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TargetIsoform Bcl-X(L) of Bcl-2-like protein 1 (Bcl-xL)(Human)
Walter and Eliza Hall Institute of Medical Research

LigandPNGBDBM50436643(CHEMBL2398292 | 3-(5-(1-(2-(Benzo[d]thiazol-2-yl)h...)
Affinity DataKd:  850nMpH: 2.2 T: 2°CAssay Description:A concentration series of each compound was injected at a flow rate of 90 µL/min over three spots at 25°C. The times allowed for compound a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2014
Entry Details Article
PubMed
TargetIsoform Bcl-X(L) of Bcl-2-like protein 1 (Bcl-xL)(Human)
Walter and Eliza Hall Institute of Medical Research

LigandPNGBDBM109231(N-(3-(5-(1-(2-(Benzo[d]thiazol-2-yl)hydrazono)ethy...)
Affinity DataKd:  230nMpH: 2.2 T: 2°CAssay Description:A concentration series of each compound was injected at a flow rate of 90 µL/min over three spots at 25°C. The times allowed for compound a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2014
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242755(CHEMBL4101006)
Affinity DataEC50:  120nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242756(CHEMBL4083023)
Affinity DataEC50:  80nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242757(CHEMBL4090814)
Affinity DataEC50:  100nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242758(CHEMBL4085525)
Affinity DataEC50:  100nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242759(CHEMBL4063950)
Affinity DataEC50:  100nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242767(CHEMBL4072542)
Affinity DataEC50:  3.10E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242768(CHEMBL4060580)
Affinity DataEC50:  7.90E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242769(CHEMBL4082468)
Affinity DataEC50:  5.00E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242770(CHEMBL4071981)
Affinity DataEC50:  1.60E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242772(CHEMBL4091218)
Affinity DataEC50:  200nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242781(CHEMBL4083428)
Affinity DataEC50:  40nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242782(CHEMBL4101417)
Affinity DataEC50:  31nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242783(CHEMBL4072997)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242784(CHEMBL4090191)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242785(CHEMBL4069128)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242786(CHEMBL4082347)
Affinity DataEC50:  1.00E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242792(CHEMBL4071846)
Affinity DataEC50:  4.00E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242793(CHEMBL4098841)
Affinity DataEC50:  630nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242794(CHEMBL4091097)
Affinity DataEC50:  1.20E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242795(CHEMBL4098957)
Affinity DataEC50:  1.20E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242796(CHEMBL4063355)
Affinity DataEC50:  790nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242797(CHEMBL4093697)
Affinity DataEC50:  500nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242798(CHEMBL4060445)
Affinity DataEC50:  2.00E+3nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242814(CHEMBL4063218)
Affinity DataEC50:  630nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242815(CHEMBL4062882)
Affinity DataEC50:  100nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetHexokinase-4(Human)
Takeda California

Curated by ChEMBL
LigandPNGBDBM50242816(CHEMBL4093271)
Affinity DataEC50:  120nMAssay Description:Activation of full length human C-terminal FLAG-tagged glucokinase (12 to 465 residues) expressed in Escherichia coli DH10b using glucose as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467131(CHEMBL4288964)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508101(CHEMBL4521388)
Affinity DataEC50:  1.66E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508102(CHEMBL4537335)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508103(CHEMBL4589453)
Affinity DataEC50:  2.25E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508104(CHEMBL4591405)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508105(CHEMBL4542891)
Affinity DataEC50:  730nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508106(CHEMBL4517263)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508107(CHEMBL4574542)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508108(CHEMBL4567211)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508109(CHEMBL4592935)
Affinity DataEC50:  1.03E+4nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508110(CHEMBL4444760)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508111(CHEMBL4520827)
Affinity DataEC50:  460nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508113(CHEMBL4453360)
Affinity DataEC50:  2.72E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508114(CHEMBL4466241)
Affinity DataEC50:  1.32E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508115(CHEMBL4469751)
Affinity DataEC50:  1.81E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508116(CHEMBL4535401)
Affinity DataEC50:  2.78E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508117(CHEMBL4463602)
Affinity DataEC50:  2.53E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508118(CHEMBL4436393)
Affinity DataEC50:  7.36E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508119(CHEMBL4472191)
Affinity DataEC50:  1.23E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508120(CHEMBL4531918)
Affinity DataEC50:  2.62E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508121(CHEMBL4527893)
Affinity DataEC50:  2.36E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508122(CHEMBL4456647)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
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