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TargetApoptosis regulator Bcl-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50162774(ABT-199 | US11420968, Example ABT-199 | Venetoclax)
Affinity DataKi: <0.0100nMAssay Description:Inhibition of Bcl2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50162797(CHEMBL3793424)
Affinity DataKi: <0.0100nMAssay Description:Inhibition of Bcl-xL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50514200(CHEMBL4446378 | US10703733, Comparative Example 1)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of human Biotin-DMRPEIWIAQELRRIGDEFNAYYARR peptide binding to 6XHis-tagged human MCl-1 (171 to 327 residues) expressed in Escherichia coli...More data for this Ligand-Target Pair
LigandPNGBDBM333146(Compound I | US10196404, Example 1 | US10196404, E...)
Affinity DataKi:  0.170nMAssay Description:Inhibition of N-terminal GST-tagged MCl-1 (unknown origin) expressed in Escherichia coli cells after 120 to 180 mins by TR-FRET-binding affinity assa...More data for this Ligand-Target Pair
LigandPNGBDBM50519614(CHEMBL4439276)
Affinity DataKi:  0.190nMAssay Description:Inhibition of MCl-1 (unknown origin)More data for this Ligand-Target Pair
LigandPNGBDBM50078163(CHEMBL3417704)
Affinity DataKi:  0.450nMAssay Description:Inhibition of GST-tagged MCl-1 (unknown origin) after 60 mins by TR-FRET-binding affinity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50270877((R)-4-(4-((2-(4-chlorophenyl)-5,5-dimethylcyclohex...)
Affinity DataKi: <0.5nMAssay Description:Inhibition of Flu-Bax peptide binding to Bcl-xL (unknown origin) by time-resolved fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
TargetBcl-2-like protein 1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50394837(CHEMBL343002 | HOE-33342)
Affinity DataKi:  0.900nMAssay Description:Inhibition of FAM-GQVGRQLAIIGDDINR peptide binding to human Bcl-xL after 15 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50270877((R)-4-(4-((2-(4-chlorophenyl)-5,5-dimethylcyclohex...)
Affinity DataKi: <1nMAssay Description:Inhibition of Flu-Bax peptide binding to Bcl2 (unknown origin) by time-resolved fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50266959(CHEMBL4085804)
Affinity DataKi: <1nMAssay Description:Inhibition of Bcl-xL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50266959(CHEMBL4085804)
Affinity DataKi: <1nMAssay Description:Inhibition of Bcl2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50270877((R)-4-(4-((2-(4-chlorophenyl)-5,5-dimethylcyclohex...)
Affinity DataKi: <1nMAssay Description:Inhibition of Flu-Bax peptide binding to MCl-1 (unknown origin) by time-resolved fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50030764(CHEMBL3342187)
Affinity DataKi:  1.10nMAssay Description:Inhibition of Bcl-xL (unknown origin)More data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227831(CHEMBL52242)
Affinity DataKi:  1.20nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM177786(US9120791, Example 1 | US9120791, Example 38 | US9...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of Bcl2 (unknown origin) after 2 hrs by fluorescein-PUMA based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227791(CHEMBL53815)
Affinity DataKi:  4.60nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227978(CHEMBL53316)
Affinity DataKi:  6.30nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50228190(CHEMBL54263)
Affinity DataKi:  9.80nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50266967(CHEBI:66678 | CHEMBL3393621)
Affinity DataKi:  10nMAssay Description:Inhibition of MCl-1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227787(CHEMBL1743933)
Affinity DataKi:  13nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227837(CHEMBL52131)
Affinity DataKi:  14nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50093789(CHEMBL541829 | Succinic acid mono-(2-dimethylamino...)
Affinity DataKi:  18nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227788(CHEMBL1743936)
Affinity DataKi:  23nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50330247(6,6',7,7'-Tetrahydroxy-5,5'-diisopropyl-3,3'-dimet...)
Affinity DataKi:  25nMAssay Description:Inhibition of Flu-BakBH3 peptide binding to recombinant human MCL1 after 15 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50330250(5,5'-Dibenzyl-6,6',7,7'-tetrahydroxy-3,3'-dimethyl...)
Affinity DataKi:  25nMAssay Description:Inhibition of MCl-1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227974(CHEMBL298554)
Affinity DataKi:  26nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50330250(5,5'-Dibenzyl-6,6',7,7'-tetrahydroxy-3,3'-dimethyl...)
Affinity DataKi:  31nMAssay Description:Inhibition of Bcl2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50330247(6,6',7,7'-Tetrahydroxy-5,5'-diisopropyl-3,3'-dimet...)
Affinity DataKi:  35nMAssay Description:Inhibition of Flu-BakBH3 peptide binding to recombinant human Bcl2 after 15 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227976(CHEMBL299389)
Affinity DataKi:  38nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227653(CHEMBL299207)
Affinity DataKi:  41nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50525271(CHEMBL4519497)
Affinity DataKi:  58nMAssay Description:Inhibition of MCl-1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227977(CHEMBL300631)
Affinity DataKi:  68nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227790(CHEMBL53344)
Affinity DataKi:  71nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227789(CHEMBL412653)
Affinity DataKi:  75nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50330250(5,5'-Dibenzyl-6,6',7,7'-tetrahydroxy-3,3'-dimethyl...)
Affinity DataKi:  76nMAssay Description:Inhibition of Bcl-xL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50330250(5,5'-Dibenzyl-6,6',7,7'-tetrahydroxy-3,3'-dimethyl...)
Affinity DataKi:  122nMAssay Description:Inhibition of adenosine receptor A1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50266958(CHEMBL4077940)
Affinity DataKi:  179nMAssay Description:Inhibition of FITC-Ahx-GQVGRQLAIIGDDINR-CONH2 peptide binding to Bcl2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataKi:  180nMAssay Description:Inhibition of MCl-1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM174838(US9115061, I)
Affinity DataKi:  190nMAssay Description:Inhibition of Flu-BakBH3 peptide binding to GST-tagged Bcl-xL (unknown origin) preincubated for 10 mins followed by substrate addition measured after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50227832(CHEMBL54101)
Affinity DataKi:  198nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM21447(4-(4-{[2-(4-chlorophenyl)phenyl]methyl}piperazin-1...)
Affinity DataKi:  283nMAssay Description:Inhibition of Bcl2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM21447(4-(4-{[2-(4-chlorophenyl)phenyl]methyl}piperazin-1...)
Affinity DataKi:  284nMAssay Description:Inhibition of Bcl-xL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM21447(4-(4-{[2-(4-chlorophenyl)phenyl]methyl}piperazin-1...)
Affinity DataKi:  285nMAssay Description:Inhibition of Bcl-w (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM50525271(CHEMBL4519497)
Affinity DataKi:  310nMAssay Description:Inhibition of Bcl2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataKi:  320nMAssay Description:Inhibition of Bcl2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM174838(US9115061, I)
Affinity DataKi:  360nMAssay Description:Inhibition of Flu-BakBH3 peptide binding to GST-tagged Bcl2 (unknown origin) after 2 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50228189(CHEMBL52710)
Affinity DataKi:  416nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBcl-2-like protein 1(Human)
Tsinghua University

Curated by ChEMBL
LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataKi:  480nMAssay Description:Inhibition of Bcl-xL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM53290(2-[4-[(4-bromophenyl)sulfonylamino]-1-hydroxynapht...)
Affinity DataKi:  490nMAssay Description:Inhibition of human MCl-1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Mitsubishi Kasei

Curated by ChEMBL
LigandPNGBDBM50228052(CHEMBL52982)
Affinity DataKi:  517nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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