DataEC50:  4nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28787((3E)-2-({4-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)met...)
Affinity DataEC50:  13nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28788((3E)-3-(ethoxyimino)-2-[(4-{[2-(4-fluorophenyl)-5-...)
Affinity DataEC50:  6.80nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28789((3E)-2-[(4-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazo...)
Affinity DataEC50:  28nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28790((3E)-3-[(2-fluoroethoxy)imino]-2-[(4-{[2-(4-fluoro...)
Affinity DataEC50:  7.70nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28791((3E)-3-(ethoxyimino)-2-[(4-{2-[2-(4-fluorophenyl)-...)
Affinity DataEC50:  3nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28792((3E)-2-[(4-{2-[2-(4-fluorophenyl)-5-methyl-1,3-oxa...)
Affinity DataEC50:  2.10nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28793((3E)-3-[(2-fluoroethoxy)imino]-2-[(4-{2-[2-(4-fluo...)
Affinity DataEC50:  2.90nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28794(E/Z=5/1 | (3E)-3-(ethoxyimino)-2-[(4-{[5-methyl-2-...)
Affinity DataEC50:  48nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28795(E/Z=5/1 | (3E)-2-[(4-{[5-methyl-2-(propan-2-yl)-1,...)
Affinity DataEC50:  5nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28796((3E)-3-(ethoxyimino)-2-[(4-{2-[5-methyl-2-(propan-...)
Affinity DataEC50:  20nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28797((3E)-2-[(4-{2-[5-methyl-2-(propan-2-yl)-1,3-oxazol...)
Affinity DataEC50:  5.20nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  82nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataEC50:  3.53E+3nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28776((3E)-3-(methoxyimino)-2-({4-[2-(5-methyl-2-phenyl-...)
Affinity DataEC50:  19nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28777((3E)-3-(ethoxyimino)-2-({4-[2-(5-methyl-2-phenyl-1...)
Affinity DataEC50:  12nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28778((3E)-2-({4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)e...)
Affinity DataEC50:  4.90nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28779((3E)-2-({4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)e...)
Affinity DataEC50:  2.20nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28780((3E)-3-(butoxyimino)-2-({4-[2-(5-methyl-2-phenyl-1...)
Affinity DataEC50:  1.30nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28781((3E)-3-[(cyclopropylmethoxy)imino]-2-({4-[2-(5-met...)
Affinity DataEC50:  3.10nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28782((3E)-3-(methoxyimino)-2-({4-[2-(5-methyl-2-phenyl-...)
Affinity DataEC50:  32nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28783(E/Z=4/1 | (3E)-3-(ethoxyimino)-2-({4-[2-(5-methyl-...)
Affinity DataEC50:  26nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28784((3E)-3-{[(4-fluorophenyl)methoxy]imino}-2-({4-[2-(...)
Affinity DataEC50:  10.6nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28785((3Z)-3-{[(4-fluorophenyl)methoxy]imino}-2-({4-[2-(...)
Affinity DataEC50:  596nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28786((3E)-3-(ethoxyimino)-2-({4-[(5-methyl-2-phenyl-1,3...)
Affinity DataEC50:  91nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28787((3E)-2-({4-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)met...)
Affinity DataEC50:  19nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28788((3E)-3-(ethoxyimino)-2-[(4-{[2-(4-fluorophenyl)-5-...)
Affinity DataEC50:  12nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28789((3E)-2-[(4-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazo...)
Affinity DataEC50:  11.7nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28790((3E)-3-[(2-fluoroethoxy)imino]-2-[(4-{[2-(4-fluoro...)
Affinity DataEC50:  23nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28791((3E)-3-(ethoxyimino)-2-[(4-{2-[2-(4-fluorophenyl)-...)
Affinity DataEC50:  11.5nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28792((3E)-2-[(4-{2-[2-(4-fluorophenyl)-5-methyl-1,3-oxa...)
Affinity DataEC50:  4nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28793((3E)-3-[(2-fluoroethoxy)imino]-2-[(4-{2-[2-(4-fluo...)
Affinity DataEC50:  3.5nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28794(E/Z=5/1 | (3E)-3-(ethoxyimino)-2-[(4-{[5-methyl-2-...)
Affinity DataEC50:  1.24E+3nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28795(E/Z=5/1 | (3E)-2-[(4-{[5-methyl-2-(propan-2-yl)-1,...)
Affinity DataEC50:  105nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28796((3E)-3-(ethoxyimino)-2-[(4-{2-[5-methyl-2-(propan-...)
Affinity DataEC50:  139nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28797((3E)-2-[(4-{2-[5-methyl-2-(propan-2-yl)-1,3-oxazol...)
Affinity DataEC50:  10nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataEC50:  9.80E+3nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  78nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. EC50 is the concentration...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Crinetics Pharmaceuticals

US Patent
LigandPNGBDBM405553(US10351547, Compound 1-1 | US10597377, Compound 1-...)
Affinity DataEC50: <10nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC #CCL-61) stably expressing the human SSTR2 are plated in each well of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2020
Entry Details
Go to US Patent

TargetSomatostatin receptor type 2(Human)
Crinetics Pharmaceuticals

US Patent
LigandPNGBDBM405554(US10351547, Compound 1-2 | US10597377, Compound 1-...)
Affinity DataEC50: <10nMAssay Description:Four days prior to the assay, 5,000 Chinese hamster ovary cells (CHO-K1, ATCC #CCL-61) stably expressing the human SSTR2 are plated in each well of a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2020
Entry Details
Go to US Patent

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