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Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataEC50:  1.5nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144838((S)-2-(5-Fluoro-6-iodo-2,3-dihydro-indol-1-yl)-1-m...)
Affinity DataEC50:  22nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144844((S)-1-Methyl-2-(2,3,8,9-tetrahydro-7H-pyrano[2,3-g...)
Affinity DataEC50:  36nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144842((S)-1-Methyl-2-(2,3,7,8-tetrahydro-furo[2,3-g]indo...)
Affinity DataEC50:  3nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144843((S)-2-(5-Fluoro-6-trifluoromethyl-2,3-dihydro-indo...)
Affinity DataEC50:  49nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144839((S)-2-(6-Ethylsulfanyl-5-fluoro-2,3-dihydro-indol-...)
Affinity DataEC50:  31nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144845((S)-2-(6-Chloro-5-fluoro-2,3-dihydro-indol-1-yl)-1...)
Affinity DataEC50:  7.30nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144845((S)-2-(6-Chloro-5-fluoro-2,3-dihydro-indol-1-yl)-1...)
Affinity DataEC50:  31nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144845((S)-2-(6-Chloro-5-fluoro-2,3-dihydro-indol-1-yl)-1...)
Affinity DataEC50:  367nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144838((S)-2-(5-Fluoro-6-iodo-2,3-dihydro-indol-1-yl)-1-m...)
Affinity DataEC50:  64nMAssay Description:Functional activity against human 5-hydroxytryptamine 2C receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144835((S)-1-Methyl-2-(6-methylsulfanyl-2,3-dihydro-indol...)
Affinity DataEC50:  10nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataEC50:  131nMAssay Description:Affinity for human 5-hydroxytryptamine 2A receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144846(VER-5593 | (S)-2-(5-Fluoro-6-methylsulfanyl-2,3-di...)
Affinity DataEC50:  76nMAssay Description:Affinity for human 5-hydroxytryptamine 2A receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144837((S)-2-(6-Chloro-2,3-dihydro-indol-1-yl)-1-methyl-e...)
Affinity DataEC50:  602nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144837((S)-2-(6-Chloro-2,3-dihydro-indol-1-yl)-1-methyl-e...)
Affinity DataEC50:  6.5nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144844((S)-1-Methyl-2-(2,3,8,9-tetrahydro-7H-pyrano[2,3-g...)
Affinity DataEC50:  28nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144835((S)-1-Methyl-2-(6-methylsulfanyl-2,3-dihydro-indol...)
Affinity DataEC50:  164nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144843((S)-2-(5-Fluoro-6-trifluoromethyl-2,3-dihydro-indo...)
Affinity DataEC50:  130nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144839((S)-2-(6-Ethylsulfanyl-5-fluoro-2,3-dihydro-indol-...)
Affinity DataEC50:  21nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataEC50:  18nMAssay Description:Functional activity against human 5-hydroxytryptamine 2C receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataEC50:  1.70nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144838((S)-2-(5-Fluoro-6-iodo-2,3-dihydro-indol-1-yl)-1-m...)
Affinity DataEC50:  432nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144842((S)-1-Methyl-2-(2,3,7,8-tetrahydro-furo[2,3-g]indo...)
Affinity DataEC50:  4.5nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144842((S)-1-Methyl-2-(2,3,7,8-tetrahydro-furo[2,3-g]indo...)
Affinity DataEC50:  62nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144836((S)-2-(6-Ethylsulfanyl-2,3-dihydro-indol-1-yl)-1-m...)
Affinity DataEC50:  40nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144846(VER-5593 | (S)-2-(5-Fluoro-6-methylsulfanyl-2,3-di...)
Affinity DataEC50:  4.10nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144840(CHEMBL309760 | (S)-2-(6-Bromo-2,3-dihydro-indol-1-...)
Affinity DataEC50:  719nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataEC50:  11nMAssay Description:Affinity for human 5-hydroxytryptamine 2A receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144840(CHEMBL309760 | (S)-2-(6-Bromo-2,3-dihydro-indol-1-...)
Affinity DataEC50:  11nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50001915(mCPP | 1-(3-chlorophenyl)piperazine | CHEMBL478 | ...)
