Report error Found 1335 with Last Name = 'li' and Initial = 'hy'
TargetPeroxisome proliferator-activated receptor alpha(Human)
The University of Sydney
Curated by ChEMBL
The University of Sydney
Curated by ChEMBL
Affinity DataEC50: 2.46E+4nMAssay Description:Agonist activity at human PPARalpha assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
The University of Sydney
Curated by ChEMBL
The University of Sydney
Curated by ChEMBL
Affinity DataEC50: 2.23E+4nMAssay Description:Agonist activity at human PPARgamma assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
The University of Sydney
Curated by ChEMBL
The University of Sydney
Curated by ChEMBL
Affinity DataEC50: 1.89E+4nMAssay Description:Agonist activity at human PPARgamma assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
The University of Sydney
Curated by ChEMBL
The University of Sydney
Curated by ChEMBL
Affinity DataEC50: 3.31E+4nMAssay Description:Agonist activity at human PPARalpha assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
The University of Sydney
Curated by ChEMBL
The University of Sydney
Curated by ChEMBL
Affinity DataEC50: 2.31E+4nMAssay Description:Agonist activity at human PPARalpha assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
The University of Sydney
Curated by ChEMBL
The University of Sydney
Curated by ChEMBL
Affinity DataEC50: 1.54E+4nMAssay Description:Agonist activity at human PPARgamma assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
The University of Sydney
Curated by ChEMBL
The University of Sydney
Curated by ChEMBL
Affinity DataEC50: 8.90E+3nMAssay Description:Agonist activity at human PPARalpha assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
The University of Sydney
Curated by ChEMBL
The University of Sydney
Curated by ChEMBL
Affinity DataEC50: 2.69E+4nMAssay Description:Agonist activity at human PPARgamma assessed as induction of transactivation activity by cell based assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.66E+4nMAssay Description:Binding affinity to SARS-CoV-2 3CL protease at 1.875 to 50 uM by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.43E+4nMAssay Description:Binding affinity to SARS-CoV-2 3CL protease at 1.875 to 50 uM by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 3.13E+4nMAssay Description:Binding affinity to SARS-CoV-2 3CL protease at 1.875 to 50 uM by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+4nMAssay Description:Binding affinity to SARS-CoV-2 3CL protease at 1.875 to 50 uM in presence of wallichins D by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+4nMAssay Description:Binding affinity to SARS-CoV-2 3CL protease at 1.875 to 50 uM in presence of wallichins C by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 9.17E+4nMAssay Description:Binding affinity to SARS-CoV-2 Spike glycoprotein receptor-binding domain at 1.875 to 50 uM by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 6.79E+4nMAssay Description:Binding affinity to SARS-CoV-2 Spike glycoprotein receptor-binding domain at 1.875 to 50 uM by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 6.47E+4nMAssay Description:Binding affinity to SARS-CoV-2 Spike glycoprotein receptor-binding domain at 1.875 to 50 uM in presence of wallichins D by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 6.47E+4nMAssay Description:Binding affinity to SARS-CoV-2 Spike glycoprotein receptor-binding domain at 1.875 to 50 uM in presence of wallichins C by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 6.62E+3nMAssay Description:Binding affinity to biotinylated ALKBH5 (66 to 292 residues)(unknown origin) expressed in Escherichia coli BL21(DE3) assessed as equilibrium dissocia...More data for this Ligand-Target Pair
Affinity DataKd: 1.12E+4nMAssay Description:Binding affinity to NT-647-NHS fluorescent dye-labeled wild-type ALKBH5 (66 to 292 residues)(unknown origin) expressed in Escherichia coli BL21(DE3) ...More data for this Ligand-Target Pair
Affinity DataKd: 3.73E+5nMAssay Description:Binding affinity to NT-647-NHS fluorescent dye-labeled ALKBH5 R130A mutant (unknown origin) expressed in Escherichia coli BL21(DE3) using m6A-ssDNA a...More data for this Ligand-Target Pair
Affinity DataKd: 5.30E+4nMAssay Description:Binding affinity to NT-647-NHS fluorescent dye-labeled ALKBH5 K132A mutant (unknown origin) expressed in Escherichia coli BL21(DE3) using m6A-ssDNA a...More data for this Ligand-Target Pair
Affinity DataKd: 2.90E+5nMAssay Description:Binding affinity to NT-647-NHS fluorescent dye-labeled ALKBH5 Y139A mutant (unknown origin) expressed in Escherichia coli BL21(DE3) using m6A-ssDNA a...More data for this Ligand-Target Pair
Affinity DataKd: 1.58E+4nMAssay Description:Binding affinity to NT-647-NHS fluorescent dye-labeled ALKBH5 Y139A/R277A mutant (unknown origin) expressed in Escherichia coli BL21(DE3) using m6A-s...More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.0200nMAssay Description:Inhibition of human c-KIT A loop exon 17 D820Y single mutant using poly (Glu,Tyr) 4:1 as substrate in presence of 33P-gamma-ATP by hotspot kinase ass...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of wild type FLT3 (unknown origin) expressed in HEK293T cells assessed as decrease in FLT3 phosphorylation at 0.1 to 1000 nM after 1 hr by...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of wild type FLT3 D835Y mutant (unknown origin) expressed in HEK293T cells assessed as decrease in FLT3 D835Y phosphorylation at 0.1 to 10...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of wild type FLT3 ITD mutant (unknown origin) expressed in HEK293T cells assessed as decrease in FLT3 ITD phosphorylation at 0.1 to 1000 n...More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.120nMAssay Description:Inhibition of human c-KIT A loop exon 17 Y823D single mutant using poly (Glu,Tyr) 4:1 as substrate in presence of 33P-gamma-ATP by hotspot kinase ass...More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.180nMAssay Description:Inhibition of human c-KIT A loop exon 11/17 V560G/N822K double mutant using poly (Glu,Tyr) 4:1 as substrate in presence of 33P-gamma-ATP by hotspot k...More data for this Ligand-Target Pair
Affinity DataIC50: 0.316nMAssay Description:Inhibition of recombinant human full-length His-tagged Aurora B expressed in baculovirus expression system using 5-FAM-LRRASLG-CONH2 as substrate pre...More data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Inhibition of human TGFbeta receptor 1 in human HEK293 cells preincubated for 24 hrs followed by addition of TGFbeta1 and measured after 24 hrs by lu...More data for this Ligand-Target Pair
Affinity DataIC50: 0.326nMAssay Description:Inhibition of recombinant human full-length His-tagged Aurora B expressed in baculovirus expression system using 5-FAM-LRRASLG-CONH2 as substrate pre...More data for this Ligand-Target Pair
Affinity DataIC50: 0.336nMAssay Description:Inhibition of recombinant human full-length His-tagged Aurora B expressed in baculovirus expression system using 5-FAM-LRRASLG-CONH2 as substrate pre...More data for this Ligand-Target Pair
Affinity DataIC50: 0.340nMAssay Description:Inhibition of human TGFbeta receptor 1 in human HEK293 cells preincubated for 24 hrs followed by addition of TGFbeta1 and measured after 24 hrs by lu...More data for this Ligand-Target Pair
Affinity DataIC50: 0.350nMAssay Description:Inhibition of human TGFbeta receptor 1 in human HEK293 cells preincubated for 24 hrs followed by addition of TGFbeta1 and measured after 24 hrs by lu...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Human)
University of Arkansas For Medical Sciences
Curated by ChEMBL
University of Arkansas For Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of TRKA G595R mutant (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Human)
University of Arkansas For Medical Sciences
Curated by ChEMBL
University of Arkansas For Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of BTK (unknown origin) after 60 mins by FRET assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Human)
University of Arkansas For Medical Sciences
Curated by ChEMBL
University of Arkansas For Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Irreversible inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.510nMAssay Description:Inhibition of human TGFbeta receptor 1 in human HEK293 cells preincubated for 24 hrs followed by addition of TGFbeta1 and measured after 24 hrs by lu...More data for this Ligand-Target Pair
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human TGFbeta receptor 1 in human HEK293 cells preincubated for 24 hrs followed by addition of TGFbeta1 and measured after 24 hrs by lu...More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Aurora A (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.620nMAssay Description:Inhibition of human TGFbeta receptor 1 in human HEK293 cells preincubated for 24 hrs followed by addition of TGFbeta1 and measured after 24 hrs by lu...More data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Inhibition of human TGFbeta receptor 1 in human HEK293 cells preincubated for 24 hrs followed by addition of TGFbeta1 and measured after 24 hrs by lu...More data for this Ligand-Target Pair
Affinity DataIC50: 0.650nMAssay Description:Inhibition of human TGFbeta receptor 1 in human HEK293 cells preincubated for 24 hrs followed by addition of TGFbeta1 and measured after 24 hrs by lu...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataIC50: 0.670nMAssay Description:Inhibition of RET isoform 9 M918T mutant in human MZ-CRC-1 cells assessed as reduction in cell proliferation supplemented with fresh medium containin...More data for this Ligand-Target Pair
TargetCoiled-coil domain-containing protein 6(Human)
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataIC50: 0.670nMAssay Description:Inhibition of CCDC6/RET in human TPC1 cells assessed as reduction in cell proliferation supplemented with fresh medium containing compound for every ...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataIC50: 0.670nMAssay Description:Inhibition of RET isoform 9 C634W mutant in human TT cells assessed as reduction in cell proliferation supplemented with fresh medium containing comp...More data for this Ligand-Target Pair
TargetCoiled-coil domain-containing protein 6(Human)
University of Naples Federico II
Curated by ChEMBL
University of Naples Federico II
Curated by ChEMBL
Affinity DataIC50: 0.670nMAssay Description:Inhibition of CCDC6/RET in human LC2/ad cells assessed as reduction in cell proliferation supplemented with fresh medium containing compound for ever...More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Human)
National Health Research Institutes
Curated by ChEMBL
National Health Research Institutes
Curated by ChEMBL
Affinity DataIC50: 0.670nMAssay Description:Inhibition of human c-KIT A loop exon 17 D816H single mutant using poly (Glu,Tyr) 4:1 as substrate in presence of 33P-gamma-ATP by hotspot kinase ass...More data for this Ligand-Target Pair
Affinity DataIC50: 0.670nMAssay Description:Inhibition of human TGFbeta receptor 1 in human HEK293 cells preincubated for 24 hrs followed by addition of TGFbeta1 and measured after 24 hrs by lu...More data for this Ligand-Target Pair
