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TargetAtypical chemokine receptor 3(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50288843(CHEMBL4176134)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human CXCR7 expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment by chemiluminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2020
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50288838(CHEMBL4174297)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human CXCR7 expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment by chemiluminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2020
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50288833(CHEMBL4173913)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human CXCR7 expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment by chemiluminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2020
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50288844(CHEMBL4168948)
Affinity DataEC50:  3.97E+3nMAssay Description:Agonist activity at human CXCR7 expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment by chemiluminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2020
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50288837(CHEMBL4165525)
Affinity DataEC50:  7.81E+3nMAssay Description:Agonist activity at human CXCR7 expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment by chemiluminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2020
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50288846(CHEMBL4163618)
Affinity DataEC50:  1.05E+4nMAssay Description:Agonist activity at human CXCR7 expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment by chemiluminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2020
Entry Details Article
PubMed
TargetAtypical chemokine receptor 3(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50288842(CHEMBL4161021)
Affinity DataEC50:  5.92E+3nMAssay Description:Agonist activity at human CXCR7 expressed in CHOK1 cells assessed as induction of beta-arrestin recruitment by chemiluminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2020
Entry Details Article
PubMed
TargetCathepsin D(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 0.173nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetCathepsin E(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 0.181nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055512(CHEMBL3317812)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055513(CHEMBL3317811)
Affinity DataIC50: 0.210nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055514(CHEMBL3317810)
Affinity DataIC50: 0.290nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetCathepsin E(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50302109(Grassystatin B | CHEMBL568553)
Affinity DataIC50: 0.354nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055513(CHEMBL3317811)
Affinity DataIC50: 0.380nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50020912(Largazole Thiol)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055515(CHEMBL3317818)
Affinity DataIC50: 0.620nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055514(CHEMBL3317810)
Affinity DataIC50: 0.680nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50020912(Largazole Thiol)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetCathepsin E(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50302107(Grassystatin A | CHEMBL567893)
Affinity DataIC50: 0.886nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50020912(Largazole Thiol)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055516(CHEMBL3317817)
Affinity DataIC50: 0.960nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055512(CHEMBL3317812)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055515(CHEMBL3317818)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055513(CHEMBL3317811)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055515(CHEMBL3317818)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055516(CHEMBL3317817)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055512(CHEMBL3317812)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055514(CHEMBL3317810)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055516(CHEMBL3317817)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055517(CHEMBL3317816)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055517(CHEMBL3317816)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055518(CHEMBL3317815)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055517(CHEMBL3317816)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetCathepsin E(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 5nMAssay Description:Inhibition of cathepsin E in human MCF7 cells by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetCathepsin D(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 5nMAssay Description:Inhibition of cathepsin D in human MCF7 cells by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055510(CHEMBL3317814)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055518(CHEMBL3317815)
Affinity DataIC50: 6nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055518(CHEMBL3317815)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055510(CHEMBL3317814)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetChymase(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50288847(Chymostatin)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of chymase (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2020
Entry Details Article
PubMed
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 13nMAssay Description:Inhibition of TACE after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055510(CHEMBL3317814)
Affinity DataIC50: 21nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetCathepsin D(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50302107(Grassystatin A | CHEMBL567893)
Affinity DataIC50: 27nMAssay Description:Inhibition of cathepsin DMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 1(Pig)
Smithsonian Marine Station At Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50312532(molassamide | CHEMBL1077010)
Affinity DataIC50: 32nMAssay Description:Inhibition of pig pancreatic elastase preincubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055511(CHEMBL3317813)
Affinity DataIC50: 39nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetCathepsin E(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50302108(Grassystatin C | CHEMBL569445)
Affinity DataIC50: 43nMAssay Description:Inhibition of cathepsin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 56nMAssay Description:Inhibition of ADAM9 after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 56nMAssay Description:Inhibition of ADAM9 after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50055511(CHEMBL3317813)
Affinity DataIC50: 100nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Duke University

Curated by ChEMBL
LigandPNGBDBM50020912(Largazole Thiol)
Affinity DataIC50: 102nMAssay Description:Inhibition of HDAC8 (unknown origin) incubated at 37 degC for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
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