Affinity DataEC50: >1.00E+3nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144844((S)-1-Methyl-2-(2,3,8,9-tetrahydro-7H-pyrano[2,3-g...)
Affinity DataEC50:  125nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144836((S)-2-(6-Ethylsulfanyl-2,3-dihydro-indol-1-yl)-1-m...)
Affinity DataEC50:  378nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144843((S)-2-(5-Fluoro-6-trifluoromethyl-2,3-dihydro-indo...)
Affinity DataEC50:  1.06E+3nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50001915(mCPP | 1-(3-chlorophenyl)piperazine | CHEMBL478 | ...)
Affinity DataEC50:  75nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144839((S)-2-(6-Ethylsulfanyl-5-fluoro-2,3-dihydro-indol-...)
Affinity DataEC50:  181nMAssay Description:Functional activity against human 5-hydroxytryptamine 2A receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144836((S)-2-(6-Ethylsulfanyl-2,3-dihydro-indol-1-yl)-1-m...)
Affinity DataEC50:  72nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144846(VER-5593 | (S)-2-(5-Fluoro-6-methylsulfanyl-2,3-di...)
Affinity DataEC50:  6.70nMAssay Description:Functional activity against human 5-hydroxytryptamine 2C receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144837((S)-2-(6-Chloro-2,3-dihydro-indol-1-yl)-1-methyl-e...)
Affinity DataEC50:  44nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144840(CHEMBL309760 | (S)-2-(6-Bromo-2,3-dihydro-indol-1-...)
Affinity DataEC50:  44nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50001915(mCPP | 1-(3-chlorophenyl)piperazine | CHEMBL478 | ...)
Affinity DataEC50:  26nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144841((S)-1-(6-chloro-5-fluoro-1H-indol-1-yl)propan-2-am...)
Affinity DataEC50:  4.30nMAssay Description:Functional activity against human 5-hydroxytryptamine 2B receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50144835((S)-1-Methyl-2-(6-methylsulfanyl-2,3-dihydro-indol...)
Affinity DataEC50:  26nMAssay Description:Functional activity against human 5-hydroxytryptamine 2C receptor expressed in CHO cells using fluorometric imaging plate readerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50179073((4R,9aR)-6-Cyclopropylmethoxymethyl-4-methyl-1,2,3...)
Affinity DataEC50:  15nMAssay Description:Efficacy against human recombinant 5HT2C receptor induced intracellular calcium mobilization in CHO cells by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Vernalis Research

Curated by ChEMBL
LigandPNGBDBM50179073((4R,9aR)-6-Cyclopropylmethoxymethyl-4-methyl-1,2,3...)
Affinity DataEC50:  23nMAssay Description:Efficacy against human recombinant 5HT2B receptor induced intracellular calcium mobilization in CHO cells by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296144(2-(7,7-dimethyl-2-p-tolyl-7,8-dihydro-5H-pyrano[4,...)
Affinity DataEC50:  1.20E+3nMAssay Description:Inverse agonist activity at human CB1 receptor by [35S]GTPgammaS incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296146(ethyl 4-(3-(2-chlorophenyl)-1-(2,4-dimethylphenyl)...)
Affinity DataEC50:  200nMAssay Description:Inverse agonist activity at human CB1 receptor by [35S]GTPgammaS incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296147(3-tert-butyl-1-isopropyl-1-(2-(4-(4-methoxyphenyl)...)
Affinity DataEC50:  1.50E+3nMAssay Description:Inverse agonist activity at human CB1 receptor by [35S]GTPgammaS incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50230538(N-benzyl-5-(3,5-dimethylpiperidin-1-ylsulfonyl)-N-...)
Affinity DataEC50:  300nMAssay Description:Inverse agonist activity at human CB1 receptor by [35S]GTPgammaS incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296142(1-(1-(4-chlorophenyl)-4-(3-methoxyphenyl)-5-(4-mor...)
Affinity DataEC50:  600nMAssay Description:Inverse agonist activity at human CB1 receptor by [35S]GTPgammaS incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50296143(4-(indolin-1-ylsulfonyl)-N-(2-phenoxyphenyl)benzam...)
Affinity DataEC50:  200nMAssay Description:Inverse agonist activity at human CB1 receptor by [35S]GTPgammaS incorporation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
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