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TargetPeptidyl-prolyl cis-trans isomerase A(Human)
East China Univesity of Science and Technology

LigandPNGBDBM93251(CypA Inhibitor, 1a)
Affinity DataKd:  2.43E+4nMpH: 7.4 T: 2°CAssay Description:CypA in vitro were determined by employing surface plasmon resonance (SPR) technology. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
East China Univesity of Science and Technology

LigandPNGBDBM93252(CypA Inhibitor, 1b)
Affinity DataKd:  3.07E+3nMpH: 7.4 T: 2°CAssay Description:CypA in vitro were determined by employing surface plasmon resonance (SPR) technology. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
East China Univesity of Science and Technology

LigandPNGBDBM93253(CypA Inhibitor, 1c)
Affinity DataKd:  212nMpH: 7.4 T: 2°CAssay Description:CypA in vitro were determined by employing surface plasmon resonance (SPR) technology. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
East China Univesity of Science and Technology

LigandPNGBDBM93254(CypA Inhibitor, 1d)
Affinity DataKd:  1.72E+4nMpH: 7.4 T: 2°CAssay Description:CypA in vitro were determined by employing surface plasmon resonance (SPR) technology. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
East China Univesity of Science and Technology

LigandPNGBDBM93255(CypA Inhibitor, 1e)
Affinity DataKd:  3.41E+3nMpH: 7.4 T: 2°CAssay Description:CypA in vitro were determined by employing surface plasmon resonance (SPR) technology. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
East China Univesity of Science and Technology

LigandPNGBDBM93256(CypA Inhibitor, 2a)
Affinity DataKd:  76.2nMpH: 7.4 T: 2°CAssay Description:CypA in vitro were determined by employing surface plasmon resonance (SPR) technology. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
East China Univesity of Science and Technology

LigandPNGBDBM93257(CypA Inhibitor, 2b)
Affinity DataKd:  2.88E+4nMpH: 7.4 T: 2°CAssay Description:CypA in vitro were determined by employing surface plasmon resonance (SPR) technology. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
East China Univesity of Science and Technology

LigandPNGBDBM93258(CypA Inhibitor, 3a)
Affinity DataKd:  8.18E+3nMpH: 7.4 T: 2°CAssay Description:CypA in vitro were determined by employing surface plasmon resonance (SPR) technology. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
East China Univesity of Science and Technology

LigandPNGBDBM93259(CypA Inhibitor, 3b)
Affinity DataKd:  1.08E+4nMpH: 7.4 T: 2°CAssay Description:CypA in vitro were determined by employing surface plasmon resonance (SPR) technology. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
East China Univesity of Science and Technology

LigandPNGBDBM93261(CypA Inhibitor, 4b)
Affinity DataKd:  2.73E+4nMpH: 7.4 T: 2°CAssay Description:CypA in vitro were determined by employing surface plasmon resonance (SPR) technology. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
East China Univesity of Science and Technology

LigandPNGBDBM93263(CypA Inhibitor, 4d)
Affinity DataKd:  3.08E+4nMpH: 7.4 T: 2°CAssay Description:CypA in vitro were determined by employing surface plasmon resonance (SPR) technology. More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2013
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50247360(CHEMBL4095787)
Affinity DataEC50:  5.20E+3nMAssay Description:Binding affinity to beta galactosidase fused human PRMT3 (211 to 531 residues) expressed in human HEK293 cells after 6 hrs by InCELL hunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2019
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50247361(CHEMBL4077534)
Affinity DataEC50:  2.70E+3nMAssay Description:Binding affinity to beta galactosidase fused human PRMT3 (211 to 531 residues) expressed in human HEK293 cells after 6 hrs by InCELL hunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2019
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50247349(CHEMBL4072005)
Affinity DataEC50:  1.80E+3nMAssay Description:Binding affinity to beta galactosidase fused human PRMT3 (211 to 531 residues) expressed in human HEK293 cells after 6 hrs by InCELL hunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein arginine N-methyltransferase 3(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50247360(CHEMBL4095787)
Affinity DataEC50:  4.90E+3nMAssay Description:Binding affinity to beta galactosidase fused human PRMT3 (211 to 531 residues) expressed in human A549 cells after 6 hrs by InCELL hunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2019
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50247361(CHEMBL4077534)
Affinity DataEC50:  1.60E+3nMAssay Description:Binding affinity to beta galactosidase fused human PRMT3 (211 to 531 residues) expressed in human A549 cells after 6 hrs by InCELL hunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2019
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50247349(CHEMBL4072005)
Affinity DataEC50:  2.00E+3nMAssay Description:Binding affinity to beta galactosidase fused human PRMT3 (211 to 531 residues) expressed in human A549 cells after 6 hrs by InCELL hunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein arginine N-methyltransferase 3(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50247359(CHEMBL4062783)
Affinity DataEC50:  3.10E+3nMAssay Description:Binding affinity to beta galactosidase fused human PRMT3 (211 to 531 residues) expressed in human HEK293 cells after 6 hrs by InCELL hunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2019
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 3(Human)
Icahn School of Medicine At Mount Sinai

