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TargetHeat shock-related 70 kDa protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA2 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 6(Homo sapiens)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA6 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetVasopressin V1b receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50044777(CHEBI:34543 | Arginine Vasopressin | Beta-Hypopham...)
Affinity DataEC50:  11nMAssay Description:Activation of human 3X-HA N-tagged AVP1b expressed in CHO-K1 cells incubated for 10 mins by cell Western assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd:  334nMAssay Description:Binding affinity to HspA5 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetOxytocin receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50406327(CHEMBL5281925)
Affinity DataEC50:  3.80E+3nMAssay Description:Activation of human 3X-HA N-tagged OTR expressed in CHO-K1 cells incubated for 10 mins by cell Western assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetVasopressin V1a receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50044777(CHEBI:34543 | Arginine Vasopressin | Beta-Hypopham...)
Affinity DataEC50:  32nMAssay Description:Activation of human 3X-HA N-tagged AVP1a expressed in CHO-K1 cells incubated for 10 mins by cell Western assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
PubMed
TargetOxytocin receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50406325(CHEMBL5279634)
Affinity DataEC50:  160nMAssay Description:Activation of human 3X-HA N-tagged OTR expressed in CHO-K1 cells incubated for 10 mins by cell Western assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxytocin receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50406330(CHEMBL5271164)
Affinity DataEC50:  220nMAssay Description:Activation of human 3X-HA N-tagged OTR expressed in CHO-K1 cells incubated for 10 mins by cell Western assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxytocin receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50406324(CHEMBL5275543)
Affinity DataEC50:  0.730nMAssay Description:Activation of human 3X-HA N-tagged OTR expressed in CHO-K1 cells incubated for 10 mins by cell Western assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxytocin receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50406329(CHEMBL5273426)
Affinity DataEC50:  0.540nMAssay Description:Activation of human 3X-HA N-tagged OTR expressed in CHO-K1 cells incubated for 10 mins by cell Western assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetStress-70 protein, mitochondrial(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd:  7.48E+3nMAssay Description:Binding affinity to HspA9 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetOxytocin receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50406331(CHEMBL5286119)
Affinity DataEC50:  0.0600nMAssay Description:Activation of human 3X-HA N-tagged OTR expressed in CHO-K1 cells incubated for 10 mins by cell Western assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetOxytocin receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50406326(CHEMBL5280014)
Affinity DataEC50:  0.280nMAssay Description:Activation of human 3X-HA N-tagged OTR expressed in CHO-K1 cells incubated for 10 mins by cell Western assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA8 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetOxytocin receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  2.30nMAssay Description:Activation of human 3X-HA N-tagged OTR expressed in CHO-K1 cells incubated for 10 mins by cell Western assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA1A (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetOxytocin receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50406328(CHEMBL5266871)
Affinity DataEC50:  7.00E+3nMAssay Description:Activation of human 3X-HA N-tagged OTR expressed in CHO-K1 cells incubated for 10 mins by cell Western assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1-like(Homo sapiens)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA1L (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50008984(N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionami...)
Affinity DataIC50: 1.90nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum/longitudinal muscle with myenteric plexus assessed as inhibition of PL-017-induced...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50008984(N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionami...)
Affinity DataIC50: 7.20nMAssay Description:Agonist activity at delta opioid receptor in ICR mouse vas deferens assessed as inhibition of MVD contraction heightMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50355375(CHEMBL1835844)
Affinity DataIC50: 55nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum/longitudinal muscle with myenteric plexus assessed as inhibition of PL-017-induced...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50355374(CHEMBL1835843)
Affinity DataIC50: 410nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum/longitudinal muscle with myenteric plexus assessed as inhibition of PL-017-induced...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617288(CHEMBL5410116)
Affinity DataIC50: 500nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617266(CHEMBL5418499)
Affinity DataIC50: 500nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 6(Homo sapiens)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617288(CHEMBL5410116)
Affinity DataIC50: 500nMAssay Description:Inhibition of HspA6 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617268(CHEMBL5415571)
Affinity DataIC50: 500nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617261(CHEMBL5414287)
Affinity DataIC50: 590nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617277(CHEMBL5419391)
Affinity DataIC50: 700nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetHeat shock-related 70 kDa protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617288(CHEMBL5410116)
Affinity DataIC50: 700nMAssay Description:Inhibition of HspA2 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617276(CHEMBL5403845)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617282(CHEMBL5425293)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617273(CHEMBL5409255)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617258(CHEMBL5424525)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617258(CHEMBL5424525)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of FAM-labeled NRLLLTG binding from HspA5 (unknown origin) in presence of ATP by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617267(CHEMBL5410567)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617271(CHEMBL5407447)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetStress-70 protein, mitochondrial(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617261(CHEMBL5414287)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of HspA9 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetHeat shock-related 70 kDa protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617273(CHEMBL5409255)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of HspA2 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617260(CHEMBL5433282)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617275(CHEMBL5437667)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetHeat shock-related 70 kDa protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617272(CHEMBL5435048)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of HspA2 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617274(CHEMBL5422252)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617257(CHEMBL5308000)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of FAM-labeled NRLLLTG binding from HspA5 (unknown origin) in presence of ATP by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617288(CHEMBL5410116)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of HspA8 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetStress-70 protein, mitochondrial(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617258(CHEMBL5424525)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of HspA9 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617272(CHEMBL5435048)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617259(CHEMBL5422755)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetStress-70 protein, mitochondrial(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617260(CHEMBL5433282)
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of HspA9 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetHeat shock-related 70 kDa protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617261(CHEMBL5414287)
Affinity DataIC50: 1.39E+4nMAssay Description:Inhibition of HspA2 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetStress-70 protein, mitochondrial(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617272(CHEMBL5435048)
Affinity DataIC50: 1.43E+4nMAssay Description:Inhibition of HspA9 (unknown origin) by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
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