Curated by ChEMBL
LigandPNGBDBM50247359(CHEMBL4062783)
Affinity DataEC50:  2.70E+3nMAssay Description:Binding affinity to beta galactosidase fused human PRMT3 (211 to 531 residues) expressed in human A549 cells after 6 hrs by InCELL hunter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2019
Entry Details Article
PubMed
TargetUbiquitin-conjugating enzyme E2 D3(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50249751(CHEMBL4080789)
Affinity DataKd:  283nMAssay Description:Binding affinity to human recombinant UbcH5c by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2019
Entry Details Article
PubMed
TargetUbiquitin-conjugating enzyme E2 D3(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50249752(CHEMBL4098033)
Affinity DataKd:  6.40E+3nMAssay Description:Binding affinity to human recombinant UbcH5c by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2019
Entry Details Article
PubMed
TargetUbiquitin-conjugating enzyme E2 D3(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50249753(CHEMBL4082171)
Affinity DataKd:  2.58E+3nMAssay Description:Binding affinity to human recombinant UbcH5c by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2019
Entry Details Article
PubMed
TargetUbiquitin-conjugating enzyme E2 D3(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50249760(CHEMBL4100955)
Affinity DataKd:  3.64E+3nMAssay Description:Binding affinity to human recombinant UbcH5c by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2019
Entry Details Article
PubMed
TargetUbiquitin-conjugating enzyme E2 D3(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50249761(CHEMBL4071335)
Affinity DataKd:  353nMAssay Description:Binding affinity to human recombinant UbcH5c by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2019
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50260041(CHEMBL4097012)
Affinity DataKd:  2.20nMAssay Description:Binding affinity to human DNA-tagged DDR1 expressed in bacterial expression system measured after 1 hr by quantitative PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2020
Entry Details Article
PubMed
TargetDual specificity mitogen-activated protein kinase kinase 5(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50268010(CHEMBL4098896)
Affinity DataKd:  88nMAssay Description:Binding affinity to partial length human MEK5 expressed in HEK293 cells by active-site-dependent competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase SIK1(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50268010(CHEMBL4098896)
Affinity DataKd:  45nMAssay Description:Binding affinity to partial length human SIK expressed in Escherichia coli BL21 by active-site-dependent competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetTyrosine-protein kinase Srms(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50268010(CHEMBL4098896)
Affinity DataKd:  64nMAssay Description:Binding affinity to partial length human SRMS expressed in HEK293 cells by active-site-dependent competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50268010(CHEMBL4098896)
Affinity DataKd:  460nMAssay Description:Binding affinity to partial length human KIT expressed in Escherichia coli BL21 by active-site-dependent competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetTyrosine-protein kinase FRK(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50268010(CHEMBL4098896)
Affinity DataKd:  22nMAssay Description:Binding affinity to partial length human FRK expressed in Escherichia coli BL21 by active-site-dependent competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 20(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50268010(CHEMBL4098896)
Affinity DataKd:  2.70nMAssay Description:Binding affinity to partial length human ZAK expressed in Escherichia coli BL21 by active-site-dependent competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetAurora kinase B(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50268010(CHEMBL4098896)
Affinity DataKd:  64nMAssay Description:Binding affinity to partial length human AURKB expressed in HEK293 cells by active-site-dependent competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50368452(CHEMBL4168305)
Affinity DataKd:  370nMAssay Description:Binding affinity to human TIE2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetEphrin type-A receptor 2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50368452(CHEMBL4168305)
Affinity DataKd:  260nMAssay Description:Binding affinity to human EPHA2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50368452(CHEMBL4168305)
Affinity DataKd:  180nMAssay Description:Binding affinity to human LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetNT-3 growth factor receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50368452(CHEMBL4168305)
Affinity DataKd:  9.30nMAssay Description:Binding affinity to human TrkCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50368452(CHEMBL4168305)
Affinity DataKd:  7.90nMAssay Description:Binding affinity to human DDR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDiscoidin domain-containing receptor 2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50368452(CHEMBL4168305)
Affinity DataKd:  8nMAssay Description:Binding affinity to human DDR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetEphrin type-A receptor 7(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50368452(CHEMBL4168305)
Affinity DataKd:  200nMAssay Description:Binding affinity to human EPHA7More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetEphrin type-A receptor 8(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50368452(CHEMBL4168305)
Affinity DataKd:  79nMAssay Description:Binding affinity to human EPHA8More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetEphrin type-B receptor 2(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50368452(CHEMBL4168305)
Affinity DataKd:  260nMAssay Description:Binding affinity to human EPHB2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 10(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50368452(CHEMBL4168305)
Affinity DataKd:  10nMAssay Description:Binding affinity to human LOKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetHigh affinity nerve growth factor receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50368452(CHEMBL4168305)
Affinity DataKd:  100nMAssay Description:Binding affinity to human TrkAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetBDNF/NT-3 growth factors receptor(Human)
Jinan University

Curated by ChEMBL
LigandPNGBDBM50368452(CHEMBL4168305)
Affinity DataKd:  11nMAssay Description:Binding affinity to human TrkBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50461568(CHEMBL4225198)
Affinity DataKd:  9.40E+3nMAssay Description:Binding affinity to VBC complex (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50461569(CHEMBL4228750)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to VBC complex (unknown origin) assessed as reduction of FAM-labelled HIF1alpha peptide binding by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50461570(CHEMBL4224723)
Affinity DataKd: >1.30E+4nMAssay Description:Binding affinity to VBC complex (unknown origin) assessed as reduction of FAM-labelled HIF1alpha peptide binding by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50459942(CHEMBL4227864 | US10730870, Example 85 | US1151208...)
Affinity DataKd:  440nMAssay Description:Binding affinity to VBC complex (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50461570(CHEMBL4224723)
Affinity DataKd:  2.16E+4nMAssay Description:Binding affinity to VBC complex (unknown origin) by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetElongin-C(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM50459942(CHEMBL4227864 | US10730870, Example 85 | US1151208...)
Affinity DataKd:  690nMAssay Description:Binding affinity to VBC complex (unknown origin) assessed as reduction of FAM-labelled HIF1alpha peptide binding by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